BR9706968A - Uso de antagonistas de alfa-ppar e gama-ppar para o tratamento de sindrome x - Google Patents

Uso de antagonistas de alfa-ppar e gama-ppar para o tratamento de sindrome x

Info

Publication number
BR9706968A
BR9706968A BR9706968A BR9706968A BR9706968A BR 9706968 A BR9706968 A BR 9706968A BR 9706968 A BR9706968 A BR 9706968A BR 9706968 A BR9706968 A BR 9706968A BR 9706968 A BR9706968 A BR 9706968A
Authority
BR
Brazil
Prior art keywords
ppar
syndrome
gamma
alpha
treatment
Prior art date
Application number
BR9706968A
Other languages
English (en)
Inventor
Stephen Alistair Smith
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of BR9706968A publication Critical patent/BR9706968A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4402—Non condensed pyridines; Hydrogenated derivatives thereof only substituted in position 2, e.g. pheniramine, bisacodyl
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/423—Oxazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
BR9706968A 1996-01-09 1997-01-07 Uso de antagonistas de alfa-ppar e gama-ppar para o tratamento de sindrome x BR9706968A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9600464.3A GB9600464D0 (en) 1996-01-09 1996-01-09 Novel method
PCT/EP1997/000058 WO1997025042A1 (en) 1996-01-09 1997-01-07 Use of an agonist of ppar-alpha and ppar-gamma for the treatment of syndrom x

Publications (1)

Publication Number Publication Date
BR9706968A true BR9706968A (pt) 1999-04-06

Family

ID=10786844

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9706968A BR9706968A (pt) 1996-01-09 1997-01-07 Uso de antagonistas de alfa-ppar e gama-ppar para o tratamento de sindrome x

Country Status (25)

Country Link
US (1) US6166049A (pt)
EP (1) EP0879053A1 (pt)
JP (1) JP2000503643A (pt)
KR (1) KR19990077099A (pt)
CN (1) CN1212622A (pt)
AP (1) AP9801272A0 (pt)
AR (1) AR005404A1 (pt)
AU (1) AU1439797A (pt)
BG (1) BG102668A (pt)
BR (1) BR9706968A (pt)
CA (1) CA2242632A1 (pt)
CZ (1) CZ216398A3 (pt)
EA (1) EA199800626A1 (pt)
GB (1) GB9600464D0 (pt)
HU (1) HUP9900560A3 (pt)
IL (1) IL125106A0 (pt)
MX (1) MX9805539A (pt)
NO (1) NO983147L (pt)
NZ (1) NZ502966A (pt)
OA (1) OA10710A (pt)
PL (1) PL327731A1 (pt)
SK (1) SK92598A3 (pt)
TR (1) TR199801315T2 (pt)
WO (1) WO1997025042A1 (pt)
ZA (1) ZA97171B (pt)

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PL174610B1 (pl) * 1992-07-03 1998-08-31 Smithkline Beecham Plc Nowe związki heterocykliczne
BR9508468A (pt) * 1994-07-29 1997-11-25 Smithkline Beecham Plc Composto processo para a preparação do mesmo composição farmacéutica processos para o tratamento e/ou profilaxia de hiperglicemia em um mamifero humano ou não humano e para o tratamento de hiperlípidemia hipertensão doença cardiovascular alguns distúrbios de alimentação o tratamento e/ou profilaxia de doença renal a prevenção revers o estabilização ou retardo da progressão de microalbuminuria em um mamifero humano ou não humano uso do composto e composto intermediário

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BG102668A (en) 1999-04-30
AR005404A1 (es) 1999-04-28
KR19990077099A (ko) 1999-10-25
TR199801315T2 (xx) 1998-10-21
PL327731A1 (en) 1998-12-21
SK92598A3 (en) 1999-01-11
US6166049A (en) 2000-12-26
IL125106A0 (en) 1999-01-26
GB9600464D0 (en) 1996-03-13
WO1997025042A1 (en) 1997-07-17
ZA97171B (en) 1998-07-24
HUP9900560A3 (en) 2001-04-28
HUP9900560A2 (hu) 1999-07-28
NZ502966A (en) 2001-11-30
CZ216398A3 (cs) 1999-02-17
CN1212622A (zh) 1999-03-31
MX9805539A (es) 1998-11-29
NO983147L (no) 1998-09-08
OA10710A (en) 2002-11-28
AU1439797A (en) 1997-08-01
CA2242632A1 (en) 1997-07-17
EP0879053A1 (en) 1998-11-25
EA199800626A1 (ru) 1998-12-24
WO1997025042A8 (en) 2000-07-20
JP2000503643A (ja) 2000-03-28
AP9801272A0 (en) 1998-06-30

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