AU2014278005B2 - Stabilized polypeptide insulin receptor modulators - Google Patents
Stabilized polypeptide insulin receptor modulators Download PDFInfo
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- AU2014278005B2 AU2014278005B2 AU2014278005A AU2014278005A AU2014278005B2 AU 2014278005 B2 AU2014278005 B2 AU 2014278005B2 AU 2014278005 A AU2014278005 A AU 2014278005A AU 2014278005 A AU2014278005 A AU 2014278005A AU 2014278005 B2 AU2014278005 B2 AU 2014278005B2
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Classifications
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- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
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- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/705—Receptors; Cell surface antigens; Cell surface determinants
- C07K14/72—Receptors; Cell surface antigens; Cell surface determinants for hormones
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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Landscapes
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- Peptides Or Proteins (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2019201247A AU2019201247A1 (en) | 2013-06-14 | 2019-02-22 | Stabilized polypeptide insulin receptor modulators |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361835242P | 2013-06-14 | 2013-06-14 | |
| US61/835,242 | 2013-06-14 | ||
| PCT/US2014/042329 WO2014201370A1 (en) | 2013-06-14 | 2014-06-13 | Stabilized polypeptide insulin receptor modulators |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| AU2019201247A Division AU2019201247A1 (en) | 2013-06-14 | 2019-02-22 | Stabilized polypeptide insulin receptor modulators |
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| US20150198619A1 (en) | 2012-09-25 | 2015-07-16 | The Walter And Eliza Hall Institute Of Medical Research | Structure of insulin in complex with n- and c-terminal regions of the insulin receptor alpha-chain |
| WO2014052647A2 (en) | 2012-09-26 | 2014-04-03 | President And Fellows Of Harvard College | Proline-locked stapled peptides and uses thereof |
| US20150225471A1 (en) | 2012-10-01 | 2015-08-13 | President And Fellows Of Harvard College | Stabilized polypeptide insulin receptor modulators |
| WO2014110420A1 (en) | 2013-01-10 | 2014-07-17 | Noliva Therapeutics Llc | Peptidomimetic compounds |
| EP3391898A3 (en) * | 2013-03-13 | 2019-02-13 | President and Fellows of Harvard College | Stapled and stitched polypeptides and uses thereof |
-
2014
- 2014-06-13 JP JP2016519683A patent/JP2016523241A/ja active Pending
- 2014-06-13 KR KR1020167000920A patent/KR20160019547A/ko not_active Withdrawn
- 2014-06-13 BR BR112015031277A patent/BR112015031277A2/pt not_active Application Discontinuation
- 2014-06-13 AU AU2014278005A patent/AU2014278005B2/en not_active Ceased
- 2014-06-13 MX MX2015017274A patent/MX2015017274A/es unknown
- 2014-06-13 CA CA2915354A patent/CA2915354A1/en not_active Abandoned
- 2014-06-13 EP EP14736234.7A patent/EP3008081B1/en not_active Not-in-force
- 2014-06-13 WO PCT/US2014/042329 patent/WO2014201370A1/en not_active Ceased
- 2014-06-13 US US14/898,222 patent/US10227390B2/en not_active Expired - Fee Related
- 2014-06-13 CN CN201480045052.9A patent/CN105492460A/zh active Pending
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2015
- 2015-12-13 IL IL243088A patent/IL243088B/en not_active IP Right Cessation
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2010121288A1 (en) * | 2009-04-22 | 2010-10-28 | Walter And Eliza Hall Institute Of Medical Research | STRUCTURE OF THE C-TERMINAL REGION OF THE INSULIN RECEPTOR α-CHAIN AND OF THE INSULIN-LIKE GROWTH FACTOR RECEPTOR α-CHAIN |
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| JOHN G. MENTING ET AL, "How insulin engages its primary binding site on the insulin receptor", NATURE, (2013-01-09), vol. 493, no. 7431, pages 241 - 245 * |
Also Published As
| Publication number | Publication date |
|---|---|
| HK1223945A1 (en) | 2017-08-11 |
| EP3008081B1 (en) | 2017-08-30 |
| CN105492460A (zh) | 2016-04-13 |
| MX2015017274A (es) | 2016-08-04 |
| EP3008081A1 (en) | 2016-04-20 |
| IL243088B (en) | 2018-12-31 |
| JP2016523241A (ja) | 2016-08-08 |
| AU2014278005A1 (en) | 2016-02-04 |
| CA2915354A1 (en) | 2014-12-18 |
| WO2014201370A1 (en) | 2014-12-18 |
| AU2019201247A1 (en) | 2019-03-14 |
| US10227390B2 (en) | 2019-03-12 |
| US20160215036A1 (en) | 2016-07-28 |
| KR20160019547A (ko) | 2016-02-19 |
| BR112015031277A2 (pt) | 2017-09-19 |
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