BG104048A - Състав съдържащ 5-/4-/2-(n-метил-n-2-пиридил) амино)- етокси/ бензин/ тиазолидин-2,4-дион - Google Patents

Състав съдържащ 5-/4-/2-(n-метил-n-2-пиридил) амино)- етокси/ бензин/ тиазолидин-2,4-дион Download PDF

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Publication number
BG104048A
BG104048A BG104048A BG10404899A BG104048A BG 104048 A BG104048 A BG 104048A BG 104048 A BG104048 A BG 104048A BG 10404899 A BG10404899 A BG 10404899A BG 104048 A BG104048 A BG 104048A
Authority
BG
Bulgaria
Prior art keywords
pharmaceutically acceptable
compound
composition
acceptable form
acceptable carrier
Prior art date
Application number
BG104048A
Other languages
Bulgarian (bg)
English (en)
Inventor
Jai Patel
Hamish Ross
Jeffrey Granett
Robin Price
Paul WRAY
Original Assignee
Smithkline Beecham P.L.C.
Smithkline Beecham Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9712851.6A external-priority patent/GB9712851D0/en
Application filed by Smithkline Beecham P.L.C., Smithkline Beecham Corporation filed Critical Smithkline Beecham P.L.C.
Publication of BG104048A publication Critical patent/BG104048A/bg

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
BG104048A 1997-06-05 1999-12-27 Състав съдържащ 5-/4-/2-(n-метил-n-2-пиридил) амино)- етокси/ бензин/ тиазолидин-2,4-дион BG104048A (bg)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9711683.4A GB9711683D0 (en) 1997-06-05 1997-06-05 Composition
GBGB9712851.6A GB9712851D0 (en) 1997-06-18 1997-06-18 Composition
PCT/EP1998/003478 WO1998055122A1 (en) 1997-06-05 1998-06-02 Composition comprising 5-[4-[2-(n-methyl-n-2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione

Publications (1)

Publication Number Publication Date
BG104048A true BG104048A (bg) 2000-07-31

Family

ID=26311662

Family Applications (1)

Application Number Title Priority Date Filing Date
BG104048A BG104048A (bg) 1997-06-05 1999-12-27 Състав съдържащ 5-/4-/2-(n-метил-n-2-пиридил) амино)- етокси/ бензин/ тиазолидин-2,4-дион

Country Status (29)

Country Link
EP (1) EP0998284A1 (pt)
JP (1) JP2001521553A (pt)
KR (1) KR20010013410A (pt)
CN (3) CN1526391A (pt)
AP (1) AP1214A (pt)
AR (2) AR008198A1 (pt)
AU (1) AU8215098A (pt)
BG (1) BG104048A (pt)
BR (1) BR9810405A (pt)
CA (2) CA2333352A1 (pt)
CO (1) CO4940400A1 (pt)
DZ (1) DZ2510A1 (pt)
EA (1) EA002384B1 (pt)
GB (1) GB9711683D0 (pt)
HU (1) HUP0004070A3 (pt)
ID (1) ID24264A (pt)
IL (1) IL133074A0 (pt)
MX (1) MXPA99011322A (pt)
NO (2) NO995938L (pt)
NZ (2) NZ523725A (pt)
OA (1) OA11306A (pt)
PE (1) PE78899A1 (pt)
PL (1) PL337201A1 (pt)
SK (1) SK164899A3 (pt)
TR (2) TR200002790T2 (pt)
TW (1) TW570797B (pt)
UY (1) UY25032A1 (pt)
WO (1) WO1998055122A1 (pt)
ZA (2) ZA984826B (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AP1598A (en) * 1999-04-23 2006-04-26 Smithkline Beecham Plc Polymorph of 5-[4-[2-(N-methyl-N-(2-pyridyl) amino) ethoxy]benzyl] thiazolidine-2,4-dione, maleic acid salt.
US20040248945A1 (en) 1999-04-23 2004-12-09 Smithkline Beecham P.L.C. Thiazolidinedione derivative and its use as antidiabetic
EP1173434B1 (en) 1999-04-23 2003-08-20 SmithKline Beecham plc Thiazolidinedione derivative and its use as antidiabetic
GB0021978D0 (en) 2000-09-07 2000-10-25 Smithkline Beecham Plc Novel pharmaceutical
GB0127805D0 (en) * 2001-11-20 2002-01-09 Smithkline Beecham Plc Pharmaceutical composition
GB0129871D0 (en) * 2001-12-13 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
WO2003050112A1 (en) * 2001-12-13 2003-06-19 Smithkline Beecham Plc Toluenesulfonate hydrates of a thiazolidinedione derivative
GB0129876D0 (en) * 2001-12-13 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
GB0130509D0 (en) * 2001-12-20 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
EP2270007A1 (en) * 2006-05-09 2011-01-05 Teva Pharmaceutical Industries Ltd. 2-N-{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2-4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
US7435741B2 (en) 2006-05-09 2008-10-14 Teva Pharmaceutical Industries, Ltd. 2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
WO2015008234A1 (en) * 2013-07-17 2015-01-22 Glenmark Pharmaceuticals S.A. Bicyclic heterocyclic compounds as ror gamma modulators

