BRPI0411450A - processo para a preparação de um composto, e, composto - Google Patents

processo para a preparação de um composto, e, composto

Info

Publication number
BRPI0411450A
BRPI0411450A BRPI0411450-7A BRPI0411450A BRPI0411450A BR PI0411450 A BRPI0411450 A BR PI0411450A BR PI0411450 A BRPI0411450 A BR PI0411450A BR PI0411450 A BRPI0411450 A BR PI0411450A
Authority
BR
Brazil
Prior art keywords
compound
preparing
oxyphenoxy
ethylthio
methylsulfonyl
Prior art date
Application number
BRPI0411450-7A
Other languages
English (en)
Portuguese (pt)
Inventor
Kjell Andersson
Eva-Lotte Lindstedt Alstermark
Henrik S Rensen
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BRPI0411450A publication Critical patent/BRPI0411450A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/18Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1896Compounds having one or more Si-O-acyl linkages
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
    • C07C319/20Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides by reactions not involving the formation of sulfide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/56Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
BRPI0411450-7A 2003-06-19 2004-06-16 processo para a preparação de um composto, e, composto BRPI0411450A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0314260.1A GB0314260D0 (en) 2003-06-19 2003-06-19 Therapeutic agents
PCT/GB2004/002599 WO2004113285A1 (en) 2003-06-19 2004-06-16 Process for the preparation of racemic 2-{[2-(4-hydroxyphenyl)ethyl]thio}-3-[4-(2-{4-[(methylsulfonyl)oxy]phenoxy}ethyl)phenyl]-propanoic acid

Publications (1)

Publication Number Publication Date
BRPI0411450A true BRPI0411450A (pt) 2006-07-18

Family

ID=27636892

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0411450-7A BRPI0411450A (pt) 2003-06-19 2004-06-16 processo para a preparação de um composto, e, composto

Country Status (14)

Country Link
US (1) US7429675B2 (OSRAM)
EP (1) EP1638929A1 (OSRAM)
JP (1) JP2006527751A (OSRAM)
KR (1) KR20060010840A (OSRAM)
CN (1) CN1835918A (OSRAM)
AU (1) AU2004249487A1 (OSRAM)
BR (1) BRPI0411450A (OSRAM)
CA (1) CA2529252A1 (OSRAM)
GB (1) GB0314260D0 (OSRAM)
IL (1) IL172376A0 (OSRAM)
MX (1) MXPA05013716A (OSRAM)
NO (1) NO20055883L (OSRAM)
WO (1) WO2004113285A1 (OSRAM)
ZA (1) ZA200509944B (OSRAM)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0104333D0 (sv) 2001-12-19 2001-12-19 Astrazeneca Ab Therapeutic agents
EP1517883B8 (en) 2002-06-20 2008-05-21 AstraZeneca AB Ortho-substituted benzoic acid derivatives for the treatment of insulin resistance
GB0314075D0 (en) * 2003-06-18 2003-07-23 Astrazeneca Ab Therapeutic agents
GB0427524D0 (en) 2004-12-16 2005-01-19 Astrazeneca Ab Chemical process
KR101558005B1 (ko) * 2007-03-08 2015-10-06 알비레오 에이비 2-치환-3-페닐프로피온산 유도체 및 염증성 장 질환 치료에서의 그의 용도
FR2986804A1 (fr) * 2012-02-09 2013-08-16 Servier Lab Procede de synthese enzymatique de l'acide (7s) 3,4-dimethoxybicyclo[4.2.0]octa-1,3,5-triene 7-carboxylique ou de ses esters, et application a la synthese de l'ivabradine et de ses sels

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0193113B1 (en) * 1985-02-25 1992-01-22 Mitsubishi Gas Chemical Company, Inc. Process for optically isomerizing optically active alpha-amino acid amides and process for producing optically active alpha-amino acids
JPS61197530A (ja) * 1985-02-25 1986-09-01 Mitsubishi Gas Chem Co Inc ラセミ化法
TW472047B (en) * 1994-02-04 2002-01-11 Merck & Co Inc Process for making HIV protease inhibitors
SE9801992D0 (sv) * 1998-06-04 1998-06-04 Astra Ab New 3-aryl-2-hydroxypropionic acid derivative I
MA26634A1 (fr) * 1998-06-04 2004-12-20 Astra Ab Nouveaux derives de l'acide 3-aryl propionique et analogues
SE0104333D0 (sv) * 2001-12-19 2001-12-19 Astrazeneca Ab Therapeutic agents

Also Published As

Publication number Publication date
EP1638929A1 (en) 2006-03-29
CN1835918A (zh) 2006-09-20
ZA200509944B (en) 2006-12-27
GB0314260D0 (en) 2003-07-23
NO20055883L (no) 2006-01-09
MXPA05013716A (es) 2006-03-08
US20060167309A1 (en) 2006-07-27
KR20060010840A (ko) 2006-02-02
JP2006527751A (ja) 2006-12-07
WO2004113285A1 (en) 2004-12-29
IL172376A0 (en) 2009-02-11
AU2004249487A1 (en) 2004-12-29
CA2529252A1 (en) 2004-12-29
US7429675B2 (en) 2008-09-30

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 5A, 6A, 7A E 8A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2159 DE 22/05/2012.