AU2004287861B2 - Tetrazole derivatives and methods of treatment of metabolic-related disorders thereof - Google Patents

Tetrazole derivatives and methods of treatment of metabolic-related disorders thereof Download PDF

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Publication number
AU2004287861B2
AU2004287861B2 AU2004287861A AU2004287861A AU2004287861B2 AU 2004287861 B2 AU2004287861 B2 AU 2004287861B2 AU 2004287861 A AU2004287861 A AU 2004287861A AU 2004287861 A AU2004287861 A AU 2004287861A AU 2004287861 B2 AU2004287861 B2 AU 2004287861B2
Authority
AU
Australia
Prior art keywords
pharmaceutically acceptable
hydrate
solvate
acceptable salt
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU2004287861A
Other languages
English (en)
Other versions
AU2004287861A1 (en
Inventor
Steven L. Colletti
Tawfik Gharbaoui
Jason E. Imbriglio
Jae-Kyu Jung
Rui Liang
Subharekha Raghavan
Darby Schmidt
Thomas Schrader
Graeme Semple
Philip J. Skinner
James R. Tata
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Arena Pharmaceuticals Inc
Merck and Co Inc
Original Assignee
Arena Pharmaceuticals Inc
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arena Pharmaceuticals Inc, Merck and Co Inc filed Critical Arena Pharmaceuticals Inc
Publication of AU2004287861A1 publication Critical patent/AU2004287861A1/en
Application granted granted Critical
Publication of AU2004287861B2 publication Critical patent/AU2004287861B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/02Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU2004287861A 2003-10-31 2004-10-29 Tetrazole derivatives and methods of treatment of metabolic-related disorders thereof Ceased AU2004287861B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US51623803P 2003-10-31 2003-10-31
US60/516,238 2003-10-31
PCT/US2004/035927 WO2005044816A1 (en) 2003-10-31 2004-10-29 Tetrazole derivatives and methods of treatment of metabolic-related disorders thereof

Publications (2)

Publication Number Publication Date
AU2004287861A1 AU2004287861A1 (en) 2005-05-19
AU2004287861B2 true AU2004287861B2 (en) 2008-08-14

Family

ID=34572875

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2004287861A Ceased AU2004287861B2 (en) 2003-10-31 2004-10-29 Tetrazole derivatives and methods of treatment of metabolic-related disorders thereof

Country Status (37)

Country Link
US (2) US8637555B2 (cg-RX-API-DMAC7.html)
EP (2) EP1599469B1 (cg-RX-API-DMAC7.html)
JP (2) JP4533898B2 (cg-RX-API-DMAC7.html)
KR (1) KR100850591B1 (cg-RX-API-DMAC7.html)
CN (1) CN1867562B (cg-RX-API-DMAC7.html)
AR (1) AR046611A1 (cg-RX-API-DMAC7.html)
AT (1) ATE328880T1 (cg-RX-API-DMAC7.html)
AU (1) AU2004287861B2 (cg-RX-API-DMAC7.html)
BR (1) BRPI0415631A (cg-RX-API-DMAC7.html)
CA (1) CA2539985C (cg-RX-API-DMAC7.html)
CO (1) CO5690551A2 (cg-RX-API-DMAC7.html)
CR (1) CR8270A (cg-RX-API-DMAC7.html)
CY (1) CY1105479T1 (cg-RX-API-DMAC7.html)
DE (1) DE602004001134T2 (cg-RX-API-DMAC7.html)
DK (1) DK1599469T3 (cg-RX-API-DMAC7.html)
EA (1) EA011484B1 (cg-RX-API-DMAC7.html)
EC (1) ECSP066529A (cg-RX-API-DMAC7.html)
ES (1) ES2267077T3 (cg-RX-API-DMAC7.html)
GE (1) GEP20094801B (cg-RX-API-DMAC7.html)
HR (1) HRP20060286T3 (cg-RX-API-DMAC7.html)
IL (1) IL174042A0 (cg-RX-API-DMAC7.html)
IS (1) IS2372B (cg-RX-API-DMAC7.html)
MA (1) MA28171A1 (cg-RX-API-DMAC7.html)
MX (1) MXPA06004556A (cg-RX-API-DMAC7.html)
MY (1) MY140410A (cg-RX-API-DMAC7.html)
NO (1) NO20062509L (cg-RX-API-DMAC7.html)
NZ (1) NZ546285A (cg-RX-API-DMAC7.html)
PE (1) PE20050483A1 (cg-RX-API-DMAC7.html)
PL (1) PL1599469T3 (cg-RX-API-DMAC7.html)
PT (1) PT1599469E (cg-RX-API-DMAC7.html)
RS (1) RS20060290A (cg-RX-API-DMAC7.html)
SI (1) SI1599469T1 (cg-RX-API-DMAC7.html)
TN (1) TNSN06150A1 (cg-RX-API-DMAC7.html)
TW (1) TWI258478B (cg-RX-API-DMAC7.html)
UA (1) UA86783C2 (cg-RX-API-DMAC7.html)
WO (1) WO2005044816A1 (cg-RX-API-DMAC7.html)
ZA (2) ZA200603419B (cg-RX-API-DMAC7.html)

