BG108554A - Метод за получаване на 5-заместени изобензофурани - Google Patents

Метод за получаване на 5-заместени изобензофурани Download PDF

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Publication number
BG108554A
BG108554A BG108554A BG10855404A BG108554A BG 108554 A BG108554 A BG 108554A BG 108554 A BG108554 A BG 108554A BG 10855404 A BG10855404 A BG 10855404A BG 108554 A BG108554 A BG 108554A
Authority
BG
Bulgaria
Prior art keywords
formula
group
triphenylmethyl
citalopram
alkyl
Prior art date
Application number
BG108554A
Other languages
Bulgarian (bg)
English (en)
Inventor
Leone Dall'asta
Giovanni Coticelli
Original Assignee
Infosint Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Infosint Sa filed Critical Infosint Sa
Publication of BG108554A publication Critical patent/BG108554A/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/48—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups bound to a carbon atom of a six-membered aromatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BG108554A 2001-08-02 2004-01-30 Метод за получаване на 5-заместени изобензофурани BG108554A (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP01830517A EP1281707B1 (en) 2001-08-02 2001-08-02 Process for the preparation of 5-subtituted isobenzofurans

Publications (1)

Publication Number Publication Date
BG108554A true BG108554A (bg) 2005-03-31

Family

ID=8184643

Family Applications (1)

Application Number Title Priority Date Filing Date
BG108554A BG108554A (bg) 2001-08-02 2004-01-30 Метод за получаване на 5-заместени изобензофурани

Country Status (23)

Country Link
US (1) US7166729B2 (zh)
EP (1) EP1281707B1 (zh)
JP (1) JP2005501056A (zh)
KR (1) KR20040043176A (zh)
CN (1) CN1298713C (zh)
AR (1) AR036212A1 (zh)
AT (1) ATE286037T1 (zh)
AU (1) AU2002325385B2 (zh)
BG (1) BG108554A (zh)
BR (1) BR0211858A (zh)
CA (1) CA2456004A1 (zh)
DE (1) DE60108105T2 (zh)
DK (1) DK1281707T3 (zh)
ES (1) ES2234797T3 (zh)
HK (1) HK1070357A1 (zh)
HU (1) HUP0401166A3 (zh)
MX (1) MXPA04001030A (zh)
PL (1) PL368320A1 (zh)
PT (1) PT1281707E (zh)
RO (1) RO122147B1 (zh)
TW (1) TWI225055B (zh)
WO (1) WO2003011846A2 (zh)
ZA (1) ZA200400841B (zh)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IS7239A (is) * 2001-12-14 2004-04-29 H. Lundbeck A/S Aðferð til framleiðslu á essítalóprami
AU2003263155A1 (en) * 2002-09-20 2004-04-08 H. Lundbeck A/S Method for manufacture of dihydroisobenzofuran derivatives
GB0601286D0 (en) 2006-01-23 2006-03-01 Sandoz Ag Asymmetric synthesis
CA2932121A1 (en) 2007-11-30 2009-06-11 Newlink Genetics Corporation Ido inhibitors
CN106632182A (zh) * 2016-12-07 2017-05-10 万全万特制药（厦门）有限公司 草酸艾司西酞普兰脱甲基杂质的制备方法
DE112019006382T8 (de) * 2018-12-22 2021-12-09 Malladi Drugs And Pharmaceuticals Ltd. NEUES VERFAHREN ZUR HERSTELLUNG VONR-PHENYLACETYLCARBINOL UND β-AMINOALKOHOLEN

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8419963D0 (en) * 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) * 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
NZ501737A (en) * 1997-07-08 2001-10-26 H Method for the preparation of citalopram using Grignard reagent 4-halogen-fluorophenyl and 3-halogen-N,N-dimethyl-propylamine
CZ296537B6 (cs) * 1999-04-14 2006-04-12 H. Lundbeck A/S Zpusob výroby citalopramu a meziprodukty
ITMI991486A1 (it) * 1999-07-06 2001-01-06 Vis Farmaceutici S P A Processo per la sintesi di citalopram
IES20010143A2 (en) * 2000-02-24 2001-07-25 Lundbeck & Co As H Method for the preparation of citalopram
IT1319686B1 (it) * 2000-12-12 2003-10-23 C D Farmasint S R L Procedimento di preparazione di citalopram.

Also Published As

Publication number Publication date
AU2002325385B8 (en) 2003-02-17
PT1281707E (pt) 2005-04-29
HK1070357A1 (en) 2005-06-17
KR20040043176A (ko) 2004-05-22
EP1281707B1 (en) 2004-12-29
ES2234797T3 (es) 2005-07-01
US20040230065A1 (en) 2004-11-18
AR036212A1 (es) 2004-08-18
DE60108105T2 (de) 2005-12-08
TWI225055B (en) 2004-12-11
PL368320A1 (en) 2005-03-21
WO2003011846A3 (en) 2003-11-27
AU2002325385B2 (en) 2007-07-05
DE60108105D1 (de) 2005-02-03
WO2003011846B1 (en) 2003-12-24
US7166729B2 (en) 2007-01-23
BR0211858A (pt) 2004-09-21
CA2456004A1 (en) 2003-02-13
DK1281707T3 (da) 2005-05-02
ATE286037T1 (de) 2005-01-15
WO2003011846A2 (en) 2003-02-13
MXPA04001030A (es) 2004-12-03
EP1281707A1 (en) 2003-02-05
CN1298713C (zh) 2007-02-07
ZA200400841B (en) 2005-02-02
CN1555370A (zh) 2004-12-15
JP2005501056A (ja) 2005-01-13
HUP0401166A2 (hu) 2004-09-28
RO122147B1 (ro) 2009-01-30
HUP0401166A3 (en) 2007-05-29

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