BE1002710A5 - Preparation au diclofenac sodique a effet prolonge. - Google Patents
Preparation au diclofenac sodique a effet prolonge. Download PDFInfo
- Publication number
- BE1002710A5 BE1002710A5 BE8900683A BE8900683A BE1002710A5 BE 1002710 A5 BE1002710 A5 BE 1002710A5 BE 8900683 A BE8900683 A BE 8900683A BE 8900683 A BE8900683 A BE 8900683A BE 1002710 A5 BE1002710 A5 BE 1002710A5
- Authority
- BE
- Belgium
- Prior art keywords
- diclofenac sodium
- preparation
- long
- term effect
- component
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
- A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
- A61K9/5047—Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Abstract
Préparation au diclofénac sodique à effet prolongé, caractérisée en ce qu'elle comprend un composant de diclofénac sodique à libération retardée, ce composant comprenant une composition pharmaceutique munie d'un enrobage retard, cette composition phamaceutique comprenant du diclofénac sodique et un acide organique.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP20349888 | 1988-08-16 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE1002710A5 true BE1002710A5 (fr) | 1991-05-14 |
Family
ID=16475153
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE8900683A BE1002710A5 (fr) | 1988-08-16 | 1989-06-22 | Preparation au diclofenac sodique a effet prolonge. |
Country Status (13)
Country | Link |
---|---|
US (1) | US4968505A (fr) |
JP (1) | JPH07116028B2 (fr) |
KR (1) | KR950003610B1 (fr) |
BE (1) | BE1002710A5 (fr) |
CA (1) | CA1319616C (fr) |
CH (1) | CH678813A5 (fr) |
DE (1) | DE3915150C2 (fr) |
FR (1) | FR2635460B1 (fr) |
GB (1) | GB2221842B (fr) |
HK (1) | HK48194A (fr) |
IT (1) | IT1231517B (fr) |
NL (1) | NL194882C (fr) |
SE (1) | SE509029C2 (fr) |
Families Citing this family (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2514078B2 (ja) * | 1988-08-22 | 1996-07-10 | エスエス製薬株式会社 | 圧縮成型製剤 |
US5079001A (en) * | 1989-11-03 | 1992-01-07 | Ciba-Geigy Corporation | Liquid oral formulation of diclofenac |
US5015481A (en) * | 1990-05-03 | 1991-05-14 | G. D. Searle & Co. | Stabilized pharmaceutical admixture composition |
JPH04230625A (ja) * | 1990-12-27 | 1992-08-19 | Standard Chem & Pharmaceut Corp Ltd | 噴霧乾燥したジクロフェナクナトリウムを含み腸溶性の被覆を有するマイクロカプセルからなる微分散した錠剤組成物の製造方法 |
EP0520119A1 (fr) * | 1991-06-17 | 1992-12-30 | Spirig Ag Pharmazeutische Präparate | Composition à base de diclofenac pour l'administration orale |
US5518737A (en) * | 1991-10-16 | 1996-05-21 | Orion-Yhtyma Oy | Peroral drug delivery system |
WO1994003160A1 (fr) * | 1992-08-05 | 1994-02-17 | F.H. Faulding & Co. Limited | Composition pharmaceutique sous forme de granules |
JP3349535B2 (ja) * | 1993-01-12 | 2002-11-25 | フロイント産業株式会社 | 球形顆粒の製造方法 |
DE4403943A1 (de) * | 1994-02-08 | 1995-08-10 | Hexal Pharma Gmbh | Orale Azrneimittelzubereitung mit Diclofenac-Natrium |
US5837284A (en) | 1995-12-04 | 1998-11-17 | Mehta; Atul M. | Delivery of multiple doses of medications |
US5922736A (en) * | 1995-12-04 | 1999-07-13 | Celegene Corporation | Chronic, bolus administration of D-threo methylphenidate |
US6486177B2 (en) * | 1995-12-04 | 2002-11-26 | Celgene Corporation | Methods for treatment of cognitive and menopausal disorders with D-threo methylphenidate |
ES2262174T3 (es) * | 1996-09-30 | 2006-11-16 | Alza Corporation | Forma de dosificacion y procedimiento de administracion de medicamentos. |
EP1690531A3 (fr) * | 1996-09-30 | 2010-01-20 | Alza Corporation | Forme de dosage et méthode d'administration de médicament |
