BE1000072A4 - Derives de l'indole utiles comme medicaments et procede et intermediaires pour leur preparation. - Google Patents

Derives de l'indole utiles comme medicaments et procede et intermediaires pour leur preparation. Download PDF

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Publication number
BE1000072A4
BE1000072A4 BE8700004A BE8700004A BE1000072A4 BE 1000072 A4 BE1000072 A4 BE 1000072A4 BE 8700004 A BE8700004 A BE 8700004A BE 8700004 A BE8700004 A BE 8700004A BE 1000072 A4 BE1000072 A4 BE 1000072A4
Authority
BE
Belgium
Prior art keywords
group
general formula
compound
hydrogen atom
desc
Prior art date
Application number
BE8700004A
Other languages
English (en)
French (fr)
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of BE1000072A4 publication Critical patent/BE1000072A4/fr

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16Tryptamines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
BE8700004A 1986-01-08 1987-01-08 Derives de l'indole utiles comme medicaments et procede et intermediaires pour leur preparation. BE1000072A4 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB868600398A GB8600398D0 (en) 1986-01-08 1986-01-08 Chemical compounds

Publications (1)

Publication Number Publication Date
BE1000072A4 true BE1000072A4 (fr) 1988-02-02

Family

ID=10591075

Family Applications (1)

Application Number Title Priority Date Filing Date
BE8700004A BE1000072A4 (fr) 1986-01-08 1987-01-08 Derives de l'indole utiles comme medicaments et procede et intermediaires pour leur preparation.

Country Status (11)

Country Link
JP (1) JPS62228057A (de)
AT (1) AT386197B (de)
AU (1) AU597324B2 (de)
BE (1) BE1000072A4 (de)
CH (1) CH671017A5 (de)
DE (1) DE3700407A1 (de)
FR (1) FR2595352B1 (de)
GB (2) GB8600398D0 (de)
IT (1) IT1216772B (de)
NL (1) NL8700027A (de)
ZA (1) ZA87104B (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8600397D0 (en) * 1986-01-08 1986-02-12 Glaxo Group Ltd Chemical compounds
US5225431A (en) * 1987-10-23 1993-07-06 Burroughs Wellcome Co. Therapeutic substituted indole compounds and compositions thereof
GB8819024D0 (en) * 1988-08-10 1988-09-14 Glaxo Group Ltd Chemical compounds
IL114690A (en) * 1990-06-07 1997-02-18 Wellcome Found Antimigraine oxazolidinone substituted indole derivatives
GB9012672D0 (en) * 1990-06-07 1990-08-01 Wellcome Found Therapeutic heterocyclic compounds
TW263508B (de) * 1991-02-12 1995-11-21 Pfizer
US5206377A (en) * 1991-12-05 1993-04-27 Whitby Research, Inc. Compounds useful as antiproliferative agents
GB9201038D0 (en) * 1992-01-16 1992-03-11 Glaxo Group Ltd Chemical compounds
US5409941A (en) * 1992-02-03 1995-04-25 Pfizer Inc. 5-heteroyl indole derivatives
GB9211277D0 (en) 1992-05-28 1992-07-15 Glaxo Group Inc Pharmaceutical compositions
US5496957A (en) * 1993-09-01 1996-03-05 Virginia Commonwealth University Tryptamine analogs with 5-HT1D selectivity
EP0666847B1 (de) * 1993-09-01 1998-06-17 Allelix Biopharmaceuticals Inc. Tryptamin analoge mit 5-ht1d selektivität
JP4897221B2 (ja) * 2002-12-20 2012-03-14 チバ ホールディング インコーポレーテッド アミン類の合成及びその合成のための中間体

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2035310A (en) * 1978-10-12 1980-06-18 Glaxo Group Ltd Indole-s-carbaxamides and this anologues
GB2081717A (en) * 1980-08-12 1982-02-24 Glaxo Group Ltd Hereocyclic compounds
GB2083463A (en) * 1980-08-12 1982-03-24 Glaxo Group Ltd Heterocyclic compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB147107A (en) * 1915-04-06 1921-10-07 Zeiss Carl Improvements in finders for photographic apparatus
GB145459A (en) * 1917-03-24 1921-04-21 Anschuetz & Co Gmbh Improvements in indicators for the turning of aircraft about a vertical axis
GB8600397D0 (en) * 1986-01-08 1986-02-12 Glaxo Group Ltd Chemical compounds
FR2903394B1 (fr) * 2006-07-05 2008-09-19 Pierre Marcelli Devidoir a mandrin expansible pour bobine
US20100180029A1 (en) * 2007-04-06 2010-07-15 Clive Fourman Content delivery system and method of delivering content

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2035310A (en) * 1978-10-12 1980-06-18 Glaxo Group Ltd Indole-s-carbaxamides and this anologues
GB2081717A (en) * 1980-08-12 1982-02-24 Glaxo Group Ltd Hereocyclic compounds
GB2083463A (en) * 1980-08-12 1982-03-24 Glaxo Group Ltd Heterocyclic compounds

Also Published As

Publication number Publication date
GB8600398D0 (en) 1986-02-12
ATA2487A (de) 1987-12-15
GB2186874A (en) 1987-08-26
AT386197B (de) 1988-07-11
DE3700407A1 (de) 1987-07-09
JPS62228057A (ja) 1987-10-06
NL8700027A (nl) 1987-08-03
FR2595352B1 (fr) 1990-07-13
AU597324B2 (en) 1990-05-31
IT1216772B (it) 1990-03-14
GB8700381D0 (en) 1987-02-11
CH671017A5 (de) 1989-07-31
GB2186874B (en) 1990-02-07
IT8747506A0 (it) 1987-01-08
FR2595352A1 (fr) 1987-09-11
AU6741887A (en) 1987-07-09
ZA87104B (en) 1987-12-30

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: GLAXO GROUP LTD

Effective date: 19920131