AU2003220180A1 - Crystalline parecoxib sodium - Google Patents
Crystalline parecoxib sodium Download PDFInfo
- Publication number
- AU2003220180A1 AU2003220180A1 AU2003220180A AU2003220180A AU2003220180A1 AU 2003220180 A1 AU2003220180 A1 AU 2003220180A1 AU 2003220180 A AU2003220180 A AU 2003220180A AU 2003220180 A AU2003220180 A AU 2003220180A AU 2003220180 A1 AU2003220180 A1 AU 2003220180A1
- Authority
- AU
- Australia
- Prior art keywords
- parecoxib sodium
- sodium
- drug substance
- parecoxib
- accordance
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
- C07D457/04—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 8
- C07D457/06—Lysergic acid amides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/08—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US36456702P | 2002-03-15 | 2002-03-15 | |
| US60/364,567 | 2002-03-15 | ||
| US41798702P | 2002-10-11 | 2002-10-11 | |
| US60/417,987 | 2002-10-11 | ||
| PCT/US2003/007484 WO2003078408A1 (en) | 2002-03-15 | 2003-03-12 | Crystalline parecoxib sodium |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2003220180A1 true AU2003220180A1 (en) | 2003-09-29 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2003220180A Abandoned AU2003220180A1 (en) | 2002-03-15 | 2003-03-12 | Crystalline parecoxib sodium |
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|---|---|
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| EP (1) | EP1485362A1 (enExample) |
| JP (1) | JP2005529084A (enExample) |
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| CN (1) | CN1642926A (enExample) |
| AR (1) | AR038985A1 (enExample) |
| AU (1) | AU2003220180A1 (enExample) |
| BR (1) | BR0308431A (enExample) |
| CA (1) | CA2478500A1 (enExample) |
| CO (1) | CO5631437A2 (enExample) |
| IL (1) | IL163780A0 (enExample) |
| MX (1) | MXPA04008932A (enExample) |
| MY (1) | MY148518A (enExample) |
| NZ (1) | NZ535951A (enExample) |
| PL (1) | PL372880A1 (enExample) |
| RU (1) | RU2300529C2 (enExample) |
| TW (1) | TW200400949A (enExample) |
| WO (1) | WO2003078408A1 (enExample) |
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| US20050143431A1 (en) * | 2003-04-04 | 2005-06-30 | Hetero Drugs Limited | Novel crystalline forms of parecoxib sodium |
| JP2007507538A (ja) | 2003-10-02 | 2007-03-29 | エラン ファーマシューティカルズ，インコーポレイテッド | 疼痛軽減方法 |
| JP2007517013A (ja) * | 2003-12-24 | 2007-06-28 | ファルマシア コーポレーション | 炎症、疼痛および／または発熱の治療を目的としたｃｏｘ−２阻害薬バルデコキシブのプロドラッグとしてのパレコキシブ金属塩 |
| ITMI20040019A1 (it) * | 2004-01-12 | 2004-04-12 | Univ Bari | Derivati isossazolici e loro impiego come inibitori della ciclossigenasi |
| US7796785B2 (en) * | 2005-03-03 | 2010-09-14 | Fujifilm Corporation | Image extracting apparatus, image extracting method, and image extracting program |
| US20080108664A1 (en) * | 2005-12-23 | 2008-05-08 | Liu Belle B | Solid-state form of AMG 706 and pharmaceutical compositions thereof |
| US7989450B2 (en) | 2008-01-11 | 2011-08-02 | Universita' Degli Studi Di Bari | Functionalized diarylisoxazoles inhibitors of ciclooxygenase |
| GB0919757D0 (en) * | 2009-11-12 | 2009-12-30 | Johnson Matthey Plc | Polymorphs of bromfenac sodium and methods for preparing bromfenac sodium polymorphs |
| US8299295B2 (en) | 2009-10-15 | 2012-10-30 | Johnson Matthey Public Limited Company | Polymorphs of bromfenac sodium and methods for preparing bromfenac sodium polymorphs |
| CN105726496B (zh) * | 2014-12-12 | 2019-05-28 | 湖南科伦药物研究有限公司 | 一种帕瑞昔布钠冻干粉剂、其制备方法及其粉剂产品 |
| CN105125506A (zh) * | 2015-08-18 | 