BR9204643A - Medicamento,processo para sintese de dicloridrato melaminiltioarseniato de cisteamina ou dicloridrato de melarsomina,e preparacoes de dicloridrato de melarsomina,de diaminoclorotriazina,de cloridrato de melasenacido e de melarsenoxido di-hidratado - Google Patents

Medicamento,processo para sintese de dicloridrato melaminiltioarseniato de cisteamina ou dicloridrato de melarsomina,e preparacoes de dicloridrato de melarsomina,de diaminoclorotriazina,de cloridrato de melasenacido e de melarsenoxido di-hidratado

Info

Publication number
BR9204643A
BR9204643A BR9204643A BR9204643A BR9204643A BR 9204643 A BR9204643 A BR 9204643A BR 9204643 A BR9204643 A BR 9204643A BR 9204643 A BR9204643 A BR 9204643A BR 9204643 A BR9204643 A BR 9204643A
Authority
BR
Brazil
Prior art keywords
hydrohydrated
dychlorhydrate
melarsomine
thylarseniate
dichylhydrochlor
Prior art date
Application number
BR9204643A
Other languages
English (en)
Inventor
Floc H Robert
Jean-Pierre Etchegaray
Gerard Wolf
Patrick Lubert
Regine Jackie Anne-Mari Mazars
Original Assignee
Rhone Merieux
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Merieux filed Critical Rhone Merieux
Publication of BR9204643A publication Critical patent/BR9204643A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/66Arsenic compounds
    • C07F9/70Organo-arsenic compounds
    • C07F9/80Heterocyclic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/66Arsenic compounds
    • C07F9/70Organo-arsenic compounds
    • C07F9/74Aromatic compounds
BR9204643A 1991-12-02 1992-12-01 Medicamento,processo para sintese de dicloridrato melaminiltioarseniato de cisteamina ou dicloridrato de melarsomina,e preparacoes de dicloridrato de melarsomina,de diaminoclorotriazina,de cloridrato de melasenacido e de melarsenoxido di-hidratado BR9204643A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR919114904A FR2684382B1 (fr) 1991-12-02 1991-12-02 Medicaments et preparations pures de dichlorhydrate de melarsomine, leur procede d'obtention et produits intermediaires obtenus.

Publications (1)

Publication Number Publication Date
BR9204643A true BR9204643A (pt) 1993-06-08

Family

ID=9419573

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9204643A BR9204643A (pt) 1991-12-02 1992-12-01 Medicamento,processo para sintese de dicloridrato melaminiltioarseniato de cisteamina ou dicloridrato de melarsomina,e preparacoes de dicloridrato de melarsomina,de diaminoclorotriazina,de cloridrato de melasenacido e de melarsenoxido di-hidratado

Country Status (15)

Country Link
US (3) US5459263A (pt)
JP (1) JP3578277B2 (pt)
AU (1) AU667329B2 (pt)
BR (1) BR9204643A (pt)
CA (1) CA2083766C (pt)
ES (1) ES2039311B1 (pt)
FR (1) FR2684382B1 (pt)
GR (1) GR920100526A (pt)
IT (1) IT1256117B (pt)
MA (1) MA22723A1 (pt)
MX (1) MX9206890A (pt)
MY (1) MY111175A (pt)
PH (1) PH31115A (pt)
PT (1) PT101105B (pt)
TW (1) TW358099B (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2684382B1 (fr) * 1991-12-02 1994-10-21 Rhone Merieux Medicaments et preparations pures de dichlorhydrate de melarsomine, leur procede d'obtention et produits intermediaires obtenus.
US6191123B1 (en) * 1999-03-19 2001-02-20 Parker Hughes Institute Organic-arsenic compounds
AUPQ296799A0 (en) 1999-09-20 1999-10-14 Unisearch Limited A cell-membrane impermeable trivalent organoarsenical derivative and use thereof
EP2088206B1 (en) 2002-11-07 2013-07-03 Newsouth Innovations Pty Limited Induction of the mitochondrial permeability transition
US6686344B1 (en) 2003-01-30 2004-02-03 Paker Hughes Institute Organic-arsonic compounds
AU2007314076B2 (en) 2006-11-01 2012-07-19 Newsouth Innovations Pty Limited Organo-arsenoxide compounds and use thereof
US8324895B2 (en) * 2009-01-23 2012-12-04 Baker Hughes Incorporated MWD/LWD NMR imaging with long echo trains
US8373412B2 (en) * 2009-01-23 2013-02-12 Baker Hughes Incorporated NMR-LWD imaging tool
CN102558234B (zh) * 2011-04-08 2015-01-07 浙江工商大学 一种通过对氨基苯胂酸重氮化制备阿散酸制剂的方法
CN102558235B (zh) * 2011-04-08 2015-01-07 浙江工商大学 一种通过三甲氧苄氨嘧啶重氮化制备阿散酸制剂的方法
US20140051840A1 (en) * 2012-08-17 2014-02-20 The Curators Of The University Of Missouri Arsenic complexes for potential diagnostic applications
US9593052B2 (en) 2012-08-17 2017-03-14 The Curators Of The University Of Missouri Arsenic complexes for potential diagnostic applications

