BR0014591A - Cloridrato polimórfico de n-[3-[[2-(3, 4-dimetoxifenil) etil] amino ]propil]-4-nitro benzamida - Google Patents

Cloridrato polimórfico de n-[3-[[2-(3, 4-dimetoxifenil) etil] amino ]propil]-4-nitro benzamida

Info

Publication number
BR0014591A
BR0014591A BR0014591-2A BR0014591A BR0014591A BR 0014591 A BR0014591 A BR 0014591A BR 0014591 A BR0014591 A BR 0014591A BR 0014591 A BR0014591 A BR 0014591A
Authority
BR
Brazil
Prior art keywords
polymorphic
dimethoxyphenyl
propyl
ethyl
amino
Prior art date
Application number
BR0014591-2A
Other languages
English (en)
Portuguese (pt)
Inventor
David Busby
Original Assignee
Glaxosmithkline Lab Sas
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Lab Sas, Smithkline Beecham Plc filed Critical Glaxosmithkline Lab Sas
Publication of BR0014591A publication Critical patent/BR0014591A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00Carboxylic acid amides
    • C07C233/64Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/77Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups
    • C07C233/78Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BR0014591-2A 1999-10-08 2000-10-06 Cloridrato polimórfico de n-[3-[[2-(3, 4-dimetoxifenil) etil] amino ]propil]-4-nitro benzamida BR0014591A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9923933.7A GB9923933D0 (en) 1999-10-08 1999-10-08 Novel pharmaceutical
PCT/GB2000/003847 WO2001027071A1 (fr) 1999-10-08 2000-10-06 Hydrochlorure de benzamide n-[3-[[2-(3,4-dimethexyphenyl)ethyl]amino]propyl]-4-nitro polymorphe

Publications (1)

Publication Number Publication Date
BR0014591A true BR0014591A (pt) 2002-06-11

Family

ID=10862442

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0014591-2A BR0014591A (pt) 1999-10-08 2000-10-06 Cloridrato polimórfico de n-[3-[[2-(3, 4-dimetoxifenil) etil] amino ]propil]-4-nitro benzamida

Country Status (18)

Country Link
EP (1) EP1218334A1 (fr)
JP (1) JP2003511437A (fr)
KR (1) KR20020043618A (fr)
CN (1) CN1384817A (fr)
AU (1) AU7546000A (fr)
BR (1) BR0014591A (fr)
CA (1) CA2386845A1 (fr)
CZ (1) CZ20021189A3 (fr)
GB (1) GB9923933D0 (fr)
HK (1) HK1049147A1 (fr)
HU (1) HUP0203582A2 (fr)
IL (1) IL148966A0 (fr)
MX (1) MXPA02003516A (fr)
NO (1) NO20021639L (fr)
PL (1) PL354137A1 (fr)
TR (1) TR200200949T2 (fr)
WO (1) WO2001027071A1 (fr)
ZA (1) ZA200202679B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2664189T3 (es) 2002-01-09 2018-04-18 Emisphere Technologies, Inc. Polimorfos de 4-(4-cloro-2-hidroxibenzoil)aminobutanoato de sodio
KR101125932B1 (ko) * 2006-12-06 2012-03-22 아이디유엔 파마슈티칼즈, 인코포레이티드 (3s)-3-[n-(n'-(2-tert-부틸페닐)옥사밀)알라니닐]아미노-5-(2',3',5',6'-테트라플루오로페녹시)-4-옥소펜탄산의 결정 형태

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2726267B1 (fr) * 1994-10-26 1998-01-02 Smithkline Beecham Lab Nouveaux agents anti-arythmiques, compositions pharmaceutiques les contenant, et procede pour les preparer
GB9706376D0 (en) * 1997-03-27 1997-05-14 Smithkline Beecham Plc Novel pharmaceutical

Also Published As

Publication number Publication date
TR200200949T2 (tr) 2002-08-21
JP2003511437A (ja) 2003-03-25
EP1218334A1 (fr) 2002-07-03
WO2001027071A1 (fr) 2001-04-19
CZ20021189A3 (cs) 2002-09-11
GB9923933D0 (en) 1999-12-08
IL148966A0 (en) 2002-11-10
MXPA02003516A (es) 2004-09-10
HUP0203582A2 (en) 2004-03-01
PL354137A1 (en) 2003-12-29
NO20021639L (no) 2002-05-30
ZA200202679B (en) 2003-05-28
HK1049147A1 (zh) 2003-05-02
CA2386845A1 (fr) 2001-04-19
NO20021639D0 (no) 2002-04-05
AU7546000A (en) 2001-04-23
CN1384817A (zh) 2002-12-11
KR20020043618A (ko) 2002-06-10

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]