AU2013323435C1 - Apixaban liquid formulations - Google Patents
Apixaban liquid formulations Download PDFInfo
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- AU2013323435C1 AU2013323435C1 AU2013323435A AU2013323435A AU2013323435C1 AU 2013323435 C1 AU2013323435 C1 AU 2013323435C1 AU 2013323435 A AU2013323435 A AU 2013323435A AU 2013323435 A AU2013323435 A AU 2013323435A AU 2013323435 C1 AU2013323435 C1 AU 2013323435C1
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- Prior art keywords
- vehicle
- apixaban
- liquid formulation
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- 229960003886 apixaban Drugs 0.000 title claims abstract description 154
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Landscapes
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| US61/773,032 | 2013-03-05 | ||
| PCT/US2013/062051 WO2014052678A1 (en) | 2012-09-26 | 2013-09-26 | Apixaban liquid formulations |
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| EP2907507A1 (en) * | 2014-02-17 | 2015-08-19 | Sandoz Ag | Pharmaceutical composition comprising apixaban |
| WO2017221209A1 (en) | 2016-06-23 | 2017-12-28 | Lupin Limited | Pharmaceutical formulations of apixaban |
| DK3781132T3 (da) * | 2018-04-16 | 2024-04-22 | Bristol Myers Squibb Co | Apixabanformuleringer |
| CN112261935A (zh) | 2018-08-14 | 2021-01-22 | 江苏恒瑞医药股份有限公司 | 一种可注射的药物组合物及其制备方法 |
| US20220211689A1 (en) | 2019-11-13 | 2022-07-07 | Unison Pharmaceuticals Pvt. Ltd. | Orally disintegrating pharmaceutical compositions of apixaban |
| CA3202161A1 (en) | 2020-12-13 | 2022-06-16 | Matthaios VIDALIS | Liquid apixaban formulation in small dose volume |
| CN113384526A (zh) * | 2021-08-03 | 2021-09-14 | 合肥医工医药股份有限公司 | 一种稳定的阿哌沙班口服溶液制剂及其制备方法 |
| NL2029536B1 (en) | 2021-10-27 | 2023-05-26 | Pharma Data S A | Apixaban suspension and preparation method |
| EP4412586A1 (en) | 2021-10-27 | 2024-08-14 | Pharma-Data S.A. | Apixaban suspension and preparation method |
| US12194028B2 (en) * | 2022-03-09 | 2025-01-14 | Slayback Pharma Llc | Stable pharmaceutical compositions of apixaban |
| WO2023218482A1 (en) * | 2022-05-09 | 2023-11-16 | Syri Research Private Limited | Liquid oral formulation of apixaban or pharmaceutically acceptable salt thereof |
| US12213972B2 (en) * | 2022-07-27 | 2025-02-04 | Slayback Pharma Llc | Stable pharmaceutical compositions of apixaban |
| WO2024160789A1 (en) | 2023-01-30 | 2024-08-08 | Tap Pharmaceuticals Ag | Liquid pharmaceutical formulations of apixaban |
| US11833138B1 (en) | 2023-01-30 | 2023-12-05 | Tap Pharmaceuticals Ag | Liquid pharmaceutical formulations of apixaban |
| EP4450064A1 (en) | 2023-04-14 | 2024-10-23 | Novick BioSciences Private Limited | Apixaban compositions |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007022165A2 (en) * | 2005-08-17 | 2007-02-22 | Bristol-Myers Squibb Company | Factor xa inhibitor inclusion complex with cyclodextrin |
| WO2010147978A1 (en) * | 2009-06-16 | 2010-12-23 | Pfizer Inc. | Dosage forms of apixaban |
| WO2011106478A2 (en) * | 2010-02-25 | 2011-09-01 | Bristol-Myers Squibb Company | Apixaban formulations |
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| US5763449A (en) * | 1996-08-07 | 1998-06-09 | Ascent Pediatrics, Inc. | Pleasant-tasting aqueous liquid composition of a bitter-tasting drug |
| CZ20022047A3 (cs) | 1999-12-23 | 2003-09-17 | Pfizer Products Inc. | Farmaceutické kompozice poskytující zvýšenou koncentraci léčiva |
| MY129350A (en) * | 2001-04-25 | 2007-03-30 | Bristol Myers Squibb Co | Aripiprazole oral solution |
| EP1269994A3 (en) | 2001-06-22 | 2003-02-12 | Pfizer Products Inc. | Pharmaceutical compositions comprising drug and concentration-enhancing polymers |
| TWI331526B (en) | 2001-09-21 | 2010-10-11 | Bristol Myers Squibb Pharma Co | Lactam-containing compounds and derivatives thereof as factor xa inhibitors |
| SI1427415T1 (sl) * | 2001-09-21 | 2009-12-31 | Bristol Myers Squibb Co | Sestavine, ki vsebujejo laktame in njihovi derivati kot inhibitorji faktorja xa |
| US7101572B2 (en) * | 2001-12-07 | 2006-09-05 | Unilab Pharmatech, Ltd. | Taste masked aqueous liquid pharmaceutical composition |
| CA2597155A1 (en) * | 2005-02-25 | 2006-09-08 | Biomarin Pharmaceutical Inc. | Room temperature stable aqueous liquid pharmaceutical composition |
| CA2712120A1 (en) * | 2008-01-14 | 2009-07-23 | Foamix Ltd. | Poloxamer foamable pharmaceutical compositions with active agents and/or therapeutic cells and uses |
| DK3100728T3 (da) * | 2009-05-13 | 2020-02-17 | Cydex Pharmaceuticals Inc | Farmaceutiske sammensætninger omfattende prasugrel og cyclodextrin-derivativ og fremgangsmåder til fremstilling og brug af samme |
| EP2484775A1 (de) | 2011-02-07 | 2012-08-08 | Siemens Healthcare Diagnostics Products GmbH | Heparin-insensitives Verfahren zur Bestimmung von direkten Gerinnungsfaktorinhibitoren |
| RU2638155C1 (ru) * | 2016-02-29 | 2017-12-12 | Общество С Ограниченной Ответственностью "Сай Фарма" | Производные бензо[d]изоксазола и их применение |
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Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007022165A2 (en) * | 2005-08-17 | 2007-02-22 | Bristol-Myers Squibb Company | Factor xa inhibitor inclusion complex with cyclodextrin |
| WO2010147978A1 (en) * | 2009-06-16 | 2010-12-23 | Pfizer Inc. | Dosage forms of apixaban |
| WO2011106478A2 (en) * | 2010-02-25 | 2011-09-01 | Bristol-Myers Squibb Company | Apixaban formulations |
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| IL237804A0 (en) | 2015-05-31 |
| HK1212900A1 (zh) | 2016-06-24 |
| US20160263097A1 (en) | 2016-09-15 |
| SG10201702048VA (en) | 2017-04-27 |
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