AU2011293612B2 - Aminopyridine- and aminopyrimidinecarboxamides as CXCR2 modulators - Google Patents

Aminopyridine- and aminopyrimidinecarboxamides as CXCR2 modulators Download PDF

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AU2011293612B2
AU2011293612B2 AU2011293612A AU2011293612A AU2011293612B2 AU 2011293612 B2 AU2011293612 B2 AU 2011293612B2 AU 2011293612 A AU2011293612 A AU 2011293612A AU 2011293612 A AU2011293612 A AU 2011293612A AU 2011293612 B2 AU2011293612 B2 AU 2011293612B2
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Dean Y. Maeda
Aaron D. Schuler
John A. Zebala
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Syntrix Biosystems Inc
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AU2011293612A 2010-08-23 2011-08-22 Aminopyridine- and aminopyrimidinecarboxamides as CXCR2 modulators Active AU2011293612B2 (en)

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US8748623B2 (en) 2009-02-17 2014-06-10 Syntrix Biosystems, Inc. Pyridinecarboxamides as CXCR2 modulators
CA2811990C (en) * 2010-08-23 2023-03-21 Dean Y. Maeda Aminopyridine- and aminopyrimidinecarboxamides as cxcr2 modulators
WO2014205127A2 (en) 2013-06-18 2014-12-24 New York University Cellular factors involved in the cytotoxicity of staphylococcus aureus leukocidins: novel therapeutic targets
EP3027627B1 (en) * 2013-08-02 2018-01-31 Syntrix Biosystems Inc. 2-[5-[n-(4-fluorophenyl)carbamoyl]pyrimidin-2-ylsulfanylmethyl]-4-(trifluoromethoxy)phenyl]boronic acid
US10046002B2 (en) 2013-08-02 2018-08-14 Syntrix Biosystems Inc. Method for treating cancer using chemokine antagonists
US8969365B2 (en) 2013-08-02 2015-03-03 Syntrix Biosystems, Inc. Thiopyrimidinecarboxamides as CXCR1/2 modulators
US10561676B2 (en) 2013-08-02 2020-02-18 Syntrix Biosystems Inc. Method for treating cancer using dual antagonists of CXCR1 and CXCR2
WO2017070589A1 (en) * 2015-10-22 2017-04-27 Duke University Methods and compositions for the diagnosis and treatment of central nervous system autoimmune diseases
CN109152780B (zh) * 2016-03-11 2021-10-01 阿迪亚生命科学公司 用于治疗结晶性关节病症的cxcr-2抑制剂
WO2018071687A1 (en) * 2016-10-13 2018-04-19 The Regents Of The University Of California Methods of treating pruritis
US10660909B2 (en) 2016-11-17 2020-05-26 Syntrix Biosystems Inc. Method for treating cancer using chemokine antagonists
WO2021163683A1 (en) 2020-02-14 2021-08-19 President And Fellows Of Harvard College Inhibitors of nicotinamide n-methyltransferase, compositions and uses thereof
WO2024218236A1 (en) 2023-04-18 2024-10-24 Centre National De La Recherche Scientifique 3,5-diaminotriazole derivatives and uses thereof for treating ocular diseases

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