BR112014027841B1 - Uso de derivados de pirazola na fabricação de um fármaco para prevenir ou tratar constipação - Google Patents
Uso de derivados de pirazola na fabricação de um fármaco para prevenir ou tratar constipação Download PDFInfo
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- BR112014027841B1 BR112014027841B1 BR112014027841-5A BR112014027841A BR112014027841B1 BR 112014027841 B1 BR112014027841 B1 BR 112014027841B1 BR 112014027841 A BR112014027841 A BR 112014027841A BR 112014027841 B1 BR112014027841 B1 BR 112014027841B1
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/7056—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing five-membered rings with nitrogen as a ring hetero atom
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
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- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
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| PL3400944T3 (pl) | 2010-11-04 | 2020-11-16 | Albireo Ab | Inhibitory ibat w leczeniu chorób wątroby |
| PL2848254T3 (pl) * | 2012-05-07 | 2017-03-31 | Kissei Pharmaceutical Co., Ltd. | Pochodne pirazolu i ich zastosowanie w celach medycznych |
| MX346453B (es) | 2013-02-04 | 2017-03-17 | Taisho Pharmaceutical Co Ltd | Medicamento profilactico o terapeutico para el estreñimiento. |
| KR102560954B1 (ko) | 2014-06-25 | 2023-07-31 | 이에이 파마 가부시키가이샤 | 고형 제제 및 그의 착색 방지 또는 착색 감소 방법 |
| WO2015199146A1 (ja) * | 2014-06-25 | 2015-12-30 | 味の素株式会社 | 固形製剤及びその安定化方法 |
| BR112020019624A8 (pt) | 2018-03-28 | 2022-03-03 | Avolynt | Método para tratar a hipoglicemia pós-prandial |
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| EP3810084A1 (en) | 2018-06-20 | 2021-04-28 | Albireo AB | Pharmaceutical formulation of odevixibat |
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| US10941127B2 (en) | 2019-02-06 | 2021-03-09 | Albireo Ab | Benzothiadiazepine compounds and their use as bile acid modulators |
| DK3921028T3 (da) | 2019-02-06 | 2023-01-23 | Albireo Ab | Benzothiadiazepinforbindelser og anvendelse deraf som galdesyremodulatorer |
| CN114761018B (zh) | 2019-12-04 | 2025-12-02 | 阿尔比里奥公司 | 苯并硫杂二氮杂环庚三烯化合物及其作为胆汁酸调节剂的用途 |
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| JP7696897B2 (ja) | 2019-12-04 | 2025-06-23 | アルビレオ・アクチボラグ | ベンゾチア（ジ）アゼピン化合物及び胆汁酸モジュレータとしてのそれらの使用 |
| US11014898B1 (en) | 2020-12-04 | 2021-05-25 | Albireo Ab | Benzothiazepine compounds and their use as bile acid modulators |
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| JP2023549226A (ja) | 2020-11-12 | 2023-11-22 | アルビレオ エービー | 進行性家族性肝内胆汁うっ滞症（ｐｆｉｃ）を処置するためのオデビキシバット |
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| TW202313579A (zh) | 2021-06-03 | 2023-04-01 | 瑞典商艾爾比瑞歐公司 | 苯并噻(二)氮呯(benzothia(di)azepine)化合物及其作為膽酸調節劑之用途 |
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| MX2008013583A (es) * | 2006-04-26 | 2008-10-31 | Genentech Inc | Compuestos del inhibidor de fosfoinositido 3-cinasa y composiciones farmaceuticas que los contienen. |
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| TW201105336A (en) * | 2009-07-01 | 2011-02-16 | Kissei Pharmaceutical | Combined medicine of pyrazole derivative and biguanide drug |
| AR087701A1 (es) | 2011-08-31 | 2014-04-09 | Japan Tobacco Inc | Derivados de pirazol con actividad inhibidora de sglt1 |
| PL2848254T3 (pl) * | 2012-05-07 | 2017-03-31 | Kissei Pharmaceutical Co., Ltd. | Pochodne pirazolu i ich zastosowanie w celach medycznych |
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| US20150141631A1 (en) | 2015-05-21 |
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| DK2848254T3 (en) | 2016-10-31 |
| JPWO2013168671A1 (ja) | 2016-01-07 |
| CA2872002C (en) | 2019-01-15 |
| PL2848254T3 (pl) | 2017-03-31 |
| PT2848254T (pt) | 2016-10-05 |
| CA2872002A1 (en) | 2013-11-14 |
| CN104284665B (zh) | 2016-11-16 |
| US9273085B2 (en) | 2016-03-01 |
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| JP2015083580A (ja) | 2015-04-30 |
| KR101868991B1 (ko) | 2018-06-19 |
| BR112014027841A2 (pt) | 2017-06-27 |
| AU2013258566B2 (en) | 2017-03-16 |
| KR20150013671A (ko) | 2015-02-05 |
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| MX2014013696A (es) | 2015-02-05 |
| EP2848254A1 (en) | 2015-03-18 |
| BR112014027841A8 (pt) | 2021-09-28 |
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