AU2016279099B2 - Pharmaceutical composition of carboplatin based co-crystals and use thereof - Google Patents

Pharmaceutical composition of carboplatin based co-crystals and use thereof Download PDF

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Publication number
AU2016279099B2
AU2016279099B2 AU2016279099A AU2016279099A AU2016279099B2 AU 2016279099 B2 AU2016279099 B2 AU 2016279099B2 AU 2016279099 A AU2016279099 A AU 2016279099A AU 2016279099 A AU2016279099 A AU 2016279099A AU 2016279099 B2 AU2016279099 B2 AU 2016279099B2
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AU
Australia
Prior art keywords
crystal
cancer
nmp
cbp
virus
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Ceased
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AU2016279099A
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English (en)
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AU2016279099A1 (en
Inventor
Xiaozhong Liu
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Syn Nat Products Enterprise LLC
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Syn Nat Products Enterprise LLC
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Publication of AU2016279099A1 publication Critical patent/AU2016279099A1/en
Application granted granted Critical
Publication of AU2016279099B2 publication Critical patent/AU2016279099B2/en
Ceased legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0086—Platinum compounds
    • C07F15/0093—Platinum compounds without a metal-carbon linkage
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/28—Compounds containing heavy metals
    • A61K31/282—Platinum compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
    • C07D207/263—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
    • C07D207/267—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU2016279099A 2015-06-19 2016-06-20 Pharmaceutical composition of carboplatin based co-crystals and use thereof Ceased AU2016279099B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562182142P 2015-06-19 2015-06-19
US62/182,142 2015-06-19
PCT/US2016/038340 WO2016205785A1 (en) 2015-06-19 2016-06-20 Pharmaceutical composition of carboplatin based co-crystals and use thereof

Publications (2)

Publication Number Publication Date
AU2016279099A1 AU2016279099A1 (en) 2018-01-04
AU2016279099B2 true AU2016279099B2 (en) 2021-09-23

Family

ID=57546414

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2016279099A Ceased AU2016279099B2 (en) 2015-06-19 2016-06-20 Pharmaceutical composition of carboplatin based co-crystals and use thereof

Country Status (9)

Country Link
US (1) US10421770B2 (enExample)
EP (1) EP3297636B1 (enExample)
JP (1) JP6768716B2 (enExample)
KR (1) KR20180018800A (enExample)
CN (1) CN107847508B (enExample)
AU (1) AU2016279099B2 (enExample)
BR (1) BR112017027285A2 (enExample)
CA (1) CA2988992A1 (enExample)
WO (1) WO2016205785A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3297624B1 (en) * 2015-05-18 2021-03-03 Syn-Nat Products Enterprise LLC A pharmaceutical co-crystal and use thereof
AU2016279099B2 (en) 2015-06-19 2021-09-23 Syn-Nat Products Enterprise LLC Pharmaceutical composition of carboplatin based co-crystals and use thereof
CN108697093A (zh) 2015-06-19 2018-10-23 新纳特产品公司 含卡铂的组合物及其用途
EP3297640A4 (en) 2015-06-25 2019-01-02 Syn-Nat Products Enterprise LLC Pharmaceutical co-crystal composition and use thereof

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7927613B2 (en) * 2002-02-15 2011-04-19 University Of South Florida Pharmaceutical co-crystal compositions

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AU2016250616B2 (en) 2015-04-22 2021-01-21 Syn-Nat Products Enterprise LLC Co-crystal composition and its pharmaceutical use
EP3297624B1 (en) 2015-05-18 2021-03-03 Syn-Nat Products Enterprise LLC A pharmaceutical co-crystal and use thereof
AU2016279099B2 (en) 2015-06-19 2021-09-23 Syn-Nat Products Enterprise LLC Pharmaceutical composition of carboplatin based co-crystals and use thereof
CN108697093A (zh) 2015-06-19 2018-10-23 新纳特产品公司 含卡铂的组合物及其用途
EP3297640A4 (en) 2015-06-25 2019-01-02 Syn-Nat Products Enterprise LLC Pharmaceutical co-crystal composition and use thereof

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7927613B2 (en) * 2002-02-15 2011-04-19 University Of South Florida Pharmaceutical co-crystal compositions

Also Published As

Publication number Publication date
US10421770B2 (en) 2019-09-24
CN107847508B (zh) 2020-10-02
EP3297636B1 (en) 2021-02-17
WO2016205785A1 (en) 2016-12-22
CA2988992A1 (en) 2016-12-22
KR20180018800A (ko) 2018-02-21
CN107847508A (zh) 2018-03-27
EP3297636A4 (en) 2018-11-14
JP2018524320A (ja) 2018-08-30
JP6768716B2 (ja) 2020-10-14
EP3297636A1 (en) 2018-03-28
AU2016279099A1 (en) 2018-01-04
US20180179240A1 (en) 2018-06-28
BR112017027285A2 (pt) 2018-09-11

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