AU2006315436A1 - Azaindazoles useful as inhibitors of kinases - Google Patents
Azaindazoles useful as inhibitors of kinases Download PDFInfo
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- AU2006315436A1 AU2006315436A1 AU2006315436A AU2006315436A AU2006315436A1 AU 2006315436 A1 AU2006315436 A1 AU 2006315436A1 AU 2006315436 A AU2006315436 A AU 2006315436A AU 2006315436 A AU2006315436 A AU 2006315436A AU 2006315436 A1 AU2006315436 A1 AU 2006315436A1
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Classifications
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Hematology (AREA)
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- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US73710505P | 2005-11-15 | 2005-11-15 | |
| US60/737,105 | 2005-11-15 | ||
| PCT/US2006/044361 WO2007059219A1 (en) | 2005-11-15 | 2006-11-15 | Azaindazoles useful as inhibitors of kinases |
Publications (1)
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| AU2006315436A1 true AU2006315436A1 (en) | 2007-05-24 |
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| AU2006315436A Abandoned AU2006315436A1 (en) | 2005-11-15 | 2006-11-15 | Azaindazoles useful as inhibitors of kinases |
Country Status (7)
| Country | Link |
|---|---|
| US (2) | US8017781B2 (https=) |
| EP (2) | EP1948657A1 (https=) |
| JP (1) | JP2009515984A (https=) |
| CN (1) | CN101365700A (https=) |
| AU (1) | AU2006315436A1 (https=) |
| CA (1) | CA2628179A1 (https=) |
| WO (1) | WO2007059219A1 (https=) |
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| US7553639B2 (en) * | 2006-01-31 | 2009-06-30 | Elan Pharma International Limited | Alpha-synuclein kinase |
| CN101790532B (zh) * | 2007-07-31 | 2013-11-20 | 沃泰克斯药物股份有限公司 | 5-氟-1H-吡唑并[3，4-b]吡啶-3-胺及其衍生物的制备方法 |
| CA2696288A1 (en) | 2007-08-15 | 2009-02-19 | Schering Corporation | 6-substituted sulfonyl azabicyclo[3.2.1]octanes useful to inhibit 11.beta.-hydroxysteroid dehydrogenase type-1 |
| US8841304B2 (en) | 2008-01-08 | 2014-09-23 | Array Biopharma, Inc. | Pyrrolopyridines as kinase inhibitors |
| CN101965347B (zh) | 2008-01-09 | 2013-01-02 | 阵列生物制药公司 | 作为激酶抑制剂的吡唑并吡啶 |
| EP2247748A2 (en) * | 2008-02-13 | 2010-11-10 | Elan Pharma International Limited | Alpha-synuclein kinase |
| UA118010C2 (uk) | 2011-08-01 | 2018-11-12 | Вертекс Фармасьютікалз Інкорпорейтед | Інгібітори реплікації вірусів грипу |
| RS59144B1 (sr) | 2013-11-13 | 2019-09-30 | Vertex Pharma | Inhibitori replikacije virusa influence |
| HRP20181272T1 (hr) | 2013-11-13 | 2018-10-05 | Vertex Pharmaceuticals Incorporated | Postupci priprave inhibitora replikacije virusa influence |
| JP6704416B2 (ja) | 2015-05-13 | 2020-06-03 | バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ | インフルエンザウイルスの複製の阻害剤を調製する方法 |
| JP6857617B2 (ja) | 2015-05-13 | 2021-04-14 | バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ | インフルエンザウイルスの複製の阻害剤 |
| US10590077B2 (en) * | 2016-09-20 | 2020-03-17 | Glaxosmithkline Intellectual Property Development Limited | TRPV4 antagonists |
| CN116687951B (zh) * | 2023-06-06 | 2026-01-02 | 河北渤腾医药技术有限公司 | 一种plk1的干扰rna及其应用 |
