AU596258B2 - Novel aminoalkanoyl-dibenzo(d,g)(1,3,6)dioxazocines and a process for the preparation thereof - Google Patents

Novel aminoalkanoyl-dibenzo(d,g)(1,3,6)dioxazocines and a process for the preparation thereof Download PDF

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Publication number
AU596258B2
AU596258B2 AU83140/87A AU8314087A AU596258B2 AU 596258 B2 AU596258 B2 AU 596258B2 AU 83140/87 A AU83140/87 A AU 83140/87A AU 8314087 A AU8314087 A AU 8314087A AU 596258 B2 AU596258 B2 AU 596258B2
Authority
AU
Australia
Prior art keywords
formula
dibenzo
compound
carbon atoms
moles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU83140/87A
Other languages
English (en)
Other versions
AU8314087A (en
Inventor
Marton Fekete
Istvan Gacsalyi
Maria Hegedus
Lujza Petocz
Lazslo Rozsa
Eniko Sziri
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Egis Pharmaceuticals PLC
Original Assignee
Egyt Gyogyszervegyeszeti Gyar
Egis Pharmaceuticals PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egyt Gyogyszervegyeszeti Gyar, Egis Pharmaceuticals PLC filed Critical Egyt Gyogyszervegyeszeti Gyar
Publication of AU8314087A publication Critical patent/AU8314087A/en
Application granted granted Critical
Publication of AU596258B2 publication Critical patent/AU596258B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • C07D273/01—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00 having one nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
    • A61P23/02—Local anaesthetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AU83140/87A 1986-12-30 1987-12-30 Novel aminoalkanoyl-dibenzo(d,g)(1,3,6)dioxazocines and a process for the preparation thereof Ceased AU596258B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU5513/86 1986-12-30
HU865513A HU198194B (en) 1986-12-30 1986-12-30 Process for production of new derivatives of dioxazocin and medical compositions containing them

Publications (2)

Publication Number Publication Date
AU8314087A AU8314087A (en) 1988-06-30
AU596258B2 true AU596258B2 (en) 1990-04-26

Family

ID=10970381

Family Applications (1)

Application Number Title Priority Date Filing Date
AU83140/87A Ceased AU596258B2 (en) 1986-12-30 1987-12-30 Novel aminoalkanoyl-dibenzo(d,g)(1,3,6)dioxazocines and a process for the preparation thereof

Country Status (26)

Country Link
JP (1) JPS63174978A (el)
KR (1) KR880007502A (el)
CN (1) CN87108190A (el)
AT (1) AT389304B (el)
AU (1) AU596258B2 (el)
BE (1) BE1001240A3 (el)
CH (1) CH675877A5 (el)
CS (1) CS270579B2 (el)
DD (1) DD267038A5 (el)
DE (1) DE3744549A1 (el)
DK (1) DK691087A (el)
ES (1) ES2006539A6 (el)
FI (1) FI875767A (el)
FR (1) FR2609030B1 (el)
GB (1) GB2199827B (el)
GR (1) GR872083B (el)
HU (1) HU198194B (el)
IL (1) IL84976A (el)
IT (1) IT1233443B (el)
NL (1) NL8703150A (el)
NO (1) NO169230B (el)
PL (1) PL151402B1 (el)
SE (1) SE465429B (el)
SU (1) SU1575938A3 (el)
YU (1) YU235287A (el)
ZA (1) ZA879733B (el)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU610678B2 (en) * 1987-12-31 1991-05-23 Egis Gyogyszergyar Dioxazocine derivatives, their preparation and compositions containing them

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2058761T3 (es) * 1989-10-20 1994-11-01 Akzo Nv Proceso para la preparacion de derivados de dibenzodioxazecina y dibenzodioxaazacicloundecina.

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6676586A (en) * 1985-12-20 1987-06-25 Egis Gyogyszergyar Rt. Optically active 2-chloro-12-(3-dimethylamino-2- methylpropyl)-12H-dibenzo(d,g)(1,3,6)dioxazocines and a process for the preparation thereof
AU2763788A (en) * 1987-12-31 1989-07-06 Egis Gyogyszergyar Dioxazocine derivatives, their preparation and compositions containing them

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2659M (fr) * 1963-04-25 1964-08-14 Millot Lab Médicament a base de dérivé de la phénothiazine.
HU174126B (hu) * 1977-08-02 1979-11-28 Egyt Gyogyszervegyeszeti Gyar Sposob poluchenija novykh proizvodnykh dibenzo-kvadratnaja skobka-d,g-kvadratnaja skobka zakryta-kvadratnaja skobka-1,3,6-kvadratnaja skobka zakryta-dioksazocina

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6676586A (en) * 1985-12-20 1987-06-25 Egis Gyogyszergyar Rt. Optically active 2-chloro-12-(3-dimethylamino-2- methylpropyl)-12H-dibenzo(d,g)(1,3,6)dioxazocines and a process for the preparation thereof
AU2763788A (en) * 1987-12-31 1989-07-06 Egis Gyogyszergyar Dioxazocine derivatives, their preparation and compositions containing them

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU610678B2 (en) * 1987-12-31 1991-05-23 Egis Gyogyszergyar Dioxazocine derivatives, their preparation and compositions containing them

Also Published As

Publication number Publication date
FR2609030B1 (fr) 1991-05-31
DK691087A (da) 1988-07-01
SE465429B (sv) 1991-09-09
GB8730298D0 (en) 1988-02-03
SE8705187L (sv) 1988-07-01
SU1575938A3 (ru) 1990-06-30
CN87108190A (zh) 1988-07-13
DD267038A5 (de) 1989-04-19
GB2199827A (en) 1988-07-20
AT389304B (de) 1989-11-27
AU8314087A (en) 1988-06-30
NO875465L (no) 1988-07-01
IT1233443B (it) 1992-04-01
NO875465D0 (no) 1987-12-29
PL151402B1 (en) 1990-08-31
CH675877A5 (el) 1990-11-15
HUT47260A (en) 1989-02-28
GR872083B (en) 1988-04-27
ZA879733B (en) 1988-06-24
JPS63174978A (ja) 1988-07-19
ES2006539A6 (es) 1989-05-01
FI875767A (fi) 1988-07-01
ATA345087A (de) 1989-04-15
NL8703150A (nl) 1988-07-18
PL269812A1 (en) 1988-09-15
SE8705187D0 (sv) 1987-12-29
DK691087D0 (da) 1987-12-29
CS270579B2 (en) 1990-07-12
FR2609030A1 (fr) 1988-07-01
HU198194B (en) 1989-08-28
IT8723271A0 (it) 1987-12-30
KR880007502A (ko) 1988-08-27
YU235287A (en) 1988-10-31
BE1001240A3 (fr) 1989-08-29
GB2199827B (en) 1990-10-03
IL84976A (en) 1991-09-16
DE3744549A1 (de) 1988-07-14
FI875767A0 (fi) 1987-12-30
IL84976A0 (en) 1988-06-30
NO169230B (no) 1992-02-17
CS1009187A2 (en) 1989-11-14

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