BG108324A - Нафтотиазин положителни алостерични модулатори на амра - рецептор - Google Patents
Нафтотиазин положителни алостерични модулатори на амра - рецептор Download PDFInfo
- Publication number
- BG108324A BG108324A BG108324A BG10832403A BG108324A BG 108324 A BG108324 A BG 108324A BG 108324 A BG108324 A BG 108324A BG 10832403 A BG10832403 A BG 10832403A BG 108324 A BG108324 A BG 108324A
- Authority
- BG
- Bulgaria
- Prior art keywords
- alkyl
- different
- halogen atoms
- optionally substituted
- general formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10123952A DE10123952A1 (de) | 2001-05-17 | 2001-05-17 | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG108324A true BG108324A (bg) | 2004-12-30 |
Family
ID=7685080
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG108324A Pending BG108324A (bg) | 2001-05-17 | 2003-11-07 | Нафтотиазин положителни алостерични модулатори на амра - рецептор |
Country Status (26)
| Country | Link |
|---|---|
| EP (1) | EP1404340A1 (no) |
| JP (1) | JP2004529980A (no) |
| KR (1) | KR20040007572A (no) |
| CN (1) | CN1533278A (no) |
| AR (1) | AR036332A1 (no) |
| BG (1) | BG108324A (no) |
| BR (1) | BR0209796A (no) |
| CA (1) | CA2449189A1 (no) |
| CO (1) | CO5550460A2 (no) |
| CZ (1) | CZ20033112A3 (no) |
| DE (1) | DE10123952A1 (no) |
| EA (1) | EA006608B1 (no) |
| EC (1) | ECSP034852A (no) |
| EE (1) | EE200300566A (no) |
| HR (1) | HRP20030933A2 (no) |
| HU (1) | HUP0401273A3 (no) |
| IL (1) | IL158642A0 (no) |
| MX (1) | MXPA03010373A (no) |
| NO (1) | NO20035088L (no) |
| NZ (1) | NZ530154A (no) |
| PL (1) | PL364053A1 (no) |
| SK (1) | SK14222003A3 (no) |
| UY (1) | UY27290A1 (no) |
| WO (1) | WO2002100411A1 (no) |
| YU (1) | YU90403A (no) |
| ZA (1) | ZA200308466B (no) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2009002180A (es) * | 2006-08-31 | 2009-06-05 | Univ Alberta | Metodo de inhibicion de la depresion respiratoria mediante el uso de moduladores alostericos positivos del receptor ampa. |
| CN111518058B (zh) * | 2020-05-29 | 2021-03-09 | 四川大学华西医院 | 一种噁噻嗪类化合物及其用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU4345297A (en) * | 1996-09-17 | 1998-04-14 | Regents Of The University Of California, The | Benzothiadiazide derivatives and their use as allosteric up-modulators of the ampa receptor |
| AU4711899A (en) * | 1998-06-25 | 2000-01-10 | Merck & Co., Inc. | Naphtho(1,8-de)thiasin-2-yl methyl carbapenem antibacterials |
| DE10004572A1 (de) * | 2000-02-02 | 2001-08-09 | Boehringer Ingelheim Pharma | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
-
2001
- 2001-05-17 DE DE10123952A patent/DE10123952A1/de not_active Withdrawn
-
2002
- 2002-05-15 BR BR0209796-6A patent/BR0209796A/pt not_active Expired - Fee Related
- 2002-05-15 YU YU90403A patent/YU90403A/sh unknown
- 2002-05-15 CA CA002449189A patent/CA2449189A1/en not_active Abandoned
- 2002-05-15 EE EEP200300566A patent/EE200300566A/xx unknown
- 2002-05-15 KR KR10-2003-7014965A patent/KR20040007572A/ko not_active Application Discontinuation
- 2002-05-15 EP EP02750931A patent/EP1404340A1/en not_active Withdrawn
- 2002-05-15 EA EA200301167A patent/EA006608B1/ru not_active IP Right Cessation
- 2002-05-15 JP JP2003503232A patent/JP2004529980A/ja not_active Abandoned
- 2002-05-15 MX MXPA03010373A patent/MXPA03010373A/es unknown
- 2002-05-15 UY UY27290A patent/UY27290A1/es not_active Application Discontinuation
- 2002-05-15 HU HU0401273A patent/HUP0401273A3/hu unknown
- 2002-05-15 SK SK1422-2003A patent/SK14222003A3/sk unknown
- 2002-05-15 NZ NZ530154A patent/NZ530154A/en unknown
- 2002-05-15 WO PCT/EP2002/005338 patent/WO2002100411A1/en not_active Application Discontinuation
- 2002-05-15 CZ CZ20033112A patent/CZ20033112A3/cs unknown
- 2002-05-15 IL IL15864202A patent/IL158642A0/xx unknown
- 2002-05-15 PL PL02364053A patent/PL364053A1/xx not_active Application Discontinuation
- 2002-05-15 CN CNA028100832A patent/CN1533278A/zh active Pending
- 2002-05-17 AR ARP020101827A patent/AR036332A1/es not_active Suspension/Interruption
-
2003
- 2003-10-30 ZA ZA200308466A patent/ZA200308466B/en unknown
- 2003-11-07 BG BG108324A patent/BG108324A/bg active Pending
- 2003-11-14 NO NO20035088A patent/NO20035088L/no not_active Application Discontinuation
- 2003-11-14 HR HR20030933A patent/HRP20030933A2/xx not_active Application Discontinuation
- 2003-11-17 EC EC2003004852A patent/ECSP034852A/es unknown
- 2003-12-01 CO CO03105591A patent/CO5550460A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2002100411A1 (en) | 2002-12-19 |
| KR20040007572A (ko) | 2004-01-24 |
| ECSP034852A (es) | 2003-12-24 |
| SK14222003A3 (sk) | 2004-05-04 |
| DE10123952A1 (de) | 2002-11-21 |
| EP1404340A1 (en) | 2004-04-07 |
| IL158642A0 (en) | 2004-05-12 |
| HRP20030933A2 (en) | 2004-04-30 |
| NO20035088D0 (no) | 2003-11-14 |
| NO20035088L (no) | 2003-11-14 |
| PL364053A1 (en) | 2004-12-13 |
| HUP0401273A3 (en) | 2006-11-28 |
| YU90403A (sh) | 2006-05-25 |
| BR0209796A (pt) | 2004-06-01 |
| MXPA03010373A (es) | 2004-03-16 |
| JP2004529980A (ja) | 2004-09-30 |
| CA2449189A1 (en) | 2002-12-19 |
| EA006608B1 (ru) | 2006-02-24 |
| EE200300566A (et) | 2004-02-16 |
| HUP0401273A2 (hu) | 2004-10-28 |
| ZA200308466B (en) | 2004-05-24 |
| CZ20033112A3 (en) | 2004-03-17 |
| NZ530154A (en) | 2005-09-30 |
| AR036332A1 (es) | 2004-09-01 |
| UY27290A1 (es) | 2002-12-31 |
| CN1533278A (zh) | 2004-09-29 |
| CO5550460A2 (es) | 2005-08-31 |
| EA200301167A1 (ru) | 2004-06-24 |
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