BE881675A - B-lactames derives de l'acide penicillanique leur preparation et leurs utilisations therapeutiques - Google Patents
B-lactames derives de l'acide penicillanique leur preparation et leurs utilisations therapeutiques Download PDFInfo
- Publication number
- BE881675A BE881675A BE0/199363A BE199363A BE881675A BE 881675 A BE881675 A BE 881675A BE 0/199363 A BE0/199363 A BE 0/199363A BE 199363 A BE199363 A BE 199363A BE 881675 A BE881675 A BE 881675A
- Authority
- BE
- Belgium
- Prior art keywords
- emi
- preparation
- formula
- therapeutic uses
- aqueous phase
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D503/00—Heterocyclic compounds containing 4-oxa-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxapenicillins, clavulanic acid derivatives; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB7905020 | 1979-02-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE881675A true BE881675A (fr) | 1980-08-12 |
Family
ID=10503160
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE0/199363A BE881675A (fr) | 1979-02-13 | 1980-02-12 | B-lactames derives de l'acide penicillanique leur preparation et leurs utilisations therapeutiques |
Country Status (4)
Country | Link |
---|---|
JP (2) | JPS55113790A (ko) |
KR (1) | KR830001903B1 (ko) |
BE (1) | BE881675A (ko) |
ZA (1) | ZA80796B (ko) |
Cited By (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4309347A (en) | 1979-05-16 | 1982-01-05 | Pfizer Inc. | Penicillanoyloxymethyl penicillanate 1,1,1',1'-tetraoxide |
EP0059046A1 (en) * | 1981-02-20 | 1982-09-01 | Pfizer Inc. | Bis-esters of alkanediols, pharmaceutical compositions thereof and intermediates therefor |
US4420426A (en) | 1979-03-05 | 1983-12-13 | Pfizer Inc. | 6-Alpha-halopenicillanic acid 1,1-dioxides |
US4432970A (en) * | 1979-11-23 | 1984-02-21 | Pfizer Inc. | 6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors |
US4444686A (en) * | 1982-01-25 | 1984-04-24 | Pfizer Inc. | Crystalline penicillin ester intermediate |
US4478748A (en) * | 1981-02-20 | 1984-10-23 | Pfizer Inc. | Bis-esters of alkanediols |
US4540687A (en) * | 1981-09-09 | 1985-09-10 | Pfizer Inc. | Antibacterial 6'-(2-amino-2-[4-acyloxyphenyl]acetamido)penicillanoyloxymethyl penicillanate 1,1-dioxide compounds |
US4582829A (en) * | 1981-09-09 | 1986-04-15 | Pfizer Inc. | Antibacterial 6'-(2-amino-2-[4-acyloxyphenyl]acetamido)penicillanoyloxymethyl penicillanate 1,1-dioxide compounds |
US4714761A (en) * | 1979-03-05 | 1987-12-22 | Pfizer Inc. | 6,6-dihalopenicillanic acid 1,1-dioxides and process |
US4831025A (en) * | 1980-10-31 | 1989-05-16 | Leo Pharmaceutical Products Ltd. | Crystalline penicillin derivative tosylate hydrates |
US4882325A (en) * | 1980-10-06 | 1989-11-21 | Leo Pharmaceutical Products Ltd. A/S | Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-amino-phenylacetamido)penicillanate napsylate and method of using the same |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4244951A (en) * | 1979-05-16 | 1981-01-13 | Pfizer Inc. | Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide |
ZA821903B (en) * | 1981-03-23 | 1983-01-26 | Pfizer | Process for the preparation of penicillanic acid esters |
US4419284A (en) * | 1981-03-23 | 1983-12-06 | Pfizer Inc. | Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide |
IN159362B (ko) * | 1981-03-23 | 1987-05-09 | Pfizer | |
JPS5857384A (ja) * | 1981-09-09 | 1983-04-05 | フアイザ−・インコ−ポレ−テツド | 抗菌性のペニシラン酸6′‐(2‐アミノ‐2‐〔4‐アシルオキシフェニル〕アセタミド)ペニシラノイルオキシメチル1,1‐ジオキシド化合物 |
