YU90403A - Naftotiazinski pozitivno alosterični modulatori ampa receptora (paarm) - Google Patents
Naftotiazinski pozitivno alosterični modulatori ampa receptora (paarm)Info
- Publication number
- YU90403A YU90403A YU90403A YUP90403A YU90403A YU 90403 A YU90403 A YU 90403A YU 90403 A YU90403 A YU 90403A YU P90403 A YUP90403 A YU P90403A YU 90403 A YU90403 A YU 90403A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- receptor modulators
- paarm
- naphtothiazine
- positive allosteric
- ampa receptor
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Abstract
Ovaj pronalazak odnosi se na nove pozitivno alosterične modulatore AMPA receptora, opšte formule (I), u kojoj R1, R2, R3, R4 i R5 mogu da imaju značenja data u opisu i patentnim zahtevima, na postupke za njihovo pripremanje i na njihovu primenu kao farmaceutskih preparata.[The present invention relates to new positive allosteric AMPA-receptor modulators of general formula (I), wherein R1, R2, R3, R4 and R5 may have the meanings given in the specification and claims, processes for preparing them and the use thereof as pharmaceutical compositions.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10123952A DE10123952A1 (de) | 2001-05-17 | 2001-05-17 | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| YU90403A true YU90403A (sh) | 2006-05-25 |
Family
ID=7685080
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| YU90403A YU90403A (sh) | 2001-05-17 | 2002-05-15 | Naftotiazinski pozitivno alosterični modulatori ampa receptora (paarm) |
Country Status (26)
| Country | Link |
|---|---|
| EP (1) | EP1404340A1 (sh) |
| JP (1) | JP2004529980A (sh) |
| KR (1) | KR20040007572A (sh) |
| CN (1) | CN1533278A (sh) |
| AR (1) | AR036332A1 (sh) |
| BG (1) | BG108324A (sh) |
| BR (1) | BR0209796A (sh) |
| CA (1) | CA2449189A1 (sh) |
| CO (1) | CO5550460A2 (sh) |
| CZ (1) | CZ20033112A3 (sh) |
| DE (1) | DE10123952A1 (sh) |
| EA (1) | EA006608B1 (sh) |
| EC (1) | ECSP034852A (sh) |
| EE (1) | EE200300566A (sh) |
| HR (1) | HRP20030933A2 (sh) |
| HU (1) | HUP0401273A3 (sh) |
| IL (1) | IL158642A0 (sh) |
| MX (1) | MXPA03010373A (sh) |
| NO (1) | NO20035088L (sh) |
| NZ (1) | NZ530154A (sh) |
| PL (1) | PL364053A1 (sh) |
| SK (1) | SK14222003A3 (sh) |
| UY (1) | UY27290A1 (sh) |
| WO (1) | WO2002100411A1 (sh) |
| YU (1) | YU90403A (sh) |
| ZA (1) | ZA200308466B (sh) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20090047534A (ko) * | 2006-08-31 | 2009-05-12 | 더 거버너스 오브 더 유니버시티 오브 앨버타 | 양성 알로스테릭 ａｍｐａ 수용체 조절인자를 사용하여 호흡 저하를 억제하는 방법 |
| CN111518058B (zh) * | 2020-05-29 | 2021-03-09 | 四川大学华西医院 | 一种噁噻嗪类化合物及其用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU4345297A (en) * | 1996-09-17 | 1998-04-14 | Regents Of The University Of California, The | Benzothiadiazide derivatives and their use as allosteric up-modulators of the ampa receptor |
| JP2002518498A (ja) * | 1998-06-25 | 2002-06-25 | メルク エンド カムパニー インコーポレーテッド | ナフト［１，８−ｄｅ］チアジン−２−イルメチルカルバペネム抗菌物質 |
