BR112016027824B1 - Processo de preparação de derivados de di-hidroisoxazole - Google Patents
Processo de preparação de derivados de di-hidroisoxazole Download PDFInfo
- Publication number
- BR112016027824B1 BR112016027824B1 BR112016027824-0A BR112016027824A BR112016027824B1 BR 112016027824 B1 BR112016027824 B1 BR 112016027824B1 BR 112016027824 A BR112016027824 A BR 112016027824A BR 112016027824 B1 BR112016027824 B1 BR 112016027824B1
- Authority
- BR
- Brazil
- Prior art keywords
- formula
- compounds
- chlorine
- preparation
- derivatives
- Prior art date
Links
- 0 CC1O*=C(C)C1 Chemical compound CC1O*=C(C)C1 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14170155 | 2014-05-28 | ||
| EP14170155.7 | 2014-05-28 | ||
| PCT/EP2015/061623 WO2015181189A1 (en) | 2014-05-28 | 2015-05-27 | Process for preparing dihydroisoxazole derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112016027824B1 true BR112016027824B1 (pt) | 2021-03-23 |
Family
ID=50828731
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112016027824-0A BR112016027824B1 (pt) | 2014-05-28 | 2015-05-27 | Processo de preparação de derivados de di-hidroisoxazole |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US9796690B2 (https=) |
| EP (1) | EP3148976B1 (https=) |
| JP (1) | JP6533798B2 (https=) |
| KR (1) | KR102337028B1 (https=) |
| CN (1) | CN106414417B (https=) |
| BR (1) | BR112016027824B1 (https=) |
| DK (1) | DK3148976T3 (https=) |
| ES (1) | ES2730048T3 (https=) |
| IL (1) | IL248568B (https=) |
| MX (1) | MX382631B (https=) |
| TW (1) | TWI665192B (https=) |
| WO (1) | WO2015181189A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102595410B1 (ko) * | 2015-03-05 | 2023-10-27 | 바이엘 크롭사이언스 악티엔게젤샤프트 | 3-클로로-2-비닐페닐설포네이트의 제조 방법 |
| EP3548463B1 (de) * | 2016-12-05 | 2020-10-14 | Bayer CropScience Aktiengesellschaft | Verfahren zur herstellung von 3-substituierten 2-vinylphenylsulfonaten |
| WO2020251006A1 (ja) * | 2019-06-14 | 2020-12-17 | クミアイ化学工業株式会社 | ジヒドロイソキサゾールの製造方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| OA09122A (en) | 1988-07-08 | 1991-10-31 | Schering Agrochemicals Ltd | Triazole insecticides. |
| DE4331448A1 (de) | 1993-09-16 | 1995-03-23 | Hoechst Schering Agrevo Gmbh | Substituierte Isoxazoline, Verfahren zu deren Herstellung, diese enthaltende Mittel und deren Verwendung als Safener |
| EP1878730A1 (en) | 2006-07-12 | 2008-01-16 | Bayer Schering Pharma Aktiengesellschaft | Substituted isoxazolines, pharmaceutical compositions containing the same, methods of preparing the same, and uses of the same |
| WO2008013622A2 (en) * | 2006-07-27 | 2008-01-31 | E. I. Du Pont De Nemours And Company | Fungicidal azocyclic amides |
| CN101970432B (zh) * | 2008-01-25 | 2014-05-28 | 杜邦公司 | 杀真菌杂环化合物 |
| CN101925598B (zh) * | 2008-01-25 | 2014-03-05 | 杜邦公司 | 杀真菌酰胺 |
| TW201021852A (en) | 2008-11-17 | 2010-06-16 | Enzon Pharmaceuticals Inc | Releasable fusogenic lipids for nucleic acids delivery systems |
| KR20120112755A (ko) * | 2010-01-07 | 2012-10-11 | 이 아이 듀폰 디 네모아 앤드 캄파니 | 살진균제 복소환 화합물 |
| DK2921493T3 (da) * | 2011-12-27 | 2017-11-27 | Bayer Ip Gmbh | Heteroarylpiperidin og ¿piperazinderivater |
| EP2820015A1 (en) * | 2012-03-02 | 2015-01-07 | Syngenta Participations AG | Microbiocidal pyrazole derivatives |
-
2015
- 2015-05-26 TW TW104116745A patent/TWI665192B/zh active
- 2015-05-27 CN CN201580027637.2A patent/CN106414417B/zh active Active
- 2015-05-27 ES ES15724677T patent/ES2730048T3/es active Active
- 2015-05-27 DK DK15724677.8T patent/DK3148976T3/da active
- 2015-05-27 MX MX2016015623A patent/MX382631B/es unknown
- 2015-05-27 BR BR112016027824-0A patent/BR112016027824B1/pt active IP Right Grant
- 2015-05-27 KR KR1020167035419A patent/KR102337028B1/ko active Active
- 2015-05-27 EP EP15724677.8A patent/EP3148976B1/en active Active
- 2015-05-27 US US15/314,446 patent/US9796690B2/en active Active
- 2015-05-27 WO PCT/EP2015/061623 patent/WO2015181189A1/en not_active Ceased
- 2015-05-27 JP JP2016569396A patent/JP6533798B2/ja active Active
-
2016
- 2016-10-27 IL IL248568A patent/IL248568B/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| CN106414417A (zh) | 2017-02-15 |
| DK3148976T3 (da) | 2019-05-27 |
| WO2015181189A1 (en) | 2015-12-03 |
| TW201625567A (zh) | 2016-07-16 |
| KR102337028B1 (ko) | 2021-12-07 |
| EP3148976A1 (en) | 2017-04-05 |
| MX382631B (es) | 2025-03-13 |
| CN106414417B (zh) | 2019-04-16 |
| EP3148976B1 (en) | 2019-03-13 |
| JP2017517513A (ja) | 2017-06-29 |
| MX2016015623A (es) | 2017-02-27 |
| TWI665192B (zh) | 2019-07-11 |
| ES2730048T3 (es) | 2019-11-07 |
| IL248568A0 (en) | 2016-12-29 |
| JP6533798B2 (ja) | 2019-06-19 |
| US9796690B2 (en) | 2017-10-24 |
| IL248568B (en) | 2019-03-31 |
| KR20170012331A (ko) | 2017-02-02 |
| US20170247345A1 (en) | 2017-08-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06U | Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette] | ||
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 27/05/2015, OBSERVADAS AS CONDICOES LEGAIS. |