AU2012322835A1 - Guanidinyl-substituted polyamides useful for treating human papilloma virus - Google Patents
Guanidinyl-substituted polyamides useful for treating human papilloma virus Download PDFInfo
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- AU2012322835A1 AU2012322835A1 AU2012322835A AU2012322835A AU2012322835A1 AU 2012322835 A1 AU2012322835 A1 AU 2012322835A1 AU 2012322835 A AU2012322835 A AU 2012322835A AU 2012322835 A AU2012322835 A AU 2012322835A AU 2012322835 A1 AU2012322835 A1 AU 2012322835A1
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- compound
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
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- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
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- A—HUMAN NECESSITIES
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- A61P31/20—Antivirals for DNA viruses
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
- A61P31/22—Antivirals for DNA viruses for herpes viruses
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/001—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof by chemical synthesis
- C07K14/003—Peptide-nucleic acids (PNAs)
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- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Virology (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Biochemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Genetics & Genomics (AREA)
- Engineering & Computer Science (AREA)
- Biotechnology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Gastroenterology & Hepatology (AREA)
- Biophysics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Polyamides (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Investigating Or Analysing Biological Materials (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Materials For Medical Uses (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161545311P | 2011-10-10 | 2011-10-10 | |
| US61/545,311 | 2011-10-10 | ||
| PCT/US2012/059604 WO2013055825A2 (en) | 2011-10-10 | 2012-10-10 | Guanidinyl-substituted polyamides useful for treating human papilloma virus |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2012322835A1 true AU2012322835A1 (en) | 2014-04-17 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2012322835A Abandoned AU2012322835A1 (en) | 2011-10-10 | 2012-10-10 | Guanidinyl-substituted polyamides useful for treating human papilloma virus |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US9133228B2 (enExample) |
| EP (1) | EP2751096A4 (enExample) |
| JP (1) | JP2015502330A (enExample) |
| KR (1) | KR20140074996A (enExample) |
| CN (1) | CN104024247B (enExample) |
| AU (1) | AU2012322835A1 (enExample) |
| BR (1) | BR112014008464A2 (enExample) |
| CA (1) | CA2851516C (enExample) |
| HK (1) | HK1201064A1 (enExample) |
| RU (1) | RU2014113702A (enExample) |
| SG (1) | SG11201401226YA (enExample) |
| WO (1) | WO2013055825A2 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US9982020B2 (en) * | 2011-10-10 | 2018-05-29 | Nanovir Llc | Antiviral compounds and methods for treating infections caused by double-stranded DNA viruses |
| WO2016022664A1 (en) * | 2014-08-05 | 2016-02-11 | Nanovir Llc | Antiviral compounds and methods for treating infections caused by double-stranded dna viruses |
| US20220193241A1 (en) * | 2019-03-20 | 2022-06-23 | Chiba-Prefecture | Agent targeting double-membrane organelle dna |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
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| AU7380294A (en) | 1993-08-06 | 1995-02-28 | Synphar Laboratories, Inc. | Oligopeptide antiretroviral agents |
| EP0973740A1 (en) | 1996-02-26 | 2000-01-26 | California Institute Of Technology | Design, synthesis and use of specific polyamide dna-binding ligands |
| CN1260006A (zh) | 1996-02-26 | 2000-07-12 | 加利福尼亚州技术学院 | 双链dna和杂环低聚物之间复合物的形成 |
| AU734715B2 (en) | 1996-02-26 | 2001-06-21 | California Institute Of Technology | Improved polyamides for binding in the minor groove of double stranded DNA |