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| US5420297A (en) * | 1990-10-24 | 1995-05-30 | Fujisawa Pharmaceutical Co., Ltd. | Peptides having substance P antagonistic activity |
| GB9113219D0 (en) | 1991-06-19 | 1991-08-07 | Fujisawa Pharmaceutical Co | Peptide compound,processes for preparation thereof and pharmaceutical composition comprising the same |
| US5654400A (en) * | 1991-10-04 | 1997-08-05 | Fujisawa Pharmaceutical Co., Ltd. | Process for making peptide compounds having tachykinin antagonistic activity |
| JP3485198B2 (ja) * | 1993-11-10 | 2004-01-13 | 富士写真フイルム株式会社 | ヒドラジン化合物及び該化合物を含むハロゲン化銀写真感光材料 |
| PL181323B1 (pl) | 1994-02-18 | 2001-07-31 | Boehringer Ingelheim Pharma | 2-heteroarylo-5,11-dihydro-6H-dipirydo[3,2-b:2’,3'-e][1,4] diazepinyi ich zastosowanie w zapobieganiu i leczeniu zakazen HIV PL PL PL |
| GB9412719D0 (en) | 1994-06-24 | 1994-08-17 | Erba Carlo Spa | Substituted azaindolylidene compounds and process for their preparation |
| JPH11501289A (ja) | 1994-12-02 | 1999-02-02 | 藤沢薬品工業株式会社 | Ｎｏ介在疾患の予防および／または治療のためのペプチド化合物 |
| US5837704A (en) * | 1995-02-17 | 1998-11-17 | Boehringer Ingelheim Pharmaceuticals, Inc. | 2-heteroaryl-5,11-dihydro-6H-dipyrido 3,2-B:2',3'-E! 1,4!diazepines and their use in the prevention or treatment of HIV infection |
| US5804585A (en) | 1996-04-15 | 1998-09-08 | Texas Biotechnology Corporation | Thieno-pyridine sulfonamides derivatives thereof and related compounds that modulate the activity of endothelin |
| US6537999B2 (en) * | 1996-06-06 | 2003-03-25 | Duquesne University Of The Holy Ghost | Pyrimidine derivatives and methods of making and using these derivatives |
| JP4028607B2 (ja) | 1996-07-24 | 2007-12-26 | 富山化学工業株式会社 | 新規なセファロスポリン誘導体またはその塩 |
| US6040321A (en) * | 1997-11-12 | 2000-03-21 | Bristol-Myers Squibb Company | Aminothiazole inhibitors of cyclin dependent kinases |
| US6025366A (en) * | 1998-04-02 | 2000-02-15 | Merck & Co., Inc. | Antagonists of gonadotropin releasing hormone |
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-
2006
- 2006-11-15 US US11/600,311 patent/US8017781B2/en not_active Expired - Fee Related
- 2006-11-15 AU AU2006315436A patent/AU2006315436A1/en not_active Abandoned
- 2006-11-15 WO PCT/US2006/044361 patent/WO2007059219A1/en not_active Ceased
- 2006-11-15 CA CA002628179A patent/CA2628179A1/en not_active Abandoned
- 2006-11-15 JP JP2008541312A patent/JP2009515984A/ja active Pending
- 2006-11-15 CN CNA2006800507344A patent/CN101365700A/zh active Pending
- 2006-11-15 EP EP06837683A patent/EP1948657A1/en not_active Withdrawn
- 2006-11-15 EP EP11191099A patent/EP2514751A1/en not_active Withdrawn
-
2011
- 2011-07-29 US US13/193,739 patent/US8445681B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US8017781B2 (en) | 2011-09-13 |
| EP2514751A1 (en) | 2012-10-24 |
| CA2628179A1 (en) | 2007-05-24 |
| EP1948657A1 (en) | 2008-07-30 |
| JP2009515984A (ja) | 2009-04-16 |
| US20070179177A1 (en) | 2007-08-02 |
| US8445681B2 (en) | 2013-05-21 |
| CN101365700A (zh) | 2009-02-11 |
| WO2007059219A1 (en) | 2007-05-24 |
| US20120165367A1 (en) | 2012-06-28 |
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