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0306228B1 (en) * 1987-09-04 1999-11-17 Beecham Group Plc Substituted thiazolidinedione derivatives
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds
WO1995021608A1 (en) * 1994-02-10 1995-08-17 Smithkline Beecham Plc Use of insulin sensitisers for treating renal diseases
SK16498A3 (en) * 1995-08-10 1999-03-12 Warner Lambert Co A method of reducing the amount of exogenous insulin administered to a patient having noninsulin-dependent diabetes mellitus
WO1997018811A1 (en) * 1995-11-17 1997-05-29 Warner-Lambert Company A method of treating myotonic dystrophy
IL120443A (en) * 1996-03-18 2000-07-16 Sankyo Co Use of an insulin sensitizer for the manufacture of a medicament for the treatment or prophylaxis of pancreatitis
BR9710272A (pt) * 1996-07-12 1999-08-10 Smithkline Beecham Plc Novo tratamento de resisténcia a leptina

Also Published As

Publication number Publication date
CN1526391A (zh) 2004-09-08
NO995938L (no) 2000-02-02
CA2292629A1 (en) 1998-12-10
TR199902963T2 (xx) 2000-02-21
AR008198A1 (es) 1999-12-29
OA11306A (en) 2003-10-22
UY25032A1 (es) 1998-11-26
PL337201A1 (en) 2000-08-14
BR9810405A (pt) 2000-08-29
GB9711683D0 (en) 1997-08-06
DZ2510A1 (fr) 2003-01-25
CO4940400A1 (es) 2000-07-24
ID24264A (id) 2000-07-13
CA2292629C (en) 2004-01-06
TW570797B (en) 2004-01-11
EA002384B1 (ru) 2002-04-25
WO1998055122A1 (en) 1998-12-10
ZA9811572B (en) 1999-07-22
IL133074A0 (en) 2001-03-19
HUP0004070A2 (hu) 2002-02-28
CN1112926C (zh) 2003-07-02
TR200002790T2 (tr) 2001-11-21
KR20010013410A (ko) 2001-02-26
MXPA99011322A (es) 2004-12-02
NZ523725A (en) 2004-09-24
SK164899A3 (en) 2000-11-07
PE78899A1 (es) 1999-10-22
AU8215098A (en) 1998-12-21
AR015120A1 (es) 2001-04-18
NO995938D0 (no) 1999-12-03
NZ513922A (en) 2001-09-28
NO20040738L (no) 2000-02-02
EP0998284A1 (en) 2000-05-10
CN1259050A (zh) 2000-07-05
AP1214A (en) 2003-10-08
ZA984826B (en) 1999-08-03
EA199901116A1 (ru) 2000-06-26
AP9901696A0 (en) 1999-12-31
CN1430959A (zh) 2003-07-23
CA2333352A1 (en) 1998-12-10
JP2001521553A (ja) 2001-11-06
HUP0004070A3 (en) 2002-03-28

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