BR112016019469B1 - Tratamento de infecções por h. pylori utilizando -se inibidores de mtan - Google Patents
Tratamento de infecções por h. pylori utilizando -se inibidores de mtan Download PDFInfo
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- BR112016019469B1 BR112016019469B1 BR112016019469-1A BR112016019469A BR112016019469B1 BR 112016019469 B1 BR112016019469 B1 BR 112016019469B1 BR 112016019469 A BR112016019469 A BR 112016019469A BR 112016019469 B1 BR112016019469 B1 BR 112016019469B1
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- pylori
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- silica gel
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Images
Classifications
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
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- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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- Chemical & Material Sciences (AREA)
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- Organic Chemistry (AREA)
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- Nitrogen Condensed Heterocyclic Rings (AREA)
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| PCT/US2015/014778 WO2015123101A1 (en) | 2014-02-12 | 2015-02-06 | Treatment of h. pylori infections using mtan inhibitors |
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| BR112016019469A2 BR112016019469A2 (pt) | 2018-07-24 |
| BR112016019469B1 true BR112016019469B1 (pt) | 2022-12-06 |
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| CN108794628A (zh) * | 2018-05-28 | 2018-11-13 | 广东工业大学 | 一种抗幽门螺杆菌的卵黄抗体制备方法及应用 |
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| AU2003245442B2 (en) * | 2002-06-13 | 2009-02-05 | Vertex Pharmaceuticals Incorporated | 2-ureido-6-heteroaryl-3h-benzoimidazole-4-carboxylic acid derivatives and related compounds as gyrase and/or topoisomerase IV inhibitors for the treatment of bacterial infections |
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| NZ533360A (en) | 2004-06-04 | 2007-02-23 | Ind Res Ltd | Improved method for preparing 3-hydroxy-4-hydroxymethyl-pyrrolidine compounds |
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| DK2114925T3 (da) | 2006-12-22 | 2012-05-29 | Ind Res Ltd | Azetidin-analoger af nucleosidase- og phosphorylase-inhibitorer |
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| WO2010033236A2 (en) * | 2008-09-22 | 2010-03-25 | Albert Einstein College Of Medicine Of Yeshiva University | Methods and compositions for treating bacterial infections by inhibiting quorum sensing |
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| US9290501B2 (en) * | 2010-11-29 | 2016-03-22 | Albert Einstein College Of Medicine, Inc. | Methods, assays and compounds for treating bacterial infections by inhibiting methylthioinosine phosphorylase |
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- 2015-02-06 RU RU2016136533A patent/RU2663803C2/ru active
- 2015-02-06 BR BR112016019469-1A patent/BR112016019469B1/pt active IP Right Grant
- 2015-02-06 SG SG10201806381VA patent/SG10201806381VA/en unknown
- 2015-02-06 JP JP2016552328A patent/JP6512613B2/ja active Active
- 2015-02-06 US US15/118,113 patent/US10118928B2/en active Active
- 2015-02-06 AU AU2015217416A patent/AU2015217416B2/en active Active
- 2015-02-06 NZ NZ724103A patent/NZ724103A/en unknown
- 2015-02-06 SG SG11201606595RA patent/SG11201606595RA/en unknown
- 2015-02-06 CA CA2974916A patent/CA2974916C/en active Active
- 2015-02-06 HK HK17105755.5A patent/HK1232071A1/zh unknown
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2016
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2018
- 2018-09-20 US US16/136,314 patent/US10294233B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| CA2974916A1 (en) | 2015-08-20 |
| AU2015217416B2 (en) | 2018-10-04 |
| WO2015123101A1 (en) | 2015-08-20 |
| RU2016136533A3 (enExample) | 2018-06-06 |
| JP2017506238A (ja) | 2017-03-02 |
| RU2663803C2 (ru) | 2018-08-09 |
| US10118928B2 (en) | 2018-11-06 |
| IL247218A0 (en) | 2016-09-29 |
| NZ724103A (en) | 2020-07-31 |
| BR112016019469A2 (pt) | 2018-07-24 |
| SG10201806381VA (en) | 2018-08-30 |
| CA2974916C (en) | 2022-05-31 |
| US20190016730A1 (en) | 2019-01-17 |
| EP3104707A1 (en) | 2016-12-21 |
| AU2015217416A1 (en) | 2016-09-29 |
| US20170166571A1 (en) | 2017-06-15 |
| SG11201606595RA (en) | 2016-09-29 |
| EP3104707B1 (en) | 2020-07-15 |
| US10294233B2 (en) | 2019-05-21 |
| HK1232071A1 (zh) | 2018-01-05 |
| IL247218B (en) | 2020-06-30 |
| EP3104707A4 (en) | 2017-12-13 |
| JP6512613B2 (ja) | 2019-05-15 |
| RU2016136533A (ru) | 2018-03-13 |
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