AU2016293316A1 - 2-amino-1,3,4-thiadiazine and 2-amino-1,3,4-oxadiazine based antifungal agents - Google Patents
2-amino-1,3,4-thiadiazine and 2-amino-1,3,4-oxadiazine based antifungal agents Download PDFInfo
- Publication number
- AU2016293316A1 AU2016293316A1 AU2016293316A AU2016293316A AU2016293316A1 AU 2016293316 A1 AU2016293316 A1 AU 2016293316A1 AU 2016293316 A AU2016293316 A AU 2016293316A AU 2016293316 A AU2016293316 A AU 2016293316A AU 2016293316 A1 AU2016293316 A1 AU 2016293316A1
- Authority
- AU
- Australia
- Prior art keywords
- thiadiazin
- amine
- alkyl
- methoxy
- butyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- DUVVRISYWAVXBF-UHFFFAOYSA-N CCCC(C)OCCC1=NN=C(N)SC1 Chemical compound CCCC(C)OCCC1=NN=C(N)SC1 DUVVRISYWAVXBF-UHFFFAOYSA-N 0.000 description 1
- MMUTVMNWNNBCGK-UHFFFAOYSA-N CCCCCCCC1=CSC(N)=NN1 Chemical compound CCCCCCCC1=CSC(N)=NN1 MMUTVMNWNNBCGK-UHFFFAOYSA-N 0.000 description 1
- LEXRVWUCHOPIRB-UHFFFAOYSA-N CCOC(c1cc(C2=NN=C(N)SC2)ccc1)=O Chemical compound CCOC(c1cc(C2=NN=C(N)SC2)ccc1)=O LEXRVWUCHOPIRB-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/15—Six-membered rings
- C07D285/16—Thiadiazines; Hydrogenated thiadiazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/549—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame having two or more nitrogen atoms in the same ring, e.g. hydrochlorothiazide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB1512286.4 | 2015-07-14 | ||
| GBGB1512286.4A GB201512286D0 (en) | 2015-07-14 | 2015-07-14 | Chemical compounds |
| PCT/GB2016/052132 WO2017009651A1 (en) | 2015-07-14 | 2016-07-14 | 2-amino-1,3,4-thiadiazine and 2-amino-1,3,4-oxadiazine based antifungal agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2016293316A1 true AU2016293316A1 (en) | 2018-01-25 |
Family
ID=54013916
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2016293316A Abandoned AU2016293316A1 (en) | 2015-07-14 | 2016-07-14 | 2-amino-1,3,4-thiadiazine and 2-amino-1,3,4-oxadiazine based antifungal agents |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20180201592A1 (enExample) |
| EP (1) | EP3322705A1 (enExample) |
| JP (1) | JP2018527316A (enExample) |
| KR (1) | KR20180030166A (enExample) |
| CN (1) | CN108368102A (enExample) |
| AU (1) | AU2016293316A1 (enExample) |
| CA (1) | CA2991684A1 (enExample) |
| GB (1) | GB201512286D0 (enExample) |
| WO (1) | WO2017009651A1 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3610044B1 (en) * | 2017-04-12 | 2022-01-05 | Momentum Bioscience Limited | Detection and delineation of microorganisms using the ilv3 gene |
| CN108586273B (zh) * | 2018-03-07 | 2019-12-10 | 江南大学 | 一种盐酸普萘洛尔的制备方法 |
| CN120329218A (zh) * | 2025-06-23 | 2025-07-18 | 富祥(山东)新材料有限公司 | 一种抗hiv病毒类药物中间体的制备方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS428033Y1 (enExample) * | 1966-11-05 | 1967-04-24 | ||
| US3779736A (en) * | 1971-01-04 | 1973-12-18 | Gulf Research Development Co | 1,3,4-thiadiazine herbicides |
| JPS49110696A (enExample) * | 1973-03-10 | 1974-10-22 | ||
| US4254259A (en) * | 1978-11-02 | 1981-03-03 | Indiana University Foundation | 2-Amino-5-ethylovalyl-6H-1,3,4-thiadiazine oxime |
