BR0316187A - Formulações parasiticidas tópicas e métodos de tratamento - Google Patents

Formulações parasiticidas tópicas e métodos de tratamento

Info

Publication number
BR0316187A
BR0316187A BR0316187-0A BR0316187A BR0316187A BR 0316187 A BR0316187 A BR 0316187A BR 0316187 A BR0316187 A BR 0316187A BR 0316187 A BR0316187 A BR 0316187A
Authority
BR
Brazil
Prior art keywords
formulations
cattle
water
methods
treatment methods
Prior art date
Application number
BR0316187-0A
Other languages
English (en)
Inventor
Stanley Shepherd
Original Assignee
Schering Plough Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Plough Ltd filed Critical Schering Plough Ltd
Publication of BR0316187A publication Critical patent/BR0316187A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • A61K9/0017Non-human animal skin, e.g. pour-on, spot-on
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

"FORMULAçõES PARASITICIDAS TóPICAS E MéTODOS DE TRATAMENTO". A presente invenção refere-se a formulações aquosas micélicas para administração tópica de benzimidazóis e salicilanilidas com lactonas macrocíclicas em gados, para o controle de endoparasitas e ectoparasitas, compreendendo um primeiro agente ativo, selecionado entre benzimidazóis, salicilanilidas e seus derivados ou sais ativos, insolúveis em água, em combinação com um segundo agente ativo, selecionado entre lactonas macrocíclicas ou derivados ou sais ativos delas, e compreendendo também, por litro de formulação: entre cerca de 100 g e cerca de 400 g de tensoativo(s) de uso veterinário; entre cerca de 200 g e cerca de 750 g de solvente(s) miscível em água, de uso veterinário; e entre cerca de 50 e cerca de 350 g de água; bem como métodos para dosificar tais formulações para os gados, e métodos para controlar e/ou prevenir doenças ou infecção parasítica em gados.
BR0316187-0A 2002-11-11 2003-11-11 Formulações parasiticidas tópicas e métodos de tratamento BR0316187A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AU2002952597A AU2002952597A0 (en) 2002-11-11 2002-11-11 Topical parasiticide formulations and methods of treatment
PCT/AU2003/001490 WO2004043445A1 (en) 2002-11-11 2003-11-11 Topical parasiticide formulations and methods of treatment

Publications (1)

Publication Number Publication Date
BR0316187A true BR0316187A (pt) 2005-09-27

Family

ID=28795986

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0316187-0A BR0316187A (pt) 2002-11-11 2003-11-11 Formulações parasiticidas tópicas e métodos de tratamento

Country Status (14)

