BG108370A - Кристални форми на азитромицин - Google Patents

Кристални форми на азитромицин Download PDF

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Publication number
BG108370A
BG108370A BG108370A BG10837003A BG108370A BG 108370 A BG108370 A BG 108370A BG 108370 A BG108370 A BG 108370A BG 10837003 A BG10837003 A BG 10837003A BG 108370 A BG108370 A BG 108370A
Authority
BG
Bulgaria
Prior art keywords
azithromycin
ppm
peaks
crystalline
solid
Prior art date
Application number
BG108370A
Other languages
Bulgarian (bg)
English (en)
Inventor
Zheng Li
Andrew Trask
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27404135&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG108370(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of BG108370A publication Critical patent/BG108370A/bg

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682Processes
    • A61K9/1688Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2813Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/282Organic compounds, e.g. fats
    • A61K9/2826Sugars or sugar alcohols, e.g. sucrose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
BG108370A 2001-05-22 2003-11-18 Кристални форми на азитромицин BG108370A (bg)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29256501P 2001-05-22 2001-05-22
US29774101P 2001-06-12 2001-06-12
US34304101P 2001-12-21 2001-12-21

Publications (1)

Publication Number Publication Date
BG108370A true BG108370A (bg) 2004-11-30

Family

ID=27404135

Family Applications (1)

Application Number Title Priority Date Filing Date
BG108370A BG108370A (bg) 2001-05-22 2003-11-18 Кристални форми на азитромицин

Country Status (35)

Country Link
US (10) US6977243B2 (enExample)
EP (1) EP1390377B1 (enExample)
JP (3) JP2004530703A (enExample)
KR (1) KR100574153B1 (enExample)
AP (1) AP2003002906A0 (enExample)
AR (1) AR036022A1 (enExample)
AT (2) ATE319730T1 (enExample)
AU (1) AU2002256846B2 (enExample)
BG (1) BG108370A (enExample)
BR (1) BR0209918A (enExample)
CA (1) CA2391659C (enExample)
CR (1) CR7159A (enExample)
CZ (1) CZ20033154A3 (enExample)
DE (2) DE60228345D1 (enExample)
DK (1) DK1390377T3 (enExample)
EA (2) EA009611B1 (enExample)
EE (1) EE200300575A (enExample)
ES (2) ES2258142T3 (enExample)
GE (1) GEP20084399B (enExample)
HU (1) HUP0400446A2 (enExample)
IL (1) IL158591A0 (enExample)
IS (1) IS7007A (enExample)
MA (1) MA27023A1 (enExample)
MX (1) MXPA03010028A (enExample)
MY (1) MY129319A (enExample)
NO (2) NO321894B1 (enExample)
NZ (2) NZ539801A (enExample)
PA (1) PA8545701A1 (enExample)
PE (1) PE20021064A1 (enExample)
PL (1) PL367091A1 (enExample)
PT (1) PT1390377E (enExample)
SK (1) SK14402003A3 (enExample)
TN (1) TNSN03121A1 (enExample)
WO (1) WO2002094843A1 (enExample)
YU (1) YU91603A (enExample)

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Publication number Publication date
HUP0400446A2 (hu) 2004-09-28
SK14402003A3 (sk) 2004-06-08
AP2003002906A0 (en) 2003-12-31
EA200500630A1 (ru) 2006-02-24
CA2391659C (en) 2006-05-30
CZ20033154A3 (en) 2004-04-14
PL367091A1 (en) 2005-02-21
WO2002094843A1 (en) 2002-11-28
US7309782B2 (en) 2007-12-18
MA27023A1 (fr) 2004-12-20
AR036022A1 (es) 2004-08-04
PE20021064A1 (es) 2002-11-21
PA8545701A1 (es) 2003-09-05
US20050192234A1 (en) 2005-09-01
IS7007A (is) 2003-10-30
KR20040014525A (ko) 2004-02-14
JP2006152002A (ja) 2006-06-15
CR7159A (es) 2004-02-23
US7081525B2 (en) 2006-07-25
US20050256062A1 (en) 2005-11-17
US20040043944A1 (en) 2004-03-04
NO20035177D0 (no) 2003-11-21
EA009611B1 (ru) 2008-02-28
NO321894B1 (no) 2006-07-17
US6977243B2 (en) 2005-12-20
EA007618B1 (ru) 2006-12-29
DK1390377T3 (da) 2006-06-19
US20030162730A1 (en) 2003-08-28
KR100574153B1 (ko) 2006-04-25
US20050256063A1 (en) 2005-11-17
US20040043945A1 (en) 2004-03-04
JP4584162B2 (ja) 2010-11-17
ATE404575T1 (de) 2008-08-15
ES2258142T3 (es) 2006-08-16
PT1390377E (pt) 2006-06-30
EA200301115A1 (ru) 2004-04-29
BR0209918A (pt) 2004-03-30
MY129319A (en) 2007-03-30
US7053192B2 (en) 2006-05-30
US7307156B2 (en) 2007-12-11
NZ539801A (en) 2006-10-27
NO20061049L (no) 2003-05-12
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US20040138149A1 (en) 2004-07-15
YU91603A (sh) 2006-08-17
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ATE319730T1 (de) 2006-03-15
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ES2310886T3 (es) 2009-01-16
US7282486B2 (en) 2007-10-16
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AU2002256846B2 (en) 2007-04-05
MXPA03010028A (es) 2004-02-12
JP2007161726A (ja) 2007-06-28
US20040082527A1 (en) 2004-04-29
TNSN03121A1 (en) 2005-12-23
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EE200300575A (et) 2004-04-15

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