ZA97393B - Heteroatom-containing cyclopentanopyridyl-oxazolidinones - Google Patents

Heteroatom-containing cyclopentanopyridyl-oxazolidinones

Info

Publication number
ZA97393B
ZA97393B ZA97393A ZA97393A ZA97393B ZA 97393 B ZA97393 B ZA 97393B ZA 97393 A ZA97393 A ZA 97393A ZA 97393 A ZA97393 A ZA 97393A ZA 97393 B ZA97393 B ZA 97393B
Authority
ZA
South Africa
Prior art keywords
cyclopentanopyridyl
oxazolidinones
heteroatom
containing cyclopentanopyridyl
Prior art date
Application number
ZA97393A
Other languages
English (en)
Inventor
Andreas Stolle
Dieter Habich
Bernd Riedl
Martin Ruppelt
Stephan Bartel
Walter Guarnieri
Hanno Wild
Renier Endermann
Hein-Peter Kroll
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of ZA97393B publication Critical patent/ZA97393B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
ZA97393A 1996-01-18 1997-01-17 Heteroatom-containing cyclopentanopyridyl-oxazolidinones ZA97393B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19601627A DE19601627A1 (de) 1996-01-18 1996-01-18 Heteroatomhaltige Cyclopentanopyridyl-Oxazolidinone

Publications (1)

Publication Number Publication Date
ZA97393B true ZA97393B (en) 1997-07-17

Family

ID=7783042

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA97393A ZA97393B (en) 1996-01-18 1997-01-17 Heteroatom-containing cyclopentanopyridyl-oxazolidinones

Country Status (21)

Country Link
US (1) US5869659A (xx)
EP (1) EP0785201A1 (xx)
JP (1) JPH09202787A (xx)
KR (1) KR970059170A (xx)
AU (1) AU1012397A (xx)
BG (1) BG101139A (xx)
BR (1) BR9700716A (xx)
CA (1) CA2195177A1 (xx)
CZ (1) CZ15897A3 (xx)
DE (1) DE19601627A1 (xx)
EE (1) EE9700020A (xx)
HU (1) HU9700152D0 (xx)
IL (1) IL120016A0 (xx)
MA (1) MA24062A1 (xx)
NO (1) NO970210L (xx)
PL (1) PL317985A1 (xx)
SG (1) SG50001A1 (xx)
SK (1) SK6997A3 (xx)
TN (1) TNSN97010A1 (xx)
TR (1) TR199700039A2 (xx)
ZA (1) ZA97393B (xx)

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US8110578B2 (en) 2008-10-27 2012-02-07 Signal Pharmaceuticals, Llc Pyrazino[2,3-b]pyrazine mTOR kinase inhibitors for oncology indications and diseases associated with the mTOR/PI3K/Akt pathway
KR101903925B1 (ko) 2009-10-26 2018-10-02 시그날 파마소티칼 엘엘씨 헤테로아릴 화합물의 합성 및 정제 방법
MY183661A (en) 2011-10-19 2021-03-05 Signal Pharm Llc Treatment of cancer with tor kinase inhibitors
AU2012304276B2 (en) 2011-12-02 2015-01-15 Signal Pharmaceuticals, Llc Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1H)-one, a solid form thereof and methods of their use
CA2864905A1 (en) 2012-02-24 2013-08-29 Signal Pharmaceuticals, Llc Methods for treating non- small cell lung cancer using tor kinase inhibitor combination therapy
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US9358232B2 (en) 2013-04-17 2016-06-07 Signal Pharmaceuticals, Llc Methods for treating cancer using TOR kinase inhibitor combination therapy
TWI656875B (zh) 2013-04-17 2019-04-21 美商標誌製藥公司 藉二氫吡并吡治療癌症
TW201527300A (zh) 2013-04-17 2015-07-16 Signal Pharm Llc 關於１－乙基－７－（２－甲基－６－（１Ｈ－１，２，４－三唑－３－基）吡啶－３－基）－３，４－二氫吡并［２，３－ｂ］吡－２（１Ｈ）－酮之醫藥調配物、方法、固態型式及使用方法
BR112015026297B1 (pt) 2013-04-17 2022-08-23 Signal Pharmaceuticals, Llc Uso de um inibidor da quinase tor e quinazolinona 5-substituída, composição farmacêutica que os compreende, e kit
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Also Published As

Publication number Publication date
TNSN97010A1 (fr) 2005-03-15
MA24062A1 (fr) 1997-10-01
TR199700039A2 (tr) 1997-08-21
SG50001A1 (en) 1998-06-15
HU9700152D0 (en) 1997-03-28
PL317985A1 (en) 1997-07-21
EP0785201A1 (de) 1997-07-23
NO970210D0 (no) 1997-01-17
AU1012397A (en) 1997-07-24
JPH09202787A (ja) 1997-08-05
DE19601627A1 (de) 1997-07-24
IL120016A0 (en) 1997-04-15
EE9700020A (et) 1997-08-15
NO970210L (no) 1997-07-21
CA2195177A1 (en) 1997-07-19
SK6997A3 (en) 1997-09-10
CZ15897A3 (en) 1997-08-13
KR970059170A (ko) 1997-08-12
BG101139A (en) 1998-04-30
MX9700388A (es) 1997-07-31
US5869659A (en) 1999-02-09
BR9700716A (pt) 1998-10-06

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