Country Link
US (1) US20060121072A1 (pt)
EP (1) EP1560572A4 (pt)
JP (3) JP4643990B2 (pt)
KR (1) KR20050090385A (pt)
AR (1) AR041936A1 (pt)
AU (1) AU2002952597A0 (pt)
BR (1) BR0316187A (pt)
CA (1) CA2504197A1 (pt)
MX (1) MXPA05005046A (pt)
NZ (1) NZ540589A (pt)
PE (1) PE20040545A1 (pt)
TW (1) TWI314848B (pt)
WO (1) WO2004043445A1 (pt)
ZA (1) ZA200503758B (pt)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2002952597A0 (en) * 2002-11-11 2002-11-28 Schering-Plough Pty. Limited Topical parasiticide formulations and methods of treatment
GB0316377D0 (en) * 2003-07-12 2003-08-13 Norbrook Lab Ltd Parasiticidal composition
US7666444B2 (en) 2004-02-02 2010-02-23 Wyeth Antiparasitic composition
WO2005074914A1 (en) * 2004-02-03 2005-08-18 Wyeth Anthelmintic composition
MXPA06014303A (es) 2004-06-07 2007-02-19 Syngenta Participations Ag Metodos para reducir el dano producido por nematodos.
WO2006061214A1 (en) * 2004-12-10 2006-06-15 Bayer Healthcare Ag Anthelmintic composition
KR101233488B1 (ko) 2005-09-15 2013-02-14 메리얼 리미티드 구충 제형
CA2630458C (en) * 2005-12-06 2014-10-28 Wyeth Benzimidazole non-aqueous compositions
GB2451811A (en) * 2007-08-09 2009-02-18 Ems Sa Delivery composition for solubilising water-insoluble pharmaceutical active ingredients
CA2706448C (en) * 2007-11-26 2016-08-16 Merial Limited Solvent systems for pour-on formulations for combating parasites
AU2013201461B2 (en) * 2007-11-26 2015-10-29 Boehringer Ingelheim Animal Health USA Inc. Solvent systems for pour-on formulations for combating parasites
PT2331068T (pt) 2008-10-08 2017-03-13 Zoetis Services Llc Composições anti-helmínticas de benzimidazol
WO2011048040A1 (en) * 2009-10-19 2011-04-28 Intervet International B.V. Method and formulation for the control of parasites
NZ603699A (en) * 2010-05-12 2013-08-30 Merial Ltd Injectable parasiticidal formulations of levamisole and macrocyclic lactones
US11166912B2 (en) 2016-03-03 2021-11-09 Ctt Pharma Inc. Orally administrable composition
KR101855989B1 (ko) 2016-12-23 2018-05-09 강원대학교산학협력단 가용화제를 첨가한 물을 추출용매로 이용한 유용성분이 증가된 메밀 종자 추출물의 제조 방법 및 그에 따른 메밀 종자 추출물
US11298336B2 (en) 2019-05-30 2022-04-12 Soluble Technologies, Inc. Water soluble formulation
US11786475B2 (en) 2020-07-22 2023-10-17 Soluble Technologies Inc. Film-based dosage form

