CA2362085A1 - Method of synthesizing barbituric acid derivatives and their use for the synthesis of chemical libraries - Google Patents

Method of synthesizing barbituric acid derivatives and their use for the synthesis of chemical libraries Download PDF

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Publication number
CA2362085A1
CA2362085A1 CA002362085A CA2362085A CA2362085A1 CA 2362085 A1 CA2362085 A1 CA 2362085A1 CA 002362085 A CA002362085 A CA 002362085A CA 2362085 A CA2362085 A CA 2362085A CA 2362085 A1 CA2362085 A1 CA 2362085A1
Authority
CA
Canada
Prior art keywords
aryl
alkyl
substituted
formula
coo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002362085A
Other languages
English (en)
French (fr)
Inventor
Adnan M. M. Mjalli
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
vTv Therapeutics LLC
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2362085A1 publication Critical patent/CA2362085A1/en
Abandoned legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/60—Three or more oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B40/00—Libraries per se, e.g. arrays, mixtures

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CA002362085A 1999-02-04 2000-02-04 Method of synthesizing barbituric acid derivatives and their use for the synthesis of chemical libraries Abandoned CA2362085A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11854799P 1999-02-04 1999-02-04
US60/118,547 1999-02-04
PCT/US2000/002998 WO2000046211A1 (en) 1999-02-04 2000-02-04 Method of synthesizing barbituric acid derivatives and their use for the synthesis of chemical libraries

Publications (1)

Publication Number Publication Date
CA2362085A1 true CA2362085A1 (en) 2000-08-10

Family

ID=22379282

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002362085A Abandoned CA2362085A1 (en) 1999-02-04 2000-02-04 Method of synthesizing barbituric acid derivatives and their use for the synthesis of chemical libraries

Country Status (6)

Country Link
EP (1) EP1155002A4 (ja)
JP (1) JP2002536368A (ja)
AU (1) AU3223200A (ja)
CA (1) CA2362085A1 (ja)
MX (1) MXPA01007869A (ja)
WO (1) WO2000046211A1 (ja)

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3247127A (en) * 1960-04-14 1966-04-19 Eastman Kodak Co Light-absorbing water-permeable colloid layer containing an oxonol dye
US4833148A (en) * 1987-04-09 1989-05-23 Washington University Method of using alkenyl- or alkynyl-substituted thiobarbiturates to reduce neurotoxic injury
US4971889A (en) * 1988-09-01 1990-11-20 Fuji Photo Film Co., Ltd. Silver halide photographic emulsions
WO1991010165A1 (en) * 1989-12-22 1991-07-11 Eastman Kodak Company Improved performance of photographic emulsions at high silver ion activities
JPH05249593A (ja) * 1992-03-04 1993-09-28 Konica Corp ハロゲン化銀写真感光材料
JPH07276810A (ja) * 1994-04-04 1995-10-24 Fuji Photo Film Co Ltd ジアゾ感熱記録材料

Also Published As

Publication number Publication date
EP1155002A4 (en) 2003-03-19
EP1155002A1 (en) 2001-11-21
AU3223200A (en) 2000-08-25
MXPA01007869A (es) 2003-06-04
JP2002536368A (ja) 2002-10-29
WO2000046211A1 (en) 2000-08-10

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued