BG101139A - Heteroatoms-containing cyclopentanopyridyloxazolidinons - Google Patents

Heteroatoms-containing cyclopentanopyridyloxazolidinons

Info

Publication number
BG101139A
BG101139A BG101139A BG10113997A BG101139A BG 101139 A BG101139 A BG 101139A BG 101139 A BG101139 A BG 101139A BG 10113997 A BG10113997 A BG 10113997A BG 101139 A BG101139 A BG 101139A
Authority
BG
Bulgaria
Prior art keywords
heteroatoms
cyclopentanopyridyloxazolidinons
particularas
containingcyclopentanopyridyloxazolidinons
antibacerial
Prior art date
Application number
BG101139A
Other languages
Bulgarian (bg)
English (en)
Inventor
Andreas Stolle
Dieter Haebich
Bernd Riedl
Martin Ruppelt
Stephan Bartel
Walter Guarnieri
Hanno Wild
Rainer Endermann
Hein-Peter Kroll
Original Assignee
Bayer Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft
Publication of BG101139A publication Critical patent/BG101139A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
BG101139A 1996-01-18 1997-01-16 Heteroatoms-containing cyclopentanopyridyloxazolidinons BG101139A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19601627A DE19601627A1 (de) 1996-01-18 1996-01-18 Heteroatomhaltige Cyclopentanopyridyl-Oxazolidinone

Publications (1)

Publication Number Publication Date
BG101139A true BG101139A (en) 1998-04-30

Family

ID=7783042

Family Applications (1)

Application Number Title Priority Date Filing Date
BG101139A BG101139A (en) 1996-01-18 1997-01-16 Heteroatoms-containing cyclopentanopyridyloxazolidinons

Country Status (21)

Country Link
US (1) US5869659A (no)
EP (1) EP0785201A1 (no)
JP (1) JPH09202787A (no)
KR (1) KR970059170A (no)
AU (1) AU1012397A (no)
BG (1) BG101139A (no)
BR (1) BR9700716A (no)
CA (1) CA2195177A1 (no)
CZ (1) CZ15897A3 (no)
DE (1) DE19601627A1 (no)
EE (1) EE9700020A (no)
HU (1) HU9700152D0 (no)
IL (1) IL120016A0 (no)
MA (1) MA24062A1 (no)
NO (1) NO970210L (no)
PL (1) PL317985A1 (no)
SG (1) SG50001A1 (no)
SK (1) SK6997A3 (no)
TN (1) TNSN97010A1 (no)
TR (1) TR199700039A2 (no)
ZA (1) ZA97393B (no)

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US8110578B2 (en) 2008-10-27 2012-02-07 Signal Pharmaceuticals, Llc Pyrazino[2,3-b]pyrazine mTOR kinase inhibitors for oncology indications and diseases associated with the mTOR/PI3K/Akt pathway
MX341704B (es) 2009-10-26 2016-08-31 Signal Pharm Llc Métodos de síntesis y purificación de compuestos de heteroarilo.
MY183661A (en) 2011-10-19 2021-03-05 Signal Pharm Llc Treatment of cancer with tor kinase inhibitors
WO2013082344A1 (en) 2011-12-02 2013-06-06 Signal Pharmaceuticals, Llc Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1h)-one, a solid form thereof and methods of their use
ES2742398T3 (es) 2012-02-24 2020-02-14 Signal Pharm Llc Métodos para tratar el cáncer de pulmón no microcítico usando una terapia de combinación de inhibidores de TOR quinasa
AU2013203714B2 (en) 2012-10-18 2015-12-03 Signal Pharmaceuticals, Llc Inhibition of phosphorylation of PRAS40, GSK3-beta or P70S6K1 as a marker for TOR kinase inhibitory activity
AU2014207641A1 (en) 2013-01-16 2015-08-06 Signal Pharmaceuticals, Llc Substituted Pyrrolopyrimidine Compounds, compositions thereof, and methods of treatment therewith
AU2014254050B2 (en) 2013-04-17 2018-10-04 Signal Pharmaceuticals, Llc Pharmaceutical formulations, processes, solid forms and methods of use relating to 1-ethyl-7-(2-methyl-6-(1h-1,2,4-triazol-3-yl) pyridin-3-yl) -3,4-dihydropyrazino[2,3-b]pyrazin-2(1h)-one
MX2015014590A (es) 2013-04-17 2016-03-03 Signal Pharm Llc Tratamiento de cancer con dihidropirazino-pirazinas.
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BR112015026238A8 (pt) 2013-04-17 2019-12-24 Signal Pharm Llc composto dihidropirazino-pirazina, composição farmacêutica que o compreende, uso do composto, métodos para inibir ou medir a fosforilação e para inibir a atividade da proteína quinase, bem como kit
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JP2017520603A (ja) 2014-07-14 2017-07-27 シグナル ファーマシューティカルズ，エルエルシー 置換ピロロピリミジン化合物を使用するがんの治療方法及びその組成物
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Also Published As

Publication number Publication date
SK6997A3 (en) 1997-09-10
HU9700152D0 (en) 1997-03-28
EP0785201A1 (de) 1997-07-23
NO970210L (no) 1997-07-21
IL120016A0 (en) 1997-04-15
DE19601627A1 (de) 1997-07-24
EE9700020A (et) 1997-08-15
KR970059170A (ko) 1997-08-12
ZA97393B (en) 1997-07-17
TR199700039A2 (tr) 1997-08-21
US5869659A (en) 1999-02-09
JPH09202787A (ja) 1997-08-05
MX9700388A (es) 1997-07-31
MA24062A1 (fr) 1997-10-01
CZ15897A3 (en) 1997-08-13
TNSN97010A1 (fr) 2005-03-15
CA2195177A1 (en) 1997-07-19
AU1012397A (en) 1997-07-24
NO970210D0 (no) 1997-01-17
BR9700716A (pt) 1998-10-06
PL317985A1 (en) 1997-07-21
SG50001A1 (en) 1998-06-15

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