Family Cites Families (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3914418A (en) * 1971-09-02 1975-10-21 Merck & Co Inc Methods of controlling liver fluke infections
US3989826A (en) * 1972-05-12 1976-11-02 Ici Australia Limited Method of killing internal parasites using salicylanilides
US3927071A (en) * 1972-05-12 1975-12-16 Ici Australia Ltd Salicylanilides
US3950360A (en) * 1972-06-08 1976-04-13 Sankyo Company Limited Antibiotic substances
US4336262A (en) * 1973-02-23 1982-06-22 Fisons Ltd. Pour-on veterinary anthelmintic
GB1493375A (en) * 1974-09-20 1977-11-30 Ici Ltd Salicylanilide derivatives
US4005218A (en) * 1975-03-18 1977-01-25 Janssen Pharmaceutica N.V. Antiparasitic salicylanilide derivatives
DE3029426A1 (de) * 1980-08-02 1982-03-11 Bayer Ag, 5090 Leverkusen Gegen zwecken wirksame pour-on-formulierungen
OA06863A (fr) * 1980-08-04 1983-02-28 Merck & Co Inc Solubilisation de l'invermectine dans l'eau.
US4389397A (en) * 1980-08-04 1983-06-21 Merck & Co., Inc. Solubilization of ivermectin in water
US4607050A (en) * 1981-10-19 1986-08-19 Wellcome Australia Limited Method of controlling insects and parasites with an aqueous localized pour-on formulation
NZ203574A (en) * 1982-03-16 1986-04-11 Wellcome Australia Pour on compositions containing pyrethroids and thiazoles
EP0179583A1 (en) * 1984-10-04 1986-04-30 Merck & Co. Inc. A system for enhancing the water dissolution rate and solubility of poorly soluble drugs
GB8723347D0 (en) * 1987-10-05 1987-11-11 Shell Int Research Ectoparasiticidal pour-on formulation
US5639949A (en) * 1990-08-20 1997-06-17 Ciba-Geigy Corporation Genes for the synthesis of antipathogenic substances
NZ335166A (en) * 1999-04-14 2001-11-30 Ashmont Holdings Ltd Anthelmintic composition containing triclabendazole in at least one solvent
US5602107A (en) * 1993-05-10 1997-02-11 Merck & Co., Inc. Pour-on formulations consisting of gylcols, glycerides and avermectin compounds
PL174488B1 (pl) * 1993-05-10 1998-08-31 Merck & Co Inc Preparat do zwalczania pasożytów zwierząt oraz sposób wytwarzania preparatu do zwalczania pasożytów zwierząt
BR9406627A (pt) * 1993-05-26 1996-02-06 Commw Scient Ind Res Org Composições antiparasiticas
DK72593D0 (da) * 1993-06-18 1993-06-18 Symbicom Ab Rekombinant protein
NZ260018A (en) * 1994-03-03 1995-10-26 Bomac Lab Ltd Benzimidazole compositions and anthelmintic compositions
US6010710A (en) * 1996-03-29 2000-01-04 Merial Direct pour-on skin solution for antiparasitic use in cattle and sheep
FR2755824B1 (fr) * 1996-11-19 1999-01-08 Virbac Sa Formulation galenique des benzimidazoles a usage topique, son procede de preparation et ses utilisations
CN1069032C (zh) * 1997-03-27 2001-08-01 中国农业大学 一种含阿维菌素/依维菌素的兽用抗寄生虫药
US5968990A (en) * 1997-10-14 1999-10-19 Isp Investments Inc. Water-dilutable, microemulsion concentrate and pour-on formulations thereof
AUPP105497A0 (en) * 1997-12-19 1998-01-15 Schering-Plough Animal Health Limited Aqueous insecticidal pour-on treatment
CN1214909A (zh) * 1998-05-14 1999-04-28 王玉万 一种复方兽用抗寄生虫药
US6103248A (en) * 1998-05-22 2000-08-15 Burkhart; Craig G. Topical preparation and therapy for head lice
IL143604A0 (en) * 1998-12-30 2002-04-21 Dexcel Ltd Dispersable concentrate for the delivery of cyclosporin
AU772988B2 (en) * 1999-06-04 2004-05-13 Elanco Tiergesundheit Ag Stable biocidal compositions
US6340672B1 (en) * 2000-02-16 2002-01-22 Phoenix Scientific, Inc. Parasiticidal formulation and a method of making this formulation
US6787342B2 (en) * 2000-02-16 2004-09-07 Merial Limited Paste formulations
EP1129713A1 (en) * 2000-02-29 2001-09-05 New Pharma Research Sweden AB Veterinary compositions for the treatment of parasitic diseases
GB2386066A (en) * 2002-02-28 2003-09-10 Norbrook Lab Ltd Long-acting parasiticidal composition with improved bioavailability comprising a salicylanilide, a further anti-parasitic compound & a polymeric species
AU2002952597A0 (en) * 2002-11-11 2002-11-28 Schering-Plough Pty. Limited Topical parasiticide formulations and methods of treatment
NZ523128A (en) * 2002-12-12 2006-01-27 Ashmont Holdings Ltd Anthelmintic formulations containing avermectins and or milbemycins
GB0316377D0 (en) * 2003-07-12 2003-08-13 Norbrook Lab Ltd Parasiticidal composition

Also Published As

Publication number Publication date
MXPA05005046A (es) 2005-11-17
JP2011105765A (ja) 2011-06-02
JP2006508108A (ja) 2006-03-09
NZ540589A (en) 2008-03-28
EP1560572A1 (en) 2005-08-10
ZA200503758B (en) 2006-11-29
AU2002952597A0 (en) 2002-11-28
PE20040545A1 (es) 2004-08-28
AR041936A1 (es) 2005-06-01
JP4643990B2 (ja) 2011-03-02
EP1560572A4 (en) 2011-05-04
US20060121072A1 (en) 2006-06-08
WO2004043445A1 (en) 2004-05-27
KR20050090385A (ko) 2005-09-13
JP2007008963A (ja) 2007-01-18
TW200423871A (en) 2004-11-16
TWI314848B (en) 2009-09-21
CA2504197A1 (en) 2004-05-27

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 11A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2280 DE 16/09/2014.