BR112015025058A8 - Composição farmacêutica do tipo matriz contendo lacosamida - Google Patents
Composição farmacêutica do tipo matriz contendo lacosamidaInfo
- Publication number
- BR112015025058A8 BR112015025058A8 BR112015025058A BR112015025058A BR112015025058A8 BR 112015025058 A8 BR112015025058 A8 BR 112015025058A8 BR 112015025058 A BR112015025058 A BR 112015025058A BR 112015025058 A BR112015025058 A BR 112015025058A BR 112015025058 A8 BR112015025058 A8 BR 112015025058A8
- Authority
- BR
- Brazil
- Prior art keywords
- pharmaceutical composition
- lacosamide
- composition containing
- matrix type
- type pharmaceutical
- Prior art date
Links
- VPPJLAIAVCUEMN-GFCCVEGCSA-N lacosamide Chemical compound COC[C@@H](NC(C)=O)C(=O)NCC1=CC=CC=C1 VPPJLAIAVCUEMN-GFCCVEGCSA-N 0.000 title abstract 4
- 229960002623 lacosamide Drugs 0.000 title abstract 4
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 4
- 239000011159 matrix material Substances 0.000 title 1
- 150000003839 salts Chemical class 0.000 abstract 3
- 238000004090 dissolution Methods 0.000 abstract 2
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
Abstract
COMPOSIÇÃO FARMACÊUTICA CAPAZ DE CONTROLAR FACILMENTE O PADRÃO DE DISSOLUÇÃO DE LACOSAMIDA OU DE UM SAL FARMACEUTICAMENTE ACEITÁVEL DA MESMA. A presente invenção refere-se a uma composição farmacêutica do tipo matriz contendo lacosamida, que é um princípio ativo, ou um sal farmaceuticamente aceitável da mesma. Mais especificamente, a presente invenção refere-se a uma composição farmacêutica capaz de controlar facilmente o padrão de dissolução de uma quantidade eficaz de lacosamida ou um sal farmaceuticamente aceitável da mesma.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR10-2013-0035989 | 2013-04-02 | ||
KR1020130035989A KR101732731B1 (ko) | 2013-04-02 | 2013-04-02 | 라코사마이드(lacosamide) 또는 이의 약학적으로 허용 가능한 염의 용출 패턴 조절이 용이한 약학 조성물 |
PCT/KR2014/002454 WO2014163314A1 (ko) | 2013-04-02 | 2014-03-24 | 라코사마이드(lacosamide) 또는 이의 약학적으로 허용 가능한 염의 용출 패턴 조절이 용이한 약학 조성물 |
Publications (3)
Publication Number | Publication Date |
---|---|
BR112015025058A2 BR112015025058A2 (pt) | 2017-07-18 |
BR112015025058A8 true BR112015025058A8 (pt) | 2023-01-03 |
BR112015025058B1 BR112015025058B1 (pt) | 2023-11-21 |
Family
ID=51658558
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112015025058-0A BR112015025058B1 (pt) | 2013-04-02 | 2014-03-24 | Composição farmacêutica do tipo matriz contendo lacosamida |
Country Status (4)
Country | Link |
---|---|
KR (1) | KR101732731B1 (pt) |
CN (1) | CN105228608B (pt) |
BR (1) | BR112015025058B1 (pt) |
WO (1) | WO2014163314A1 (pt) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN104784134B (zh) * | 2015-04-12 | 2018-05-29 | 石家庄四药有限公司 | 一种拉科酰胺固体制剂及其制备方法 |
MA43532A (fr) | 2015-12-30 | 2018-11-07 | Adamas Pharmaceuticals Inc | Méthodes et compositions destinés au traitement de troubles liés à des crises épileptiques |
KR102544141B1 (ko) * | 2016-09-29 | 2023-06-16 | 에스케이케미칼 주식회사 | 라코사미드 서방성 제제 |
KR102083241B1 (ko) | 2018-02-14 | 2020-03-02 | 환인제약 주식회사 | 라코사미드를 함유하는 약제학적 서방성 조성물 |
CN109010301B (zh) * | 2018-09-05 | 2021-01-26 | 上海上药第一生化药业有限公司 | 一种拉考沙胺晶型ii片剂及其制备方法和应用 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2011008298A2 (en) * | 2009-07-16 | 2011-01-20 | Nectid, Inc. | Novel axomadol dosage forms |
WO2011055385A1 (en) * | 2009-11-03 | 2011-05-12 | Lupin Limited | Modified release formulation of lacosamide |
WO2011101863A2 (en) | 2010-02-19 | 2011-08-25 | Cadila Healthcare Limited | Extended release pharmaceutical compositions of lacosamide |
MX2013005974A (es) | 2010-12-02 | 2013-07-29 | Ucb Pharma Gmbh | Formulacion de lacosamida de administracion una vez al dia. |
EP2468261A1 (en) * | 2010-12-02 | 2012-06-27 | UCB Pharma GmbH | Formulation of lacosamide |
-
2013
- 2013-04-02 KR KR1020130035989A patent/KR101732731B1/ko active IP Right Grant
-
2014
- 2014-03-24 CN CN201480019538.5A patent/CN105228608B/zh active Active
- 2014-03-24 WO PCT/KR2014/002454 patent/WO2014163314A1/ko active Application Filing
- 2014-03-24 BR BR112015025058-0A patent/BR112015025058B1/pt active IP Right Grant
Also Published As
Publication number | Publication date |
---|---|
BR112015025058A2 (pt) | 2017-07-18 |
KR20140120191A (ko) | 2014-10-13 |
WO2014163314A1 (ko) | 2014-10-09 |
CN105228608B (zh) | 2019-05-28 |
BR112015025058B1 (pt) | 2023-11-21 |
KR101732731B1 (ko) | 2017-05-08 |
CN105228608A (zh) | 2016-01-06 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
B06U | Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette] | ||
B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
B25D | Requested change of name of applicant approved |
Owner name: BIOINNOTIS CO., LTD. (KR) |
|
B25A | Requested transfer of rights approved |
Owner name: HYUNDAI PHARM CO., LTD. (KR) |
|
B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 24/03/2014, OBSERVADAS AS CONDICOES LEGAIS |