MX2020010673A - Formulaciones de apixaban. - Google Patents
Formulaciones de apixaban.Info
- Publication number
- MX2020010673A MX2020010673A MX2020010673A MX2020010673A MX2020010673A MX 2020010673 A MX2020010673 A MX 2020010673A MX 2020010673 A MX2020010673 A MX 2020010673A MX 2020010673 A MX2020010673 A MX 2020010673A MX 2020010673 A MX2020010673 A MX 2020010673A
- Authority
- MX
- Mexico
- Prior art keywords
- apixaban
- apixaban formulations
- formulations
- formulation
- treatment
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
- A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
- A61K9/1676—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4808—Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4816—Wall or shell material
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4816—Wall or shell material
- A61K9/4825—Proteins, e.g. gelatin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Hematology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Se proporciona la formulación farmacéutica de apixaban. También se proporciona un uso de la formulación de apixaban en el tratamiento de un trastorno tromboembólico.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201862658175P | 2018-04-16 | 2018-04-16 | |
PCT/US2019/027456 WO2019204193A1 (en) | 2018-04-16 | 2019-04-15 | Apixaban formulations |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2020010673A true MX2020010673A (es) | 2020-10-28 |
Family
ID=66429558
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2020010673A MX2020010673A (es) | 2018-04-16 | 2019-04-15 | Formulaciones de apixaban. |
Country Status (15)
Country | Link |
---|---|
US (1) | US11896586B2 (es) |
EP (2) | EP3781132B1 (es) |
JP (1) | JP7382957B2 (es) |
AU (1) | AU2019255599B2 (es) |
BR (1) | BR112020020941A2 (es) |
CA (1) | CA3097176A1 (es) |
DK (1) | DK3781132T3 (es) |
FI (1) | FI3781132T3 (es) |
LT (1) | LT3781132T (es) |
MX (1) | MX2020010673A (es) |
PL (1) | PL3781132T3 (es) |
PT (1) | PT3781132T (es) |
RS (1) | RS65428B1 (es) |
SG (1) | SG11202010097WA (es) |
WO (1) | WO2019204193A1 (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW202140003A (zh) * | 2020-02-13 | 2021-11-01 | 大陸商江蘇恒瑞醫藥股份有限公司 | 阿哌沙班注射劑用於預防或者治療血栓栓塞的方法 |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU670567B2 (en) * | 1992-03-05 | 1996-07-25 | American Home Products Corporation | Pharmaceutical coated cores |
PT969821E (pt) * | 1997-03-26 | 2003-10-31 | Janssen Pharmaceutica Nv | Pastilhas tendo um nucleo revestido com um antifungico e um polimero |
TWI331526B (en) | 2001-09-21 | 2010-10-11 | Bristol Myers Squibb Pharma Co | Lactam-containing compounds and derivatives thereof as factor xa inhibitors |
AU2010260208B2 (en) | 2009-06-16 | 2014-11-13 | Bristol-Myers Squibb Holdings Ireland Unlimited Company | Dosage forms of apixaban |
EP2538925B1 (en) | 2010-02-25 | 2015-12-16 | Bristol-Myers Squibb Company | Apixaban formulations |
EP2554159A1 (en) * | 2011-08-04 | 2013-02-06 | ratiopharm GmbH | Dosage forms comprising apixaban and content uniformity enhancer |
MX351059B (es) * | 2012-08-17 | 2017-09-29 | Laboratorios Senosiain S A De C V Star | Composicion farmaceutica oral en forma de microesferas y proceso de elaboracion. |
EP2900217A1 (en) * | 2012-09-26 | 2015-08-05 | Bristol-Myers Squibb Company | Apixaban liquid formulations |
CN105663049A (zh) | 2014-11-22 | 2016-06-15 | 哈尔滨圣吉药业股份有限公司 | 一种阿哌沙班缓释微丸及其制备方法 |
US10413543B2 (en) * | 2015-09-01 | 2019-09-17 | Sun Pharma Advanced Research Company Ltd. | Stable multiparticulate pharmaceutical composition of rosuvastatin |
CN106913528A (zh) * | 2015-12-25 | 2017-07-04 | 中美华世通生物医药科技(武汉)有限公司 | 阿哌沙班微丸及其制备方法 |
-
2019
- 2019-04-15 EP EP19722333.2A patent/EP3781132B1/en active Active
- 2019-04-15 RS RS20240457A patent/RS65428B1/sr unknown
- 2019-04-15 WO PCT/US2019/027456 patent/WO2019204193A1/en unknown
- 2019-04-15 AU AU2019255599A patent/AU2019255599B2/en active Active
- 2019-04-15 EP EP24159997.6A patent/EP4353312A2/en active Pending
- 2019-04-15 FI FIEP19722333.2T patent/FI3781132T3/fi active
- 2019-04-15 PT PT197223332T patent/PT3781132T/pt unknown
- 2019-04-15 US US17/047,428 patent/US11896586B2/en active Active
- 2019-04-15 DK DK19722333.2T patent/DK3781132T3/da active
- 2019-04-15 MX MX2020010673A patent/MX2020010673A/es unknown
- 2019-04-15 PL PL19722333.2T patent/PL3781132T3/pl unknown
- 2019-04-15 SG SG11202010097WA patent/SG11202010097WA/en unknown
- 2019-04-15 BR BR112020020941-4A patent/BR112020020941A2/pt unknown
- 2019-04-15 CA CA3097176A patent/CA3097176A1/en active Pending
- 2019-04-15 LT LTEPPCT/US2019/027456T patent/LT3781132T/lt unknown
- 2019-04-15 JP JP2020556976A patent/JP7382957B2/ja active Active
Also Published As
Publication number | Publication date |
---|---|
EP3781132B1 (en) | 2024-03-20 |
CA3097176A1 (en) | 2019-10-24 |
RS65428B1 (sr) | 2024-05-31 |
FI3781132T3 (fi) | 2024-05-31 |
EP4353312A2 (en) | 2024-04-17 |
PL3781132T3 (pl) | 2024-05-20 |
EP3781132A1 (en) | 2021-02-24 |
SG11202010097WA (en) | 2020-11-27 |
AU2019255599B2 (en) | 2024-02-29 |
US11896586B2 (en) | 2024-02-13 |
BR112020020941A2 (pt) | 2021-03-02 |
JP2021521242A (ja) | 2021-08-26 |
US20210145817A1 (en) | 2021-05-20 |
AU2019255599A1 (en) | 2020-11-12 |
WO2019204193A1 (en) | 2019-10-24 |
JP7382957B2 (ja) | 2023-11-17 |
LT3781132T (lt) | 2024-04-25 |
PT3781132T (pt) | 2024-05-16 |
DK3781132T3 (da) | 2024-04-22 |
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