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ES2331521T3 (es) * 2003-11-21 2010-01-07 Arena Pharmaceuticals, Inc. Derivados de acido 4-oxo-4,5-dihidro-furan-2-carboxilico y procedimientos de tratamiento de trastornos metabolicos relacionados del mismo.
WO2006026273A2 (en) * 2004-08-25 2006-03-09 Merck & Co., Inc. Method of treating atherosclerosis, dyslipidemias and related conditions
EP1811996A1 (en) * 2004-11-05 2007-08-01 Arena Pharmaceuticals, Inc. Compositions for treating flushing and lipid-associated disorders comprising niacin receptor partial agonists
PE20060949A1 (es) * 2004-12-23 2006-10-11 Arena Pharm Inc Derivados fusionados de pirazol como agonistas del receptor de niacina
US8168799B2 (en) 2005-04-28 2012-05-01 Merck Sharpe & Dohme Ltd. Process for the preparation of tetrazolytetrahydrocyclopentapyrazoles
AU2006261839B2 (en) 2005-06-28 2011-09-01 Merck Sharp & Dohme Corp. Niacin receptor agonists, compositions containing such compounds and methods of treatment
DE102006021733A1 (de) * 2006-05-09 2007-11-22 Bayer Healthcare Ag 3-Tetrazolylindazole und 3-Tetrazolylpyrazolopyridine sowie ihre Verwendung
DE102006043443A1 (de) 2006-09-15 2008-03-27 Bayer Healthcare Ag Neue aza-bicyclische Verbindungen und ihre Verwendung
DE102008063992A1 (de) 2008-12-19 2010-09-02 Lerner, Zinoviy, Dipl.-Ing. Neue aliphatisch substituierte Pyrazolopyridine und ihre Verwendung
DE102010021637A1 (de) 2010-05-26 2011-12-01 Bayer Schering Pharma Aktiengesellschaft Substituierte 5-Fluor-1H-Pyrazolopyridine und ihre Verwendung
JP2015522080A (ja) 2012-07-11 2015-08-03 エルセリクス セラピューティクス インコーポレイテッド スタチン、ビグアナイド、およびさらなる薬剤を含む心血管代謝性リスクを減少させるための組成物
EA201500852A1 (ru) 2013-02-21 2016-02-29 Адверио Фарма Гмбх Формы метил {4,6-диамино-2-[1-(2-фторбензил)-1н-пиразоло[3,4-в]пиридино-3-ил]пиримидино-5-ил}метил карбамата
WO2015012210A1 (ja) * 2013-07-23 2015-01-29 エーザイ・アール・アンド・ディー・マネジメント株式会社 ヘテロ縮合環化合物
CN103755637A (zh) * 2013-12-26 2014-04-30 平湖优康药物研发有限公司 一种医药中间体1,4,5,6-四氢-3-环戊并吡唑甲腈的合成工艺
US12086719B2 (en) * 2019-10-11 2024-09-10 Royal Bank Of Canada System and method of machine learning using embedding networks

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US8168799B2 (en) 2005-04-28 2012-05-01 Merck Sharpe & Dohme Ltd. Process for the preparation of tetrazolytetrahydrocyclopentapyrazoles

Also Published As

Publication number Publication date
EP1599469B1 (en) 2006-06-07
AR046611A1 (es) 2005-12-14
ECSP066529A (es) 2006-10-10
IS2372B (is) 2008-06-15
TW200530221A (en) 2005-09-16
DE602004001134D1 (de) 2006-07-20
AU2004287861A1 (en) 2005-05-19
MXPA06004556A (es) 2006-07-06
UA86783C2 (ru) 2009-05-25
PT1599469E (pt) 2006-10-31
JP2007509181A (ja) 2007-04-12
EA011484B1 (ru) 2009-04-28
MY140410A (en) 2009-12-31
EA200600879A1 (ru) 2006-10-27
JP4533898B2 (ja) 2010-09-01
NO20062509L (no) 2006-06-26
CN1867562B (zh) 2011-07-13
HRP20060286T3 (en) 2007-03-31
EP1683794A1 (en) 2006-07-26
DE602004001134T2 (de) 2007-04-19
EP1599469A1 (en) 2005-11-30
TNSN06150A1 (en) 2007-11-15
TWI258478B (en) 2006-07-21
GEP20094801B (en) 2009-10-26
KR100850591B1 (ko) 2008-08-05
PE20050483A1 (es) 2005-08-25
BRPI0415631A (pt) 2006-12-12
CN1867562A (zh) 2006-11-22
CY1105479T1 (el) 2010-07-28
CR8270A (es) 2006-10-06
IS8481A (is) 2006-05-24
CO5690551A2 (es) 2006-10-31
NZ546285A (en) 2010-04-30
US8637555B2 (en) 2014-01-28
ZA200603419B (en) 2006-10-25
US20060217562A1 (en) 2006-09-28
IL174042A0 (en) 2006-08-01
DK1599469T3 (da) 2006-10-09
MA28171A1 (fr) 2006-09-01
SI1599469T1 (sl) 2006-10-31
ZA200606203B (en) 2007-04-25
PL1599469T3 (pl) 2006-10-31
ATE328880T1 (de) 2006-06-15
ES2267077T3 (es) 2007-03-01
CA2539985A1 (en) 2005-05-19
CA2539985C (en) 2010-02-16
US20070072924A1 (en) 2007-03-29
WO2005044816A1 (en) 2005-05-19
HK1076468A1 (en) 2006-01-20
KR20060073974A (ko) 2006-06-29
RS20060290A (sr) 2008-11-28
JP2010163448A (ja) 2010-07-29

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