BE891583A - Acides 5,5-azobis-salicylique et ses sels utiles notamment pour le traitement des affections inflammatoires de l'intestin. - Google Patents

Acides 5,5-azobis-salicylique et ses sels utiles notamment pour le traitement des affections inflammatoires de l'intestin.

Info

Publication number
BE891583A
BE891583A BE0/206907A BE206907A BE891583A BE 891583 A BE891583 A BE 891583A BE 0/206907 A BE0/206907 A BE 0/206907A BE 206907 A BE206907 A BE 206907A BE 891583 A BE891583 A BE 891583A
Authority
BE
Belgium
Prior art keywords
intestin
azobis
treatment
inflammatory conditions
salts useful
Prior art date
Application number
BE0/206907A
Other languages
English (en)
Inventor
H Lambert
B Pitzele
Original Assignee
Searle & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Searle & Co filed Critical Searle & Co
Publication of BE891583A publication Critical patent/BE891583A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C245/00Compounds containing chains of at least two nitrogen atoms with at least one nitrogen-to-nitrogen multiple bond
    • C07C245/02Azo compounds, i.e. compounds having the free valencies of —N=N— groups attached to different atoms, e.g. diazohydroxides
    • C07C245/06Azo compounds, i.e. compounds having the free valencies of —N=N— groups attached to different atoms, e.g. diazohydroxides with nitrogen atoms of azo groups bound to carbon atoms of six-membered aromatic rings
    • C07C245/08Azo compounds, i.e. compounds having the free valencies of —N=N— groups attached to different atoms, e.g. diazohydroxides with nitrogen atoms of azo groups bound to carbon atoms of six-membered aromatic rings with the two nitrogen atoms of azo groups bound to carbon atoms of six-membered aromatic rings, e.g. azobenzene
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • CCHEMISTRY; METALLURGY
    • C09DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09BORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
    • C09B63/00Lakes
    • C09B63/005Metal lakes of dyes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BE0/206907A 1981-03-02 1981-12-22 Acides 5,5-azobis-salicylique et ses sels utiles notamment pour le traitement des affections inflammatoires de l'intestin. BE891583A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/239,813 US4312806A (en) 1981-03-02 1981-03-02 Method and compounds for treating inflammatory bowel disease

Publications (1)

Publication Number Publication Date
BE891583A true BE891583A (fr) 1982-06-22

Family

ID=22903854

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/206907A BE891583A (fr) 1981-03-02 1981-12-22 Acides 5,5-azobis-salicylique et ses sels utiles notamment pour le traitement des affections inflammatoires de l'intestin.

Country Status (23)