US6919373B1 (en) | 1996-11-12 | 2005-07-19 | Alza Corporation | Methods and devices for providing prolonged drug therapy |
ES2129010B1 (es) * | 1997-01-02 | 2000-01-16 | Gold Oscar | Composicion de accion prolongada en granulos que contienen 4-nitro-2- fenoximetansulfonanilida y su procedimiento de preparacion. |
ES2129356B1 (es) * | 1997-03-26 | 2000-01-16 | Pierre Fabre Iberica S A | Forma farmaceutica de liberacion prolongada y procedimiento para su o btencion. |
US6312724B1 (en) | 1997-04-04 | 2001-11-06 | Isa Odidi | Sustained release pharmaceutical matrix tablet of pharmaceutically acceptable salts of diclofenac and process for preparation thereof |
US6962997B1 (en) * | 1997-05-22 | 2005-11-08 | Celgene Corporation | Process and intermediates for resolving piperidyl acetamide steroisomers |
US6699508B1 (en) | 1998-08-10 | 2004-03-02 | Asahi Kasei Pharma Corporation | Sustained release oral preparations of fasudil hydrochloride |
US6989159B2 (en) * | 2000-08-10 | 2006-01-24 | Jds Pharmaceuticals, Llc | Pharmaceutical compositions containing lithium carbonate |
FR2842735B1 (fr) * | 2002-07-26 | 2006-01-06 | Flamel Tech Sa | Microcapsules a liberation modifiee de principes actifs peu solubles pour l'administration per os |
US20050239830A1 (en) * | 2004-04-26 | 2005-10-27 | Vikram Khetani | Methods of diminishing co-abuse potential |
BRPI0517166A (pt) * | 2004-12-09 | 2008-09-30 | Celgene Corp | uso de d-treo-metilfenidato ou um sal do mesmo |
WO2012169614A1 (fr) * | 2011-06-10 | 2012-12-13 | ニプロ株式会社 | Procédé de production de comprimés orodispersibles |
US8962020B2 (en) * | 2012-07-26 | 2015-02-24 | Glycadia Inc. | Long-acting and controlled release formulations of 2-[(3-chlorophenyl) amino] phenylacetic acid |
WO2017084680A1 (fr) * | 2015-11-17 | 2017-05-26 | Rontis Hellas S.A. | Composition pharmaceutique contenant un médicament anti-inflammatoire non stéroïdien et un inhibiteur de pompe à protons |
CN114306260B (zh) * | 2021-12-29 | 2023-10-24 | 濮阳市汇元药业有限公司 | 一种新型双氯芬酸钠片及其制备方法 |
DE202022100544U1 (de) | 2022-01-31 | 2022-02-16 | Ranjitsing Babasing Bayas | Neue orale Streifen- oder Dünnfilmform von Diclofenac-Natrium |
Citations (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB2039737A (en) * | 1978-12-22 | 1980-08-20 | Panoz D | Galenical forms for administration of medicaments by oral by oral route with programmed release and processes for preparing same |
WO1981001652A1 (fr) * | 1979-12-07 | 1981-06-25 | D Panoz | Perfectionnements apportes aux procedes de preparation de formes galeniques a action retard et a liberation programmee et formes galeniques de medicaments ainsi obtenues |
EP0156077A1 (fr) * | 1983-12-21 | 1985-10-02 | ELAN CORPORATION, Plc | Formulation pharmaceutique à absorption contrôlée |
EP0209975A1 (fr) * | 1985-06-04 | 1987-01-28 | Nitto Denko Corporation | Préparation adhésive analgésique anti-inflammatoire |
EP0218148A1 (fr) * | 1985-09-26 | 1987-04-15 | Chugai Seiyaku Kabushiki Kaisha | Composition pharmaceutique à libération lente |
EP0232155A2 (fr) * | 1986-02-03 | 1987-08-12 | Elan Corporation Plc | Système pour la libération de médicaments |
GB2217598A (en) * | 1988-03-25 | 1989-11-01 | Ciba Geigy | Effervescent tablet containing diclofenac |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH655507B (fr) * | 1983-01-12 | 1986-04-30 | ||
DE3328401A1 (de) * | 1983-08-05 | 1985-02-21 | Merckle GmbH, 7902 Blaubeuren | Injizierbare loesung zur behandlung von entzuendungen |
