BR112019023246B1 - Compostos compreendendo uma fração quelante, métodos para produção dos mesmos e usos dos mesmos - Google Patents
Compostos compreendendo uma fração quelante, métodos para produção dos mesmos e usos dos mesmos Download PDFInfo
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- BR112019023246B1 BR112019023246B1 BR112019023246-0A BR112019023246A BR112019023246B1 BR 112019023246 B1 BR112019023246 B1 BR 112019023246B1 BR 112019023246 A BR112019023246 A BR 112019023246A BR 112019023246 B1 BR112019023246 B1 BR 112019023246B1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/0497—Organic compounds conjugates with a carrier being an organic compounds
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
- C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/003—Compounds containing elements of Groups 3 or 13 of the Periodic Table without C-Metal linkages
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/05—Isotopically modified compounds, e.g. labelled
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Optics & Photonics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
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- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Peptides Or Proteins (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
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| PCT/US2018/031228 WO2018204869A1 (en) | 2017-05-05 | 2018-05-04 | Pharmacokinetic enhancements of bifunctional chelates and uses thereof |
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| ES3034597T3 (en) * | 2018-04-27 | 2025-08-20 | Univ Iowa Res Found | Compositions for chelating metals at low temperatures |
| EA202191556A1 (ru) * | 2018-12-03 | 2021-10-14 | Фьюжн Фармасьютикалз Инк. | Комбинированная терапия радиоиммуноконъюгатами и ингибиторами контрольных точек |
| WO2020186328A1 (en) * | 2019-03-20 | 2020-09-24 | The University Of British Columbia | Chelators and methods of making and using same |
| WO2021142231A1 (en) * | 2020-01-10 | 2021-07-15 | Fusion Pharmaceuticals Inc. | Sustained immunotherapy |
| BR112022013678A2 (pt) * | 2020-01-10 | 2022-11-16 | Fusion Pharmaceuticals Inc | Quelatos macrocíclicos e seus usos |
| IL295999A (en) * | 2020-03-23 | 2022-10-01 | Fusion Pharmaceuticals Inc | Radioimmunoconjugates designed for 3fgfr and their use |
| KR102362962B1 (ko) * | 2020-06-12 | 2022-02-16 | (주)미래바이오팜 | 신규한 화합물 및 이를 함유하는 신경 손상, 신경 질환, 또는 발달 장애에 대한 신경세포의 증식 촉진, 분화, 및/또는 재생을 통한 치료 또는 예방용 약제학적 조성물 |
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| KR20240022616A (ko) * | 2021-06-17 | 2024-02-20 | 메이오 파운데이션 포 메디칼 에쥬케이션 앤드 리써치 | 복수의 킬레이트제와 생물학적 제제를 조합하기 위한 방법 및 재료 |
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2018
- 2018-05-04 KR KR1020197036026A patent/KR102612882B1/ko active Active
- 2018-05-04 EA EA201992595A patent/EA201992595A1/ru unknown
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- 2018-05-04 WO PCT/US2018/031228 patent/WO2018204869A1/en not_active Ceased
- 2018-05-04 CN CN201880039130.2A patent/CN111263747B/zh active Active
- 2018-05-04 MA MA048861A patent/MA48861A/fr unknown
- 2018-05-04 EP EP18793830.3A patent/EP3619191A4/en active Pending
- 2018-05-04 AU AU2018261888A patent/AU2018261888B2/en active Active
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- 2018-05-04 US US15/971,963 patent/US11191854B2/en active Active
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| IL270453B1 (en) | 2025-01-01 |
| RU2019139432A (ru) | 2021-06-07 |
| RU2019139432A3 (https=) | 2021-06-16 |
| JP7693317B2 (ja) | 2025-06-17 |
| KR102612882B1 (ko) | 2023-12-11 |
| BR112019023246A8 (pt) | 2021-02-23 |
| ZA201908071B (en) | 2023-04-26 |
| CL2019003168A1 (es) | 2020-08-28 |
| WO2018204869A1 (en) | 2018-11-08 |
| EP3619191A1 (en) | 2020-03-11 |
| CA3062553C (en) | 2024-02-06 |
| AU2024227706A1 (en) | 2024-11-21 |
| EA201992595A1 (ru) | 2020-04-21 |
| MA48861A (fr) | 2020-04-01 |
| JP2020518673A (ja) | 2020-06-25 |
| AU2018261888B2 (en) | 2022-06-30 |
| AU2018261888A1 (en) | 2019-11-28 |
| US20190030194A1 (en) | 2019-01-31 |
| CN111263747A (zh) | 2020-06-09 |
| JP2023090748A (ja) | 2023-06-29 |
| NZ759832A (en) | 2025-05-30 |
| IL270453A (https=) | 2020-12-31 |
| CA3062553A1 (en) | 2018-11-08 |
| US11191854B2 (en) | 2021-12-07 |
| KR20200006087A (ko) | 2020-01-17 |
| CN117603148A (zh) | 2024-02-27 |
| EP3619191A4 (en) | 2020-12-16 |
| US20220054664A1 (en) | 2022-02-24 |
| BR112019023246A2 (pt) | 2020-05-19 |
| CN111263747B (zh) | 2023-10-27 |
| AU2022221451A1 (en) | 2022-09-22 |
| IL270453B2 (en) | 2025-05-01 |
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