AU720135B2 - Pyrimidine derivatives and processes for the preparation thereof - Google Patents

Pyrimidine derivatives and processes for the preparation thereof Download PDF

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Publication number
AU720135B2
AU720135B2 AU48642/97A AU4864297A AU720135B2 AU 720135 B2 AU720135 B2 AU 720135B2 AU 48642/97 A AU48642/97 A AU 48642/97A AU 4864297 A AU4864297 A AU 4864297A AU 720135 B2 AU720135 B2 AU 720135B2
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AU
Australia
Prior art keywords
amino
phenylamino
phenyl
alkyl
mmol
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU48642/97A
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English (en)
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AU4864297A (en
Inventor
Guido Bold
Jorg Frei
Marc Lang
Peter Traxler
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Novartis AG
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Novartis AG
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Publication of AU4864297A publication Critical patent/AU4864297A/en
Application granted granted Critical
Publication of AU720135B2 publication Critical patent/AU720135B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Compounds Of Unknown Constitution (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
AU48642/97A 1996-10-02 1997-09-30 Pyrimidine derivatives and processes for the preparation thereof Ceased AU720135B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH2399/96 1996-10-02
CH239996 1996-10-02
PCT/EP1997/005369 WO1998014450A1 (en) 1996-10-02 1997-09-30 Pyrimidine derivatives and processes for the preparation thereof

Publications (2)

Publication Number Publication Date
AU4864297A AU4864297A (en) 1998-04-24
AU720135B2 true AU720135B2 (en) 2000-05-25

Family

ID=4232877

Family Applications (1)

Application Number Title Priority Date Filing Date
AU48642/97A Ceased AU720135B2 (en) 1996-10-02 1997-09-30 Pyrimidine derivatives and processes for the preparation thereof

Country Status (9)

Country Link
US (1) US6251911B1 (https=)
EP (1) EP0929553B1 (https=)
JP (1) JP4205168B2 (https=)
AT (1) ATE291022T1 (https=)
AU (1) AU720135B2 (https=)
CA (1) CA2266519C (https=)
DE (1) DE69732780T2 (https=)
ES (1) ES2239779T3 (https=)
WO (1) WO1998014450A1 (https=)

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AU4864297A (en) 1998-04-24
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ATE291022T1 (de) 2005-04-15
EP0929553B1 (en) 2005-03-16
CA2266519C (en) 2007-01-23
DE69732780D1 (de) 2005-04-21
CA2266519A1 (en) 1998-04-09
JP2001501216A (ja) 2001-01-30
DE69732780T2 (de) 2006-04-06
EP0929553A1 (en) 1999-07-21
US6251911B1 (en) 2001-06-26
ES2239779T3 (es) 2005-10-01

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