DE3446873A1 (de) * | 1984-12-21 | 1986-07-10 | Merckle Gmbh | Fluessige diclofenac-zubereitungen |
CH664085A5 (de) * | 1985-02-08 | 1988-02-15 | Ciba Geigy Ag | Pharmazeutische praeparate mit analgetischer wirksamkeit, sowie deren herstellung. |
US4814183A (en) * | 1987-08-31 | 1989-03-21 | Merck & Co., Inc. | Device for the controlled release of drugs with Donnan-like modulation by charged insoluble resins |
-
1989
- 1989-05-03 SE SE8901593A patent/SE509029C2/sv not_active IP Right Cessation
- 1989-05-04 GB GB8910271A patent/GB2221842B/en not_active Expired - Lifetime
- 1989-05-04 CA CA000598715A patent/CA1319616C/fr not_active Expired - Fee Related
- 1989-05-08 JP JP1114461A patent/JPH07116028B2/ja not_active Expired - Fee Related
- 1989-05-09 DE DE3915150A patent/DE3915150C2/de not_active Expired - Fee Related
- 1989-05-10 KR KR1019890006268A patent/KR950003610B1/ko not_active IP Right Cessation
- 1989-05-12 NL NL8901200A patent/NL194882C/nl not_active IP Right Cessation
- 1989-05-17 US US07/353,016 patent/US4968505A/en not_active Expired - Lifetime
- 1989-05-31 FR FR898907203A patent/FR2635460B1/fr not_active Expired - Fee Related
- 1989-06-01 IT IT8948030A patent/IT1231517B/it active
- 1989-06-22 BE BE8900683A patent/BE1002710A5/fr not_active IP Right Cessation
- 1989-06-27 CH CH2389/89A patent/CH678813A5/de not_active IP Right Cessation
-
1994
- 1994-05-19 HK HK48194A patent/HK48194A/xx not_active IP Right Cessation
Patent Citations (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB2039737A (en) * | 1978-12-22 | 1980-08-20 | Panoz D | Galenical forms for administration of medicaments by oral by oral route with programmed release and processes for preparing same |
WO1981001652A1 (fr) * | 1979-12-07 | 1981-06-25 | D Panoz | Perfectionnements apportes aux procedes de preparation de formes galeniques a action retard et a liberation programmee et formes galeniques de medicaments ainsi obtenues |
EP0156077A1 (fr) * | 1983-12-21 | 1985-10-02 | ELAN CORPORATION, Plc | Formulation pharmaceutique à absorption contrôlée |
EP0209975A1 (fr) * | 1985-06-04 | 1987-01-28 | Nitto Denko Corporation | Préparation adhésive analgésique anti-inflammatoire |
EP0218148A1 (fr) * | 1985-09-26 | 1987-04-15 | Chugai Seiyaku Kabushiki Kaisha | Composition pharmaceutique à libération lente |
EP0232155A2 (fr) * | 1986-02-03 | 1987-08-12 | Elan Corporation Plc | Système pour la libération de médicaments |
GB2217598A (en) * | 1988-03-25 | 1989-11-01 | Ciba Geigy | Effervescent tablet containing diclofenac |
Also Published As
Publication number | Publication date |
---|---|
JPH07116028B2 (ja) | 1995-12-13 |
NL194882B (nl) | 2003-02-03 |
SE8901593D0 (sv) | 1989-05-03 |
SE8901593L (sv) | 1990-12-06 |
NL8901200A (nl) | 1990-03-16 |
CA1319616C (fr) | 1993-06-29 |
HK48194A (en) | 1994-05-27 |
JPH02237918A (ja) | 1990-09-20 |
GB8910271D0 (en) | 1989-06-21 |
DE3915150A1 (de) | 1990-03-01 |
DE3915150C2 (de) | 1997-04-17 |
GB2221842B (en) | 1991-10-16 |
IT1231517B (it) | 1991-12-07 |
FR2635460A1 (fr) | 1990-02-23 |
NL194882C (nl) | 2003-06-04 |
GB2221842A (en) | 1990-02-21 |
KR900002769A (ko) | 1990-03-23 |
CH678813A5 (fr) | 1991-11-15 |
IT8948030A0 (it) | 1989-06-01 |
US4968505A (en) | 1990-11-06 |
FR2635460B1 (fr) | 1994-09-16 |
SE509029C2 (sv) | 1998-11-30 |
KR950003610B1 (ko) | 1995-04-17 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Effective date: 20030630 |