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE437342A (pt) * 1938-12-23 1900-01-01
NL60802C (pt) * 1940-12-10
CH242529A (de) * 1940-12-10 1946-05-15 Friedheim Ernst Albert Hermann Verfahren zur Darstellung von m-(2,4-Diamino-1,3,5-triazinyl-(6))-amino-phenylarsinoxyd.
US2400547A (en) * 1944-01-20 1946-05-21 Ernst A H Friedheim Substituted 1, 3, 5-triazinyl-(6)-aminophenyl-arsenic compounds
US2422724A (en) * 1944-01-20 1947-06-24 Ernst A H Friedheim Substituted 1,3,5-triazinyl-(6)-aminophenyl-arsenic compounds
US2390091A (en) * 1944-06-03 1945-11-27 Ernst A H Friedheim Substituted 1,3,5-triazinyl-(6)-aminophenyl-arsenic compounds
CH254164A (de) * 1946-11-16 1948-04-15 Dr Friedheim Ernst A H Verfahren zur Darstellung von p-(2,4-Diamino-1,3,5-triazinyl-(6)-aminophenyl-arsenoxyd.
CH245837A (de) * 1946-11-16 1946-11-30 Dr Friedheim Ernst A H Verfahren zur Darstellung von p-2,4-Diamino-1,3,5-triazinyl-(6)-amino-phenyl-arsenoxyd.
US2659723A (en) * 1947-01-28 1953-11-17 Ernst A H Friedheim Triazine organometallic compounds and process for preparing same
US2593434A (en) * 1947-02-19 1952-04-22 Ernst A H Friedheim Propylene glycol solution of arsenic medicaments
US3482171A (en) * 1966-07-15 1969-12-02 Itt Bidirectional electronic phase shifter
US3856971A (en) * 1971-07-20 1974-12-24 E Friedheim Method of combating filariasis in dogs
BE786573A (fr) * 1971-07-20 1973-01-22 Hoechst Ag Medicament a base de composes arsenicaux organiques et de derives du benzimidazole
GB2024008B (en) * 1978-06-28 1983-02-16 Merck & Co Inc Compositions for treating trypanosomiasis infections
ZW8781A1 (en) * 1980-05-23 1981-12-16 Hoffmann La Roche 2-nitroimidazoles and preparation thereof
US4514390A (en) * 1982-04-12 1985-04-30 The Rockefeller University Melaminylthioarsenites
FR2572730B1 (fr) * 1984-11-02 1987-12-11 Centre Nat Rech Scient Nouveaux derives de l'arsenic, leur preparation et leur application, notamment comme medicaments antiparasitaires
FR2640269B1 (fr) * 1988-12-13 1991-03-15 Maes Ludo Composes organometalliques, leurs modes de preparation et compositions pharmaceutiques les contenant
FR2684382B1 (fr) * 1991-12-02 1994-10-21 Rhone Merieux Medicaments et preparations pures de dichlorhydrate de melarsomine, leur procede d'obtention et produits intermediaires obtenus.

Also Published As

Publication number Publication date
FR2684382B1 (fr) 1994-10-21
ES2039311B1 (es) 1997-08-16
CA2083766A1 (en) 1993-06-03
PT101105A (pt) 1994-03-31
PT101105B (pt) 1999-10-29
ITMI922692A0 (it) 1992-11-25
MY111175A (en) 1999-09-30
GR920100526A (el) 1993-08-31
AU2972092A (en) 1993-06-03
US5459263A (en) 1995-10-17
PH31115A (en) 1998-02-23
ITMI922692A1 (it) 1994-05-25
MX9206890A (es) 1993-08-01
AU667329B2 (en) 1996-03-21
CA2083766C (en) 2002-09-10
JPH0624960A (ja) 1994-02-01
FR2684382A1 (fr) 1993-06-04
US5635499A (en) 1997-06-03
IT1256117B (it) 1995-11-28
MA22723A1 (fr) 1993-07-01
ES2039311A1 (es) 1993-09-16
JP3578277B2 (ja) 2004-10-20
TW358099B (en) 1999-05-11
US5770733A (en) 1998-06-23

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Legal Events

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EE Request for examination
TC Change of name
EG Technical examination (opinion): publication of technical examination (opinion)
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