AU3223200A - Method of synthesizing barbituric acid derivatives and their use for the synthesis of chemical libraries - Google Patents

Method of synthesizing barbituric acid derivatives and their use for the synthesis of chemical libraries Download PDF

Info

Publication number
AU3223200A
AU3223200A AU32232/00A AU3223200A AU3223200A AU 3223200 A AU3223200 A AU 3223200A AU 32232/00 A AU32232/00 A AU 32232/00A AU 3223200 A AU3223200 A AU 3223200A AU 3223200 A AU3223200 A AU 3223200A
Authority
AU
Australia
Prior art keywords
aryl
alkyl
substituted
formula
template
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU32232/00A
Other languages
English (en)
Inventor
Adnan M. M. Mjalli
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
vTv Therapeutics LLC
Original Assignee
Trans Tech Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Trans Tech Pharma Inc filed Critical Trans Tech Pharma Inc
Publication of AU3223200A publication Critical patent/AU3223200A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/60—Three or more oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B40/00—Libraries per se, e.g. arrays, mixtures

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
AU32232/00A 1999-02-04 2000-02-04 Method of synthesizing barbituric acid derivatives and their use for the synthesis of chemical libraries Abandoned AU3223200A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11854799P 1999-02-04 1999-02-04
US60118547 1999-02-04
PCT/US2000/002998 WO2000046211A1 (en) 1999-02-04 2000-02-04 Method of synthesizing barbituric acid derivatives and their use for the synthesis of chemical libraries

Publications (1)

Publication Number Publication Date
AU3223200A true AU3223200A (en) 2000-08-25

Family

ID=22379282

Family Applications (1)

Application Number Title Priority Date Filing Date
AU32232/00A Abandoned AU3223200A (en) 1999-02-04 2000-02-04 Method of synthesizing barbituric acid derivatives and their use for the synthesis of chemical libraries

Country Status (6)

Country Link
EP (1) EP1155002A4 (ja)
JP (1) JP2002536368A (ja)
AU (1) AU3223200A (ja)
CA (1) CA2362085A1 (ja)
MX (1) MXPA01007869A (ja)
WO (1) WO2000046211A1 (ja)

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3247127A (en) * 1960-04-14 1966-04-19 Eastman Kodak Co Light-absorbing water-permeable colloid layer containing an oxonol dye
US4833148A (en) * 1987-04-09 1989-05-23 Washington University Method of using alkenyl- or alkynyl-substituted thiobarbiturates to reduce neurotoxic injury
US4971889A (en) * 1988-09-01 1990-11-20 Fuji Photo Film Co., Ltd. Silver halide photographic emulsions
WO1991010165A1 (en) * 1989-12-22 1991-07-11 Eastman Kodak Company Improved performance of photographic emulsions at high silver ion activities
JPH05249593A (ja) * 1992-03-04 1993-09-28 Konica Corp ハロゲン化銀写真感光材料
JPH07276810A (ja) * 1994-04-04 1995-10-24 Fuji Photo Film Co Ltd ジアゾ感熱記録材料

Also Published As

Publication number Publication date
JP2002536368A (ja) 2002-10-29
WO2000046211A1 (en) 2000-08-10
CA2362085A1 (en) 2000-08-10
EP1155002A1 (en) 2001-11-21
EP1155002A4 (en) 2003-03-19
MXPA01007869A (es) 2003-06-04

Similar Documents

Publication Publication Date Title
US6117940A (en) Amino-ketone solid support templates
US6306959B1 (en) Rapid purification by polymer supported quench
EP0840736B1 (en) Improved synthons for the synthesis and deprotection of peptide nucleic acids under mild conditions
CA2290614C (en) Process for the preparation of polymers having nucleobases as side groups
AU689764B2 (en) Modular design and synthesis of aminimide containing molecules
EP0950045B1 (en) A solid-phase technology for the preparation of amides
US5670480A (en) Method of making polymers having specific properties
AU3223200A (en) Method of synthesizing barbituric acid derivatives and their use for the synthesis of chemical libraries
ES2213825T3 (es) Engarce sililo para sintesis organica en fase solida de moleculas que contienen arilo.
KR20160062035A (ko) 히드라지드 및 피라노피라졸의 고체상 합성용 광분해성 링커
US5962412A (en) Method of making polymers having specific properties
JPH09511225A (ja) オキサゾロン誘導分子のモジュール設計および合成
CA2279208A1 (en) Novel solid-phase synthesis techniques for preparing multiple analogous compounds
US6713580B2 (en) Quaternary amino acids on solid supports
US20020146684A1 (en) One dimensional unichemo protection (UCP) in organic synthesis
WO1997040025A1 (en) Solid phase and combinatorial synthesis of substituted 1,2,3-triazoles and of arrays of substituted 1,2,3-triazoles
US7038054B1 (en) Diazabicyclononane scaffold for combinatorial synthesis
US20020019013A1 (en) Combined resin method for high-speed synthesis of combinatorial libraries
AU705844B2 (en) Combinatorial 1,4-benzodiazepin-2, 5-dione library
JP2002265481A (ja) 高分子担持光学活性ホスフィン化合物
Rühl et al. Hexafluoroacetone as protecting and activating reagent: Site-selective functionalization of iminodiacetic acid
WO2002034728A1 (en) 4-n-acyl-δ5-2-oxopiperazines, a process for its preparation and combinatorial libraries thereof
WO2003013740A1 (en) 4- AND 5-AMINO-α, β UNSTATURATED ESTER SOLID SUPPORT TEMPLATES, METHOD OF PREPARATION AND FOR USING THE SAME
WO2000053545A1 (en) Process for the synthesis of dihydropyridones
CA2180527A1 (en) Method of making polymers having specific properties

Legal Events

Date Code Title Description
MK1 Application lapsed section 142(2)(a) - no request for examination in relevant period