AU2011293612B2 - Aminopyridine- and aminopyrimidinecarboxamides as CXCR2 modulators - Google Patents

Aminopyridine- and aminopyrimidinecarboxamides as CXCR2 modulators Download PDF

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AU2011293612B2
AU2011293612B2 AU2011293612A AU2011293612A AU2011293612B2 AU 2011293612 B2 AU2011293612 B2 AU 2011293612B2 AU 2011293612 A AU2011293612 A AU 2011293612A AU 2011293612 A AU2011293612 A AU 2011293612A AU 2011293612 B2 AU2011293612 B2 AU 2011293612B2
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Dean Y. Maeda
Aaron D. Schuler
John A. Zebala
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Syntrix Biosystems Inc
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AU2011293612A 2010-08-23 2011-08-22 Aminopyridine- and aminopyrimidinecarboxamides as CXCR2 modulators Active AU2011293612B2 (en)

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AU2011293612B2 (en) * 2010-08-23 2015-11-26 Syntrix Biosystems Inc. Aminopyridine- and aminopyrimidinecarboxamides as CXCR2 modulators
US10301378B2 (en) 2013-06-18 2019-05-28 New York University Cellular factors involved in the cytotoxicity of Staphylococcus aureus leukocidins: novel therapeutic targets
US10046002B2 (en) 2013-08-02 2018-08-14 Syntrix Biosystems Inc. Method for treating cancer using chemokine antagonists
US10561676B2 (en) 2013-08-02 2020-02-18 Syntrix Biosystems Inc. Method for treating cancer using dual antagonists of CXCR1 and CXCR2
US8969365B2 (en) 2013-08-02 2015-03-03 Syntrix Biosystems, Inc. Thiopyrimidinecarboxamides as CXCR1/2 modulators
ES2671927T3 (es) * 2013-08-02 2018-06-11 Syntrix Biosystems Inc. Ácido 2-[5-[N-(4-fluorofenil)carbamoil]pirimidin-2-ilsulfanilmetil]-4-(trifluorometoxi)fenil]borónico
WO2017070589A1 (en) * 2015-10-22 2017-04-27 Duke University Methods and compositions for the diagnosis and treatment of central nervous system autoimmune diseases
CA3017345A1 (en) * 2016-03-11 2017-09-14 Ardea Biosciences, Inc. Cxcr-2 inhibitors for treating crystal arthropathy disorders
US20190216790A1 (en) * 2016-10-13 2019-07-18 The Regents Of The University Of California Methods for Treating Pruritis
US10660909B2 (en) 2016-11-17 2020-05-26 Syntrix Biosystems Inc. Method for treating cancer using chemokine antagonists
CN121039109A (zh) 2023-04-18 2025-11-28 国家科学研究中心 3,5-二氨基三唑衍生物及其用于治疗眼部疾病的用途

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