AU2012207818B2 - Orally dispersible tablet - Google Patents
Orally dispersible tablet Download PDFInfo
- Publication number
- AU2012207818B2 AU2012207818B2 AU2012207818A AU2012207818A AU2012207818B2 AU 2012207818 B2 AU2012207818 B2 AU 2012207818B2 AU 2012207818 A AU2012207818 A AU 2012207818A AU 2012207818 A AU2012207818 A AU 2012207818A AU 2012207818 B2 AU2012207818 B2 AU 2012207818B2
- Authority
- AU
- Australia
- Prior art keywords
- oral
- preparation
- indeno
- tetrahydro
- administration
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2063—Proteins, e.g. gelatin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D307/81—Radicals substituted by nitrogen atoms not forming part of a nitro radical
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physiology (AREA)
- Nutrition Science (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Zoology (AREA)
- Pain & Pain Management (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2013203069A AU2013203069A1 (en) | 2011-01-17 | 2013-04-09 | Orally dispersible tablet |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2011-007371 | 2011-01-17 | ||
| JP2011007371 | 2011-01-17 | ||
| JP2011-227333 | 2011-10-14 | ||
| JP2011227333 | 2011-10-14 | ||
| PCT/JP2012/051279 WO2012099260A1 (en) | 2011-01-17 | 2012-01-16 | Orally dispersible tablet |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2013203069A Division AU2013203069A1 (en) | 2011-01-17 | 2013-04-09 | Orally dispersible tablet |
Publications (2)
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|---|---|
| AU2012207818A1 AU2012207818A1 (en) | 2013-05-02 |
| AU2012207818B2 true AU2012207818B2 (en) | 2015-05-14 |
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Family Applications (1)
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| AU2012207818A Ceased AU2012207818B2 (en) | 2011-01-17 | 2012-01-16 | Orally dispersible tablet |
Country Status (24)
| Country | Link |
|---|---|
| US (6) | US20120282191A1 (enExample) |
| EP (1) | EP2665465A1 (enExample) |
| JP (3) | JP5600747B2 (enExample) |
| KR (1) | KR20140014134A (enExample) |
| CN (1) | CN103429223A (enExample) |
| AR (1) | AR084865A1 (enExample) |
| AU (1) | AU2012207818B2 (enExample) |
| BR (1) | BR112013017600A2 (enExample) |
| CA (1) | CA2824430A1 (enExample) |
| CL (1) | CL2013002033A1 (enExample) |
| CO (1) | CO6791611A2 (enExample) |
| CR (1) | CR20130380A (enExample) |
| EA (1) | EA201391053A1 (enExample) |
| EC (1) | ECSP13012825A (enExample) |
| IL (1) | IL227357A0 (enExample) |
| MA (1) | MA34908B1 (enExample) |
| MX (1) | MX2013008314A (enExample) |
| PE (1) | PE20140255A1 (enExample) |
| PH (1) | PH12013501512A1 (enExample) |
| SG (1) | SG191964A1 (enExample) |
| TW (1) | TW201309347A (enExample) |
| UY (1) | UY33869A (enExample) |
| WO (1) | WO2012099260A1 (enExample) |
| ZA (1) | ZA201305567B (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012103411A2 (en) | 2011-01-28 | 2012-08-02 | Zx Pharma, Llc | Controlled-release melatonin composition and related methods |
| US9532952B2 (en) | 2011-01-28 | 2017-01-03 | Physician's Seal, LLC | Controlled-release compositions of melatonin combined with sedative and/or analgesic ingredients |
| JP6245677B2 (ja) * | 2012-01-20 | 2017-12-13 | ニプロ株式会社 | 口腔内崩壊錠 |
| CN103989643B (zh) * | 2013-07-26 | 2018-10-30 | 武汉先路医药科技有限公司 | 含有雷美替胺和共聚维酮的片剂 |
| HK1222796A1 (zh) * | 2013-07-31 | 2017-07-14 | 因特根克斯公司 | 不含表面活性剂或多元醇的即时可湿性口服薄膜剂型 |
| CN105007904A (zh) * | 2014-02-07 | 2015-10-28 | 科学实验室药物公司 | 全天然无毒舌下药物递送系统 |
| CN106389361A (zh) * | 2016-03-31 | 2017-02-15 | 北京万全德众医药生物技术有限公司 | 一种含有雷美替胺的口腔崩解片及其制备方法 |
| CN105853379A (zh) * | 2016-03-31 | 2016-08-17 | 北京万全德众医药生物技术有限公司 | 一种雷美替胺分散片及其制备工艺 |
| CA3023305C (en) | 2016-05-06 | 2024-07-02 | Societe Des Produits Nestle S.A. | COMPOSITION OF VALERIAN AND ASSOCIATED PROCESSES |
| CN106038502A (zh) * | 2016-07-01 | 2016-10-26 | 北京万全德众医药生物技术有限公司 | 一种雷美替胺口崩片及其制备方法 |
| US20210113456A1 (en) * | 2017-07-13 | 2021-04-22 | Maxinase Life Sciences Limited | Pharmaceutical compositions of ramelteon and methods of use thereof |
| US11648201B2 (en) | 2018-05-02 | 2023-05-16 | Ferring B.V. | Pharmaceutical formulations |
