BR0311834A - Composto, composição farmacêutica, métodos para mudular um receptor ativado por proliferador de peroxisoma, para tratar e prevenir diabetes mellitus em um mamìfero e para tratar sìndrome x em um mamìfero, e, uso de um composto ou seu sal farmaceuticamente aceitável - Google Patents

Composto, composição farmacêutica, métodos para mudular um receptor ativado por proliferador de peroxisoma, para tratar e prevenir diabetes mellitus em um mamìfero e para tratar sìndrome x em um mamìfero, e, uso de um composto ou seu sal farmaceuticamente aceitável

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Publication number
BR0311834A
BR0311834A BR0311834-7A BR0311834A BR0311834A BR 0311834 A BR0311834 A BR 0311834A BR 0311834 A BR0311834 A BR 0311834A BR 0311834 A BR0311834 A BR 0311834A
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Brazil
Prior art keywords
compound
mammal
treating
modulating
pharmaceutical composition
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BR0311834-7A
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English (en)
Inventor
Rafael Ferritto Crespo
Jose Alfredo Martin
Maria Dolores Martin-Or Finger
Isabel Rojo Garcia
Quanrong Shen
Alan M Warshawsky
Yanping Xu
Original Assignee
Lilly Co Eli
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Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of BR0311834A publication Critical patent/BR0311834A/pt

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    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
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  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
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Abstract

"COMPOSTO, COMPOSIçãO FARMACêUTICA, MéTODOS PARA MODULAR UM RECEPTOR ATIVADO POR PROLIFERADOR DE PEROXISOMA, PARA TRATAR E PREVENIR DIABETES MELLITUS EM UM MAMìFERO E PARA TRATAR SìNDROME X EM UM MAMìFERO, E, USO DE UM COMPOSTO OU SEU SAL FARMACEUTICAMENTE ACEITáVEL". A presente invenção refere-se a compostos, composições, e ao uso de compostos de Fórmula estrutural (I).
BR0311834-7A 2002-06-19 2003-06-11 Composto, composição farmacêutica, métodos para mudular um receptor ativado por proliferador de peroxisoma, para tratar e prevenir diabetes mellitus em um mamìfero e para tratar sìndrome x em um mamìfero, e, uso de um composto ou seu sal farmaceuticamente aceitável BR0311834A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US39010202P 2002-06-19 2002-06-19
PCT/US2003/016207 WO2004000789A1 (en) 2002-06-19 2003-06-11 Amide linker peroxisome proliferator activated receptor modulators

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BR0311834A true BR0311834A (pt) 2005-04-12

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US (1) US7220880B2 (pt)
EP (1) EP1517882A1 (pt)
JP (1) JP2005529975A (pt)
CN (1) CN1662487A (pt)
AR (1) AR039684A1 (pt)
AU (1) AU2003241579B9 (pt)
BR (1) BR0311834A (pt)
CA (1) CA2488972A1 (pt)
MX (1) MXPA04013000A (pt)
PE (1) PE20040580A1 (pt)
TW (1) TW200406371A (pt)
WO (1) WO2004000789A1 (pt)

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GB0314079D0 (en) * 2003-06-18 2003-07-23 Astrazeneca Ab Therapeutic agents
GB0229931D0 (en) 2002-12-21 2003-01-29 Astrazeneca Ab Therapeutic agents
SE0104334D0 (sv) * 2001-12-19 2001-12-19 Astrazeneca Ab Therapeutic agents
BRPI0417401A (pt) * 2003-12-15 2007-05-08 Lilly Co Eli composto, composição farmacêutica, métodos para modular um receptor ativado por proliferador de peroxissomo, para tratar doença ou condição, para abaixar glicose sanguìnea em um mamìfero, para tratar diabetes mellitus em um mamìfero, para tratar doença cardiovascular em um mamìfero, para tratar sìndrome x em um mamìfero, e, uso de composto
GB0405033D0 (en) * 2004-03-05 2004-04-07 Karobio Ab Novel pharmaceutical compositions
MXPA06014574A (es) 2004-06-24 2007-03-12 Incyte Corp Piperidinas n-sustituidas y su uso como farmaceuticos.
EP1768954A4 (en) * 2004-06-24 2008-05-28 Incyte Corp 2-METHYLPROPANAMIDES AND THEIR USE AS PHARMACEUTICALS
GT200500375A (es) * 2004-12-20 2006-11-28 Derivados de piperidina y su uso como agentes antiinflamatorios
WO2006129164A1 (en) 2005-05-31 2006-12-07 Pfizer Japan Inc. Substituted aryloxy-n-bicyclomethyl acetamide compounds as vr1 antagonists
US8097610B2 (en) * 2005-08-26 2012-01-17 Shionogi & Co., Ltd. Derivative having PPAR agonistic activity
JP2008239616A (ja) * 2007-02-28 2008-10-09 Iyaku Bunshi Sekkei Kenkyusho:Kk Ｈｄｌ上昇剤
CN107382980B (zh) * 2016-05-14 2020-05-15 湖南大学 N-[(二氢苯并呋喃-7-氧基)烷基]-2-芳氧基酰胺衍生物
EP3689324A1 (de) * 2019-02-04 2020-08-05 Symrise AG Neue kühlstoffe und zubereitungen, die diese enthalten

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PE20040580A1 (es) 2004-09-08
MXPA04013000A (es) 2005-09-12
WO2004000789A9 (en) 2004-03-11
WO2004000789A1 (en) 2003-12-31
AU2003241579B9 (en) 2009-07-30
JP2005529975A (ja) 2005-10-06
US7220880B2 (en) 2007-05-22
AR039684A1 (es) 2005-03-09
CA2488972A1 (en) 2003-12-31
CN1662487A (zh) 2005-08-31
AU2003241579A1 (en) 2004-01-06
TW200406371A (en) 2004-05-01
EP1517882A1 (en) 2005-03-30
AU2003241579B2 (en) 2009-03-19
US20060111406A1 (en) 2006-05-25

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