| JPS58177482A (ja) * | 1982-04-10 | 1983-10-18 | Mitsui Petrochem Ind Ltd | ２，６−ジ−ｔｅｒｔ−ブチル−４−アシロキシメチルフエノ−ルの製法 |
| WO2012006068A2 (en) * | 2010-06-28 | 2012-01-12 | President And Fellows Of Harvard College | Compounds for the inhibition of cellular proliferation |
| MX2015015421A (es) * | 2013-05-10 | 2016-06-21 | Nimbus Apollo Inc | Inhibidores de acetil-coa carboxilasa (acc) y usos de los mismos. |
-
2015
- 2015-07-14 GB GBGB1512286.4A patent/GB201512286D0/en not_active Ceased
-
2016
- 2016-07-14 CA CA2991684A patent/CA2991684A1/en not_active Abandoned
- 2016-07-14 AU AU2016293316A patent/AU2016293316A1/en not_active Abandoned
- 2016-07-14 JP JP2018500924A patent/JP2018527316A/ja active Pending
- 2016-07-14 US US15/744,510 patent/US20180201592A1/en not_active Abandoned
- 2016-07-14 EP EP16750201.2A patent/EP3322705A1/en not_active Withdrawn
- 2016-07-14 KR KR1020187004510A patent/KR20180030166A/ko not_active Withdrawn
- 2016-07-14 CN CN201680053383.6A patent/CN108368102A/zh active Pending
- 2016-07-14 WO PCT/GB2016/052132 patent/WO2017009651A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| EP3322705A1 (en) | 2018-05-23 |
| US20180201592A1 (en) | 2018-07-19 |
| JP2018527316A (ja) | 2018-09-20 |
| CA2991684A1 (en) | 2017-01-19 |
| WO2017009651A1 (en) | 2017-01-19 |
| KR20180030166A (ko) | 2018-03-21 |
| GB201512286D0 (en) | 2015-08-19 |
| CN108368102A (zh) | 2018-08-03 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| US7495018B2 (en) | Substituted 1,3-thiazole compounds, their production and use | |
| EP2484669B1 (en) | Phenol derivatives | |
| JP6386035B2 (ja) | 金属酵素阻害剤化合物 | |
| US20050080113A1 (en) | Medicinal compositions | |
| US8916584B2 (en) | Benzisoxazoles and azabenzisoxazoles as MGLUR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction | |
| US9180192B2 (en) | mGluR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction | |
| US20040063946A1 (en) | Jnk inhibitor | |
| EP1802583A1 (de) | Heterocyclische carbonylverbindungen | |
| US8486962B2 (en) | Antifungal agents | |
| KR20110031297A (ko) | 항진균 조합 치료방법 | |
| JPWO1998004534A1 (ja) | ６−フェニルテトラヒドロ−１，３−オキサジン−２−オン誘導体及びそれを含む医薬組成物 | |
| JP6284158B2 (ja) | 新規ピラゾール誘導体 | |
| RS61239B1 (sr) | Inhibitori aldozne reduktaze i postupci korišćenja | |
| JPWO2010007943A1 (ja) | 含窒素複素環化合物 | |
| JP2013532657A (ja) | 環式ｎ，ｎ’−ジアリールチオ尿素及びｎ，ｎ’−ジアリール尿素−アンドロゲン受容体アンタゴニスト、抗癌剤、その調製のための方法及び使用 | |
| WO2015189117A1 (de) | Heterobicyclisch substituierte 4-oxobutansäure-derivate und ihre verwendung | |
| WO2005092304A2 (en) | Antifungal agents | |
| AU2016293316A1 (en) | 2-amino-1,3,4-thiadiazine and 2-amino-1,3,4-oxadiazine based antifungal agents | |
| JPWO2007043568A1 (ja) | Ｓ１ｐ３受容体拮抗剤 | |
| DE60307804T2 (de) | Pyranon- und pyrandioninhibitoren der rna-abhängigen rna-polymerase des hepatitis-c-virus | |
| JP2023521237A (ja) | 抗ウイルス１，３－ジ－オキソ－インデン化合物 | |
| CN116102553A (zh) | 一种芳香稠环亚胺类化合物及其制备方法和应用 | |
| CA2980801A1 (en) | Pde10 inhibitors and related compositions and methods | |
| CN114671856A (zh) | 多取代的尿嘧啶衍生物及其用途 | |
| US20130303538A1 (en) | 4-Tolyl-ethynyl-octahydro-indole-1-ester derivatives |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK4 | Application lapsed section 142(2)(d) - no continuation fee paid for the application |