BR0015523A - Métodos para o tratamento e para a prevenção de condições neurodegenerativas - Google Patents

Métodos para o tratamento e para a prevenção de condições neurodegenerativas

Info

Publication number
BR0015523A
BR0015523A BR0015523-3A BR0015523A BR0015523A BR 0015523 A BR0015523 A BR 0015523A BR 0015523 A BR0015523 A BR 0015523A BR 0015523 A BR0015523 A BR 0015523A
Authority
BR
Brazil
Prior art keywords
treatment
methods
prevention
neurodegenerative conditions
adatanserin
Prior art date
Application number
BR0015523-3A
Other languages
English (en)
Inventor
Magid Abdel-Megid Abou-Gharbia
James Edward Barrett
Wayne Everett Childers Jr
John Allen Moyer
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of BR0015523A publication Critical patent/BR0015523A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Psychology (AREA)
  • Epidemiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Processing Of Meat And Fish (AREA)

Abstract

"MéTODOS PARA O TRATAMENTO E PARA A PREVENçãO DE CONDIçõES NEURODEGENERATIVAS". A adatanserina é útil para o tratamento de distúrbios neurodegenerativos, de dor crónica e de outros distúrbios associados com a liberação disfuncional de glutamato. Os métodos de tratamento dos mesmos compreendem a administração de uma quantidade terapeuticamente eficaz de adatanserina ou de um sal farmacêutico da mesma, a um paciente que necessita do dito tratamento.
BR0015523-3A 1999-11-12 2000-11-10 Métodos para o tratamento e para a prevenção de condições neurodegenerativas BR0015523A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US43921999A 1999-11-12 1999-11-12
PCT/US2000/030973 WO2001034136A2 (en) 1999-11-12 2000-11-10 Use of adatanserin for the treatment of neurodegenerative conditions

Publications (1)

Publication Number Publication Date
BR0015523A true BR0015523A (pt) 2002-10-22

Family

ID=23743796

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0015523-3A BR0015523A (pt) 1999-11-12 2000-11-10 Métodos para o tratamento e para a prevenção de condições neurodegenerativas

Country Status (22)

Country Link
EP (2) EP1242089B1 (pt)
JP (1) JP2003513915A (pt)
KR (1) KR100757226B1 (pt)
CN (1) CN100469368C (pt)
AT (1) ATE291919T1 (pt)
AU (1) AU773733B2 (pt)
BR (1) BR0015523A (pt)
CA (1) CA2390797A1 (pt)
CZ (1) CZ298535B6 (pt)
DE (1) DE60019166T2 (pt)
EA (1) EA006099B1 (pt)
ES (1) ES2235998T3 (pt)
HK (1) HK1046505B (pt)
HU (1) HUP0301847A3 (pt)
IL (1) IL149264A0 (pt)
MX (1) MXPA02004654A (pt)
NO (1) NO322371B1 (pt)
NZ (1) NZ518814A (pt)
PL (1) PL355014A1 (pt)
PT (1) PT1242089E (pt)
WO (1) WO2001034136A2 (pt)
ZA (1) ZA200204682B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1242089B1 (en) * 1999-11-12 2005-03-30 Wyeth Use of adatanserin for the treatment of acute neurodegenerative disorders
EP2236511A4 (en) 2007-12-21 2011-04-13 Alla Chem Llc LIGANDS OF ALPHA ADRENOCEPTORS AND OF DOPAMINE, HISTAMIN, IMIDAZOLIN AND SEROTONIN RECEPTORS AND THEIR APPLICATION THEREOF

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5441961A (en) * 1992-08-27 1995-08-15 Eli Lilly And Company Substituted cyclo or bicycloalkylamides of (8β)-6-(substituted) ergolines
US5877173A (en) * 1996-08-28 1999-03-02 Washington University Preventing neuronal degeneration in Alzheimer's disease
US5902815A (en) * 1996-09-03 1999-05-11 Washington University Use of 5HT-2A serotonin agonists to prevent adverse effects of NMDA receptor hypofunction
EP1242089B1 (en) * 1999-11-12 2005-03-30 Wyeth Use of adatanserin for the treatment of acute neurodegenerative disorders

Also Published As

Publication number Publication date
DE60019166D1 (de) 2005-05-04
ZA200204682B (en) 2003-09-11
PT1242089E (pt) 2005-08-31
NO322371B1 (no) 2006-09-25
AU1656701A (en) 2001-06-06
AU773733B2 (en) 2004-06-03
EP1242089B1 (en) 2005-03-30
CZ20021629A3 (cs) 2003-06-18
IL149264A0 (en) 2002-11-10
HK1046505A1 (en) 2003-01-17
ATE291919T1 (de) 2005-04-15
EP1547597A3 (en) 2006-09-27
JP2003513915A (ja) 2003-04-15
CN1390128A (zh) 2003-01-08
HK1046505B (zh) 2005-06-03
EA006099B1 (ru) 2005-08-25
ES2235998T3 (es) 2005-07-16
EP1242089A2 (en) 2002-09-25
MXPA02004654A (es) 2004-09-10
NO20022187D0 (no) 2002-05-07
EA200200559A1 (ru) 2002-12-26
CA2390797A1 (en) 2001-05-17
KR100757226B1 (ko) 2007-09-11
WO2001034136A2 (en) 2001-05-17
WO2001034136A3 (en) 2002-03-21
CN100469368C (zh) 2009-03-18
NO20022187L (no) 2002-05-07
PL355014A1 (en) 2004-03-22
NZ518814A (en) 2005-08-26
KR20020073132A (ko) 2002-09-19
HUP0301847A2 (hu) 2003-09-29
DE60019166T2 (de) 2006-05-11
HUP0301847A3 (en) 2004-01-28
CZ298535B6 (cs) 2007-10-31
EP1547597A2 (en) 2005-06-29

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: ALTERADA DA INT.CL: A61K 31/506, A61P 25/28

Ipc: A61K 31/00 (2009.01)

B10A Cessation: cessation confirmed

Free format text: HOMOLOGADA A DESISTENCIA DO PEDIDO, REQUERIDA ATRAVES DA PETICAO NO 20090068304/RJ DE 14.07.2009.