BG35042A3 - Method for preparing benzodiazepinic compounds - Google Patents

Method for preparing benzodiazepinic compounds

Info

Publication number
BG35042A3
BG35042A3 BG057344A BG5734480A BG35042A3 BG 35042 A3 BG35042 A3 BG 35042A3 BG 057344 A BG057344 A BG 057344A BG 5734480 A BG5734480 A BG 5734480A BG 35042 A3 BG35042 A3 BG 35042A3
Authority
BG
Bulgaria
Prior art keywords
benzodiazepinic
preparing
compounds
formulated
demonstrated
Prior art date
Application number
BG057344A
Other languages
Bulgarian (bg)
English (en)
Inventor
Jiban Chakrabarti
Terrence Hotten
Original Assignee
Lilly Industries Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Industries Limited filed Critical Lilly Industries Limited
Publication of BG35042A3 publication Critical patent/BG35042A3/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
BG057344A 1979-10-16 1980-10-15 Method for preparing benzodiazepinic compounds BG35042A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7935846 1979-10-16

Publications (1)

Publication Number Publication Date
BG35042A3 true BG35042A3 (en) 1983-01-16

Family

ID=10508540

Family Applications (2)

Application Number Title Priority Date Filing Date
BG057344A BG35042A3 (en) 1979-10-16 1980-10-15 Method for preparing benzodiazepinic compounds
BG049366A BG34907A3 (en) 1979-10-16 1980-10-15 Method for preparing benzodiazepine compounds

Family Applications After (1)

Application Number Title Priority Date Filing Date
BG049366A BG34907A3 (en) 1979-10-16 1980-10-15 Method for preparing benzodiazepine compounds

Country Status (33)

Country Link
US (3) US4404137A (OSRAM)
EP (1) EP0027390B1 (OSRAM)
JP (1) JPS5663987A (OSRAM)
KR (2) KR850000471B1 (OSRAM)
AR (2) AR228041A1 (OSRAM)
AT (1) AT373889B (OSRAM)
AU (1) AU538500B2 (OSRAM)
BE (1) BE885729A (OSRAM)
BG (2) BG35042A3 (OSRAM)
CA (1) CA1159056A (OSRAM)
CH (1) CH646700A5 (OSRAM)
CS (1) CS244409B2 (OSRAM)
DD (1) DD153692A5 (OSRAM)
DE (1) DE3068706D1 (OSRAM)
DK (1) DK437480A (OSRAM)
ES (1) ES495948A0 (OSRAM)
FI (1) FI67550C (OSRAM)
FR (1) FR2467851A1 (OSRAM)
GB (1) GB8327127D0 (OSRAM)
GR (1) GR70720B (OSRAM)
HU (1) HU182213B (OSRAM)
IE (1) IE50358B1 (OSRAM)
IL (1) IL61264A (OSRAM)
IT (1) IT1143047B (OSRAM)
LU (1) LU82853A1 (OSRAM)
MX (1) MX6233E (OSRAM)
NZ (1) NZ195248A (OSRAM)
PH (2) PH16288A (OSRAM)
PL (2) PL126824B1 (OSRAM)
PT (1) PT71913B (OSRAM)
RO (2) RO81351B (OSRAM)
YU (1) YU261580A (OSRAM)
ZA (1) ZA806342B (OSRAM)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4404137A (en) * 1979-10-16 1983-09-13 Lilly Industries Limited Pyrazolo [3,4-b][1,5]benzodiazepine compounds
US4431589A (en) * 1980-12-11 1984-02-14 Lilly House Benzodiazepine compounds and their use as pharmaceuticals
US4596799A (en) * 1985-01-29 1986-06-24 Ciba-Geigy Corporation 9H-pyrrolo[2,1-c]-1,2,4-triazolo[4,3-a][1,4]benzodiazepines
TW219896B (OSRAM) * 1988-07-07 1994-02-01 Duphar Int Res
GB8819059D0 (en) * 1988-08-11 1988-09-14 Lilly Industries Ltd Benzodiazepine compounds & their use as pharmaceuticals
US5637584A (en) * 1995-03-24 1997-06-10 Eli Lilly And Company Solvate of olanzapine
US5631250A (en) * 1995-03-24 1997-05-20 Eli Lilly And Company Process and solvate of 2-methyl-thieno-benzodiazepine
US20050250767A1 (en) * 2003-01-23 2005-11-10 Weiner David M Use of N-desmethylclozapine to treat human neuropsychiatric disease
NZ541014A (en) * 2003-01-23 2008-05-30 Acadia Pharm Inc Use of N-desmethylclozapine to treat schizophrenia while increasing the level of activity of a muscarinic receptor
US20050085463A1 (en) * 2003-01-23 2005-04-21 Weiner David M. Use of N-desmethylclozapine to treat human neuropsychiatric disease
ATE426405T1 (de) * 2003-12-22 2009-04-15 Acadia Pharm Inc Amino-substituierte diarylaa,ducyclohepten- analoga als muscarinische agonisten und verfahren zur behandlung von neuropsychiatrischen erkrankungen
CA2560671A1 (en) * 2004-04-01 2006-01-05 Acadia Pharmaceuticals Inc. Crystalline forms of n-desmethylclozapine
US20070105836A1 (en) * 2005-10-31 2007-05-10 Lars Pettersson Prodrugs of muscarinic agonists and methods of treatment of neuropsychiatric disorders
JP5438482B2 (ja) * 2009-12-03 2014-03-12 Ｊｕｋｉ株式会社 ミシン、ミシンの縫製データ編集装置及びミシンの縫製データ編集プログラム