| DE10004572A1 (de) * | 2000-02-02 | 2001-08-09 | Boehringer Ingelheim Pharma | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
-
2001
- 2001-05-17 DE DE10123952A patent/DE10123952A1/de not_active Withdrawn
-
2002
- 2002-05-15 BR BR0209796-6A patent/BR0209796A/pt not_active Expired - Fee Related
- 2002-05-15 IL IL15864202A patent/IL158642A0/xx unknown
- 2002-05-15 MX MXPA03010373A patent/MXPA03010373A/es unknown
- 2002-05-15 HU HU0401273A patent/HUP0401273A3/hu unknown
- 2002-05-15 EE EEP200300566A patent/EE200300566A/xx unknown
- 2002-05-15 PL PL02364053A patent/PL364053A1/xx not_active Application Discontinuation
- 2002-05-15 YU YU90403A patent/YU90403A/sh unknown
- 2002-05-15 EA EA200301167A patent/EA006608B1/ru not_active IP Right Cessation
- 2002-05-15 CZ CZ20033112A patent/CZ20033112A3/cs unknown
- 2002-05-15 CA CA002449189A patent/CA2449189A1/en not_active Abandoned
- 2002-05-15 EP EP02750931A patent/EP1404340A1/en not_active Withdrawn
- 2002-05-15 CN CNA028100832A patent/CN1533278A/zh active Pending
- 2002-05-15 JP JP2003503232A patent/JP2004529980A/ja not_active Abandoned
- 2002-05-15 KR KR10-2003-7014965A patent/KR20040007572A/ko not_active Application Discontinuation
- 2002-05-15 NZ NZ530154A patent/NZ530154A/en unknown
- 2002-05-15 WO PCT/EP2002/005338 patent/WO2002100411A1/en not_active Application Discontinuation
- 2002-05-15 SK SK1422-2003A patent/SK14222003A3/sk unknown
- 2002-05-15 UY UY27290A patent/UY27290A1/es not_active Application Discontinuation
- 2002-05-17 AR ARP020101827A patent/AR036332A1/es not_active Suspension/Interruption
-
2003
- 2003-10-30 ZA ZA200308466A patent/ZA200308466B/en unknown
- 2003-11-07 BG BG108324A patent/BG108324A/bg active Pending
- 2003-11-14 HR HR20030933A patent/HRP20030933A2/xx not_active Application Discontinuation
- 2003-11-14 NO NO20035088A patent/NO20035088L/no not_active Application Discontinuation
- 2003-11-17 EC EC2003004852A patent/ECSP034852A/es unknown
- 2003-12-01 CO CO03105591A patent/CO5550460A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN1533278A (zh) | 2004-09-29 |
| SK14222003A3 (sk) | 2004-05-04 |
| AR036332A1 (es) | 2004-09-01 |
| NZ530154A (en) | 2005-09-30 |
| ZA200308466B (en) | 2004-05-24 |
| MXPA03010373A (es) | 2004-03-16 |
| CZ20033112A3 (en) | 2004-03-17 |
| CO5550460A2 (es) | 2005-08-31 |
| BG108324A (bg) | 2004-12-30 |
| HUP0401273A2 (hu) | 2004-10-28 |
| IL158642A0 (en) | 2004-05-12 |
| CA2449189A1 (en) | 2002-12-19 |
| KR20040007572A (ko) | 2004-01-24 |
| HRP20030933A2 (en) | 2004-04-30 |
| ECSP034852A (es) | 2003-12-24 |
| PL364053A1 (en) | 2004-12-13 |
| JP2004529980A (ja) | 2004-09-30 |
| NO20035088D0 (no) | 2003-11-14 |
| NO20035088L (no) | 2003-11-14 |
| UY27290A1 (es) | 2002-12-31 |
| EA200301167A1 (ru) | 2004-06-24 |
| BR0209796A (pt) | 2004-06-01 |
| EP1404340A1 (en) | 2004-04-07 |
| DE10123952A1 (de) | 2002-11-21 |
| EE200300566A (et) | 2004-02-16 |
| WO2002100411A1 (en) | 2002-12-19 |
| HUP0401273A3 (en) | 2006-11-28 |
| EA006608B1 (ru) | 2006-02-24 |
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