| JP7552146B2 (ja) * | 2019-08-28 | 2024-09-18 | 小野薬品工業株式会社 | イバブラジンを含有する錠剤 |
| CN113243444A (zh) * | 2020-02-13 | 2021-08-13 | 罗盖特公司 | 作为口香糖中的填充剂的多孔淀粉 |
| JP7611556B2 (ja) * | 2020-05-28 | 2025-01-10 | 日医工株式会社 | 服用性、安定性等に優れた医薬組成物 |
| CN115778925A (zh) * | 2022-12-26 | 2023-03-14 | 湖北广济医药科技有限公司 | 一种雷美替胺口溶膜剂及其制备方法 |
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| US20090105490A1 (en) * | 2007-07-12 | 2009-04-23 | Nurit Perlman | Polymorphic forms of ramelteon and processes for preparation thereof |
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| JP3460538B2 (ja) | 1997-10-08 | 2003-10-27 | 救急薬品工業株式会社 | 速溶性フィルム製剤 |
| EP1153616B1 (en) | 1999-02-15 | 2004-12-01 | Sumitomo Pharmaceuticals Company, Limited | Tablets quickly disintegrated in the oral cavity |
| CA2381860C (en) * | 1999-08-26 | 2009-11-24 | Takeda Chemical Industries, Ltd. | Matrix adhering to nasal mucosa |
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-
2012
- 2012-01-16 MX MX2013008314A patent/MX2013008314A/es unknown
- 2012-01-16 SG SG2013053772A patent/SG191964A1/en unknown
- 2012-01-16 MA MA36182A patent/MA34908B1/fr unknown
- 2012-01-16 US US13/261,266 patent/US20120282191A1/en not_active Abandoned
- 2012-01-16 KR KR1020137021442A patent/KR20140014134A/ko not_active Withdrawn
- 2012-01-16 PH PH1/2013/501512A patent/PH12013501512A1/en unknown
- 2012-01-16 EP EP12702894.2A patent/EP2665465A1/en not_active Withdrawn
- 2012-01-16 CA CA2824430A patent/CA2824430A1/en not_active Abandoned
- 2012-01-16 WO PCT/JP2012/051279 patent/WO2012099260A1/en not_active Ceased
- 2012-01-16 AR ARP120100142A patent/AR084865A1/es unknown
- 2012-01-16 JP JP2012535507A patent/JP5600747B2/ja not_active Expired - Fee Related
- 2012-01-16 AU AU2012207818A patent/AU2012207818B2/en not_active Ceased
- 2012-01-16 EA EA201391053A patent/EA201391053A1/ru unknown
- 2012-01-16 TW TW101101549A patent/TW201309347A/zh unknown
- 2012-01-16 UY UY0001033869A patent/UY33869A/es not_active Application Discontinuation
- 2012-01-16 CN CN2012800138646A patent/CN103429223A/zh active Pending
- 2012-01-16 BR BR112013017600A patent/BR112013017600A2/pt not_active IP Right Cessation
- 2012-01-16 PE PE2013001568A patent/PE20140255A1/es not_active Application Discontinuation
- 2012-10-09 US US13/647,788 patent/US8642649B2/en not_active Expired - Fee Related
- 2012-10-09 US US13/647,784 patent/US8642648B2/en not_active Expired - Fee Related
-
2013
- 2013-07-07 IL IL227357A patent/IL227357A0/en unknown
- 2013-07-12 CL CL2013002033A patent/CL2013002033A1/es unknown
- 2013-07-23 ZA ZA2013/05567A patent/ZA201305567B/en unknown
- 2013-08-07 CR CR20130380A patent/CR20130380A/es unknown
- 2013-08-13 EC ECSP13012825 patent/ECSP13012825A/es unknown
- 2013-08-16 CO CO13195977A patent/CO6791611A2/es not_active Application Discontinuation
-
2014
- 2014-01-30 US US14/168,392 patent/US20140235709A1/en not_active Abandoned
- 2014-01-30 US US14/168,400 patent/US20140235879A1/en not_active Abandoned
- 2014-07-01 JP JP2014136302A patent/JP2014198723A/ja active Pending
-
2016
- 2016-01-15 JP JP2016006663A patent/JP2016053094A/ja active Pending
- 2016-11-18 US US15/355,357 patent/US20170065553A1/en not_active Abandoned
Patent Citations (6)
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|---|---|---|---|---|
| EP0914818A1 (en) * | 1996-06-14 | 1999-05-12 | Kyowa Hakko Kogyo Co., Ltd. | Intraorally rapidly disintegrable tablet |
| WO1999059544A2 (en) * | 1998-05-18 | 1999-11-25 | Takeda Chemical Industries, Ltd. | Orally disintegrable tablets |
| EP1867641A1 (en) * | 2005-04-04 | 2007-12-19 | Takeda Pharmaceutical Company Limited | Preventive or remedy for depression or anxiety neurosis |
| US20070134331A1 (en) * | 2005-12-14 | 2007-06-14 | Les Laboratoires Servier | Orodispersible pharmaceutical composition for oromucosal or sublingual administration of agomelatine |
| WO2008083204A2 (en) * | 2006-12-28 | 2008-07-10 | Braincells, Inc. | Modulation of neurogenesis by melatoninergic ligands |
| US20090105490A1 (en) * | 2007-07-12 | 2009-04-23 | Nurit Perlman | Polymorphic forms of ramelteon and processes for preparation thereof |
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