US4351840A (en) * | 1981-09-18 | 1982-09-28 | Pfizer Inc. | Antibacterial esters of resorcinol with ampicillin and penicillanic acid 1,1-dioxide derivatives |
US4359472A (en) * | 1981-12-22 | 1982-11-16 | Pfizer Inc. | Bis-hydroxymethyl carbonate bridged antibacterial agents |
US4432987A (en) * | 1982-04-23 | 1984-02-21 | Pfizer Inc. | Crystalline benzenesulfonate salts of sultamicillin |
PH20068A (en) * | 1982-12-06 | 1986-09-18 | Pfizer | Process and intermediates for sultamicillin and analogs |
US4835674A (en) * | 1986-07-28 | 1989-05-30 | Bull Hn Information Systems Inc. | Computer network system for multiple processing elements |
KR20020028298A (ko) * | 2000-10-09 | 2002-04-17 | 황해용 | 초배지 및 그 제조장치 |
DE102004021281A1 (de) * | 2004-04-29 | 2005-11-24 | Boehringer Ingelheim Vetmedica Gmbh | Verwendung von Meloxicam-Formulierungen in der Veterinärmedizin |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1578128A (en) * | 1976-03-30 | 1980-11-05 | Leo Pharm Prod Ltd | Amidinopenicillanoyloxyalkyl amoxycillinates |
-
1980
- 1980-02-12 BE BE0/199363A patent/BE881675A/fr not_active IP Right Cessation
- 1980-02-12 KR KR1019800000546A patent/KR830001903B1/ko active
- 1980-02-12 ZA ZA00800796A patent/ZA80796B/xx unknown
- 1980-02-13 JP JP1719780A patent/JPS55113790A/ja active Granted
-
1987
- 1987-05-11 JP JP62114399A patent/JPS62281879A/ja active Granted
Cited By (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4420426A (en) | 1979-03-05 | 1983-12-13 | Pfizer Inc. | 6-Alpha-halopenicillanic acid 1,1-dioxides |
US4714761A (en) * | 1979-03-05 | 1987-12-22 | Pfizer Inc. | 6,6-dihalopenicillanic acid 1,1-dioxides and process |
US4309347A (en) | 1979-05-16 | 1982-01-05 | Pfizer Inc. | Penicillanoyloxymethyl penicillanate 1,1,1',1'-tetraoxide |
US4432970A (en) * | 1979-11-23 | 1984-02-21 | Pfizer Inc. | 6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors |
US4882325A (en) * | 1980-10-06 | 1989-11-21 | Leo Pharmaceutical Products Ltd. A/S | Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-amino-phenylacetamido)penicillanate napsylate and method of using the same |
US4831025A (en) * | 1980-10-31 | 1989-05-16 | Leo Pharmaceutical Products Ltd. | Crystalline penicillin derivative tosylate hydrates |
EP0059046A1 (en) * | 1981-02-20 | 1982-09-01 | Pfizer Inc. | Bis-esters of alkanediols, pharmaceutical compositions thereof and intermediates therefor |
US4478748A (en) * | 1981-02-20 | 1984-10-23 | Pfizer Inc. | Bis-esters of alkanediols |
US4540687A (en) * | 1981-09-09 | 1985-09-10 | Pfizer Inc. | Antibacterial 6'-(2-amino-2-[4-acyloxyphenyl]acetamido)penicillanoyloxymethyl penicillanate 1,1-dioxide compounds |
US4582829A (en) * | 1981-09-09 | 1986-04-15 | Pfizer Inc. | Antibacterial 6'-(2-amino-2-[4-acyloxyphenyl]acetamido)penicillanoyloxymethyl penicillanate 1,1-dioxide compounds |
US4444686A (en) * | 1982-01-25 | 1984-04-24 | Pfizer Inc. | Crystalline penicillin ester intermediate |
Also Published As
Publication number | Publication date |
---|---|
JPH0470315B2 (ko) | 1992-11-10 |
ZA80796B (en) | 1981-02-25 |
KR830001903B1 (ko) | 1983-09-19 |
KR830001947A (ko) | 1983-05-21 |
JPS55113790A (en) | 1980-09-02 |
JPS62281879A (ja) | 1987-12-07 |
JPS6259709B2 (ko) | 1987-12-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
CCPA | Application for a supplementary protection certificate |
Free format text: 093C0069 |
|
CCPV | Grant of a supplementary protection certificate |
Free format text: 093C0069, EXPIRES 20020409 |
|
RE20 | Patent expired |
Owner name: LEO PHARMACEUTICAL PRODUCTS LTD A/S (LOVENS KEMIS Effective date: 20000212 |