| US5998140A (en) | 1996-07-31 | 1999-12-07 | The Scripps Research Institute | Complex formation between dsDNA and oligomer of cyclic heterocycles |
| JP2002515057A (ja) | 1996-08-01 | 2002-05-21 | カリフォルニア・インスティチュート・オブ・テクノロジー | ポリアミドｄｎａ結合リガンドによる遺伝子発現の阻害 |
| AU5910899A (en) | 1998-09-11 | 2000-04-03 | California Institute Of Technology | Inhibition of oncogene transcription by synthetic polyamides |
| US6673940B1 (en) | 1999-01-08 | 2004-01-06 | California Institute Of Technology | Compositions and methods relating to cyclic compounds that undergo nucleotide base pair-specific interactions with double-stranded nucleic acids |
| JP4012145B2 (ja) | 2001-06-25 | 2007-11-21 | 独立行政法人科学技術振興機構 | ピロール−イミダゾールポリアミドの固相合成法 |
| AU2002363523A1 (en) | 2001-11-07 | 2003-05-19 | Pharmacia Corporation | Methods of promoting uptake and nuclear accumulation of polyamides in eukaryotic cells |
| BR0213988A (pt) | 2001-11-07 | 2004-08-31 | Pharmacia Corp | Moduladores de poliamida de transcrição de cox2 |
| ATE468147T1 (de) | 2003-01-16 | 2010-06-15 | Femmepharma Holding Co Inc | Vaginaler oder rektaler applikator und verfahren |
| WO2004078943A2 (en) | 2003-03-04 | 2004-09-16 | California Institute Of Technology | Alternative heterocycles for dna recognition |
| MXPA05011642A (es) | 2003-04-30 | 2005-12-15 | Pharmacia Corp | Compuestos que tienen un resto biciclico condensado para unirse al surco menor del adn de doble hebra. |
| US8399013B2 (en) | 2003-06-26 | 2013-03-19 | Poly-Med, Inc. | Partially absorbable fiber-reinforced composites for controlled drug delivery |
| WO2005033282A2 (en) | 2003-10-01 | 2005-04-14 | Pharmacia & Upjohn Company Llc | Polyamide compositions and therapeutic methods for treatment of human papilloma virus |
| DE10357677A1 (de) * | 2003-12-10 | 2005-07-14 | Greiner Bio-One Gmbh | Primer und Sonden zum Nachweis genitaler HPV-Genotypen |
| WO2007045096A1 (en) * | 2005-10-21 | 2007-04-26 | University Of Saskatchewan | Oligoheteroaromatic luminiscent assemblies as high-affinity dna sequence-directed ligands |
| WO2007103584A2 (en) | 2006-03-09 | 2007-09-13 | Nanovir, Llc | Polyamides for treating human papilloma virus |
| US8993609B2 (en) | 2006-05-04 | 2015-03-31 | Nanovir, Llc | Compounds for treating papilloma virus infection |
| WO2007130616A2 (en) | 2006-05-04 | 2007-11-15 | Nanovir, Llc | Polyamides for treating human papilloma virus |
-
2012
- 2012-10-10 RU RU2014113702/04A patent/RU2014113702A/ru not_active Application Discontinuation
- 2012-10-10 JP JP2014534836A patent/JP2015502330A/ja active Pending
- 2012-10-10 US US13/649,000 patent/US9133228B2/en not_active Expired - Fee Related
- 2012-10-10 HK HK15101532.6A patent/HK1201064A1/xx unknown
- 2012-10-10 BR BR112014008464A patent/BR112014008464A2/pt not_active IP Right Cessation
- 2012-10-10 AU AU2012322835A patent/AU2012322835A1/en not_active Abandoned
- 2012-10-10 CA CA2851516A patent/CA2851516C/en active Active
- 2012-10-10 EP EP12840685.7A patent/EP2751096A4/en not_active Withdrawn
- 2012-10-10 KR KR1020147012415A patent/KR20140074996A/ko not_active Ceased
- 2012-10-10 SG SG11201401226YA patent/SG11201401226YA/en unknown
- 2012-10-10 WO PCT/US2012/059604 patent/WO2013055825A2/en not_active Ceased
- 2012-10-10 CN CN201280049712.1A patent/CN104024247B/zh not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP2015502330A (ja) | 2015-01-22 |
| EP2751096A4 (en) | 2015-04-08 |
| WO2013055825A2 (en) | 2013-04-18 |
| US20130090362A1 (en) | 2013-04-11 |
| CN104024247A (zh) | 2014-09-03 |
| RU2014113702A (ru) | 2015-11-20 |
| CA2851516C (en) | 2016-08-02 |
| US9133228B2 (en) | 2015-09-15 |
| CA2851516A1 (en) | 2013-04-18 |
| EP2751096A2 (en) | 2014-07-09 |
| NZ623292A (en) | 2016-02-26 |
| CN104024247B (zh) | 2016-05-25 |
| HK1201064A1 (en) | 2015-08-21 |
| BR112014008464A2 (pt) | 2017-04-11 |
| KR20140074996A (ko) | 2014-06-18 |
| WO2013055825A3 (en) | 2013-06-13 |
| SG11201401226YA (en) | 2014-05-29 |
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Legal Events
| Date | Code | Title | Description |
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| MK4 | Application lapsed section 142(2)(d) - no continuation fee paid for the application |