AU2005299851B2 - 2-(aryl)azacyclylmethyl carboxylates, sulfonates, phosphonates, phosphinates and heterocycles as S1P receptor agonists - Google Patents

2-(aryl)azacyclylmethyl carboxylates, sulfonates, phosphonates, phosphinates and heterocycles as S1P receptor agonists Download PDF

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AU2005299851B2
AU2005299851B2 AU2005299851A AU2005299851A AU2005299851B2 AU 2005299851 B2 AU2005299851 B2 AU 2005299851B2 AU 2005299851 A AU2005299851 A AU 2005299851A AU 2005299851 A AU2005299851 A AU 2005299851A AU 2005299851 B2 AU2005299851 B2 AU 2005299851B2
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disease
group
pct
phenyl
compound
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AU2005299851A1 (en
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Jeffrey John Hale
Lin Yan
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Merck Sharp and Dohme LLC
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Merck Sharp and Dohme Ltd
Merck Sharp and Dohme LLC
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

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  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Dermatology (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
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  • Pulmonology (AREA)
  • Rheumatology (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
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  • Endocrinology (AREA)
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  • Gastroenterology & Hepatology (AREA)
AU2005299851A 2004-10-22 2005-10-18 2-(aryl)azacyclylmethyl carboxylates, sulfonates, phosphonates, phosphinates and heterocycles as S1P receptor agonists Ceased AU2005299851B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US62131304P 2004-10-22 2004-10-22
US60/621,313 2004-10-22
PCT/US2005/037652 WO2006047195A2 (en) 2004-10-22 2005-10-18 2-(aryl)azacyclylmethyl carboxylates, sulfonates, phosphonates, phosphinates and heterocycles as s1p receptor agonists

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AU2005299851A1 AU2005299851A1 (en) 2006-05-04
AU2005299851B2 true AU2005299851B2 (en) 2011-03-17

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US (1) US7659294B2 (https=)
EP (1) EP1804793A4 (https=)
JP (1) JP2008517915A (https=)
CN (1) CN101043887A (https=)
AU (1) AU2005299851B2 (https=)
CA (1) CA2583681A1 (https=)
WO (1) WO2006047195A2 (https=)

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