Country Link
US (1) US4312806A (fr)
JP (1) JPS57144219A (fr)
AT (1) AT375637B (fr)
AU (1) AU545804B2 (fr)
BE (1) BE891583A (fr)
CA (1) CA1167031A (fr)
CH (1) CH647409A5 (fr)
DE (1) DE3149359A1 (fr)
DK (1) DK540581A (fr)
ES (1) ES8500894A1 (fr)
FI (1) FI813919L (fr)
FR (1) FR2500824B1 (fr)
GB (1) GB2093833B (fr)
GR (1) GR76684B (fr)
IE (1) IE52898B1 (fr)
IL (1) IL64459A0 (fr)
IT (1) IT1147821B (fr)
NL (1) NL8105824A (fr)
NO (1) NO153099C (fr)
NZ (1) NZ199273A (fr)
PH (1) PH17040A (fr)
SE (1) SE8107292L (fr)
ZA (1) ZA818507B (fr)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57500432A (fr) * 1980-03-20 1982-03-11
US4960765A (en) * 1980-03-20 1990-10-02 Farmaceutisk Laboratorium Ferring A/S Pharmaceutical composition and method for the treatment of colitis ulcerosa and Crohn's disease by oral administration
SE8002322L (sv) * 1980-03-26 1981-09-27 Pharmacia Ab Medel for behandling av inflammatoriska tarmsjukdomar
DE3151196A1 (de) * 1981-12-23 1983-06-30 Kurt Heinz Prof. Dr. 7800 Freiburg Bauer Verfahren zur herstellung von gut loeslichen 5-aminosalicylsaeure-arzneimittelzubereitungen
SE8303399D0 (sv) * 1983-06-15 1983-06-15 Pharmacia Ab Azo-bis-salicyl syra och salt derav, deras farmaceutiska beredning samt framstellning av syran
SE8303400D0 (sv) * 1983-06-15 1983-06-15 Pharmacia Ab Azo-bis-salicylsyra och salt derav samt deras farmaceutiska beredning och anvendning
SE8405924L (sv) * 1984-11-23 1986-05-24 Pharmacia Ab Nya azoforeningar
US5120306A (en) * 1990-03-21 1992-06-09 Gosselin Leon F Direct delivery of anti-inflammatories to the proximal small bowel
ES2104513B1 (es) * 1995-10-11 1998-07-01 Uriach & Cia Sa J Nuevos derivados del acido 5-aminosalicilico.
ES2106682B1 (es) * 1995-09-08 1998-07-01 Uriach & Cia Sa J Nuevos derivados azo del acido 5-aminosalicilico.
DE69611598T2 (de) * 1995-09-08 2001-06-07 Uriach & Cia Sa J Azoderivate von 5-aminosalicylsäure zur behandlung von enzündlichen darmerkrankungen
US6358939B1 (en) 1999-12-21 2002-03-19 Northern Lights Pharmaceuticals, Llc Use of biologically active vitamin D compounds for the prevention and treatment of inflammatory bowel disease
US6989377B2 (en) 1999-12-21 2006-01-24 Wisconsin Alumni Research Foundation Treating vitamin D responsive diseases
ES2165803B1 (es) 2000-04-10 2003-09-16 Uriach & Cia Sa J Nueva sal de un derivado azo del acido 5-aminosalicilico
CA2359812C (fr) * 2000-11-20 2004-02-10 The Procter & Gamble Company Formes posologiques pharmaceutiques a couches multiples permettant de reduire l'impact des revetement fractures
SI1706424T1 (sl) 2004-01-12 2010-01-29 Applied Molecular Evolution Variante fc regij
WO2010042933A2 (fr) 2008-10-10 2010-04-15 Northwestern University Inhibition et traitement des métastases du cancer de la prostate
WO2016073897A1 (fr) 2014-11-06 2016-05-12 Northwestern University Inhibition de la motilité de cellules cancéreuses
CN105985259B (zh) * 2015-02-04 2018-07-27 中国科学院化学研究所 偶氮苯甲酸类化合物及其制备方法和应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1157169A (en) * 1914-11-03 1915-10-19 Geigy Ag J R Mordant-dyeing azo dye.
GB408676A (en) * 1931-10-17 1934-04-16 Ig Farbenindustrie Ag The manufacture of symmetrically substituted azobenzene compounds
US2894984A (en) * 1958-05-15 1959-07-14 Pennsalt Chemicals Corp 4-trifluoromethyl salicylic acids and their preparation
US3413225A (en) * 1966-06-27 1968-11-26 Monsanto Co Functional fluid containing azo benzene derivatives as antioxidants
US3674844A (en) * 1970-04-20 1972-07-04 Merck & Co Inc Salicylic acid derivatives
US4190716A (en) * 1978-12-20 1980-02-26 Dynapol Polymeric agent for releasing 5-aminosalicylic acid or its salts into the gastrointestinal tract
SE8002322L (sv) * 1980-03-26 1981-09-27 Pharmacia Ab Medel for behandling av inflammatoriska tarmsjukdomar

Also Published As

Publication number Publication date
IT8247894A0 (it) 1982-03-02
IE813104L (en) 1982-09-02
DE3149359A1 (de) 1982-09-16
PH17040A (en) 1984-05-17
FR2500824B1 (fr) 1985-07-19
AU7828681A (en) 1982-09-09
NO153099B (no) 1985-10-07
ATA540681A (de) 1984-01-15
AU545804B2 (en) 1985-08-01
GR76684B (fr) 1984-08-24
FR2500824A1 (fr) 1982-09-03
NO814424L (no) 1982-09-03
ES507811A0 (es) 1984-11-01
GB2093833B (en) 1985-01-23
JPS57144219A (en) 1982-09-06
US4312806A (en) 1982-01-26
SE8107292L (sv) 1982-09-03
NL8105824A (nl) 1982-10-01
CA1167031A (fr) 1984-05-08
ES8500894A1 (es) 1984-11-01
NO153099C (no) 1986-01-15
CH647409A5 (de) 1985-01-31
FI813919L (fi) 1982-09-03
IL64459A0 (en) 1982-03-31
NZ199273A (en) 1985-03-20
GB2093833A (en) 1982-09-08
IT1147821B (it) 1986-11-26
AT375637B (de) 1984-08-27
DK540581A (da) 1982-09-03
IE52898B1 (en) 1988-04-13
ZA818507B (en) 1983-07-27

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: PHARMACIA A/B

Effective date: 19891231