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3450694A (en) * 1966-02-23 1969-06-17 Abbott Lab Substituted benzoxazepines and benzothiazepines
US3758479A (en) * 1967-03-22 1973-09-11 Sandoz Ag Nitro and sulphamoyl substituted dibenzodiazepines
DE1795183B1 (de) * 1968-08-20 1972-07-20 Thomae Gmbh Dr K 5,11-Dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-on-derivate und Arzneimittel
CA918659A (en) * 1969-07-31 1973-01-09 Yoshitomi Pharmaceutical Industries 11-(4-substituted-1-piperazinyl)-dibenzo (b,f) (1,4) thiazepines
US4115568A (en) * 1974-11-26 1978-09-19 Lilly Industries Limited Thieno[3,2-b]-[1,5]benzodiazepines
US4172831A (en) * 1974-11-26 1979-10-30 Lilly Industries Limited Thieno-benzodiazepines
US3953430A (en) * 1975-02-24 1976-04-27 American Cyanamid Company Substituted benzodiazepin-10-ones and method of use
US3951981A (en) * 1975-02-24 1976-04-20 American Cyanamid Company Substituted benzodiazepines and method of use
DE2707270A1 (de) * 1977-02-19 1978-08-24 Hoechst Ag Pyrazolo-diazepine und verfahren zu ihrer herstellung
DE2707269A1 (de) * 1977-02-19 1978-08-24 Hoechst Ag Heterocyclische stickstoffverbindungen und verfahren zu ihrer herstellung
US4097597A (en) * 1977-02-23 1978-06-27 Abbott Laboratories Dibenzo b,e! 1,4!diazepines
IT7851496A0 (it) * 1977-10-31 1978-10-13 Sandoz Ag Menti pirazinobenzossazepine loro preparazione e loro impiego quali medica
CH643263A5 (de) * 1979-05-11 1984-05-30 Sandoz Ag Benzodiazepine, ihre herstellung und verwendung.
NZ194529A (en) * 1979-08-03 1983-05-10 Byk Gulden Lomberg Chem Fab 9,10-dihydro-1h, 4h-pyrazolo (4,3-b)(1,5)benzodiazepin-10-ones
US4404137A (en) * 1979-10-16 1983-09-13 Lilly Industries Limited Pyrazolo [3,4-b][1,5]benzodiazepine compounds

Also Published As

Publication number Publication date
DK437480A (da) 1981-04-17
ATA510180A (de) 1983-07-15
CS244409B2 (en) 1986-07-17
NZ195248A (en) 1983-11-18
PL227306A1 (OSRAM) 1981-09-18
KR830004300A (ko) 1983-07-09
FR2467851A1 (fr) 1981-04-30
KR850000471B1 (ko) 1985-04-08
PH16288A (en) 1983-09-05
AU6325280A (en) 1981-04-30
RO85822B (ro) 1984-11-30
JPS5663987A (en) 1981-05-30
DD153692A5 (de) 1982-01-27
ES8106905A1 (es) 1981-09-16
IL61264A (en) 1985-08-30
PT71913B (en) 1981-08-31
IT8049899A0 (it) 1980-10-14
US4486591A (en) 1984-12-04
PH17759A (en) 1984-12-05
PT71913A (en) 1980-11-01
RO81351A (ro) 1983-02-15
ZA806342B (en) 1982-05-26
AT373889B (de) 1984-02-27
BG34907A3 (en) 1983-12-15
AR228041A1 (es) 1983-01-14
LU82853A1 (fr) 1982-05-10
RO81351B (ro) 1983-02-28
KR850000472B1 (ko) 1985-04-08
RO85822A (ro) 1984-11-25
KR850001463A (ko) 1985-03-18
CH646700A5 (fr) 1984-12-14
GB8327127D0 (en) 1983-11-09
PL126824B1 (en) 1983-09-30
FI67550C (fi) 1985-04-10
IT1143047B (it) 1986-10-22
AU538500B2 (en) 1984-08-16
US4542131A (en) 1985-09-17
PL231270A1 (OSRAM) 1981-12-23
IE802135L (en) 1981-04-16
ES495948A0 (es) 1981-09-16
EP0027390B1 (en) 1984-07-25
FR2467851B1 (OSRAM) 1985-04-05
MX6233E (es) 1985-01-14
HU182213B (en) 1983-12-28
DE3068706D1 (en) 1984-08-30
AR228101A1 (es) 1983-01-14
FI803253L (fi) 1981-04-17
IL61264A0 (en) 1980-12-31
IE50358B1 (en) 1986-04-02
PL135044B1 (en) 1985-09-30
YU261580A (en) 1983-12-31
CA1159056A (en) 1983-12-20
GR70720B (OSRAM) 1983-01-18
EP0027390A1 (en) 1981-04-22
FI67550B (fi) 1984-12-31
BE885729A (fr) 1981-04-15
US4404137A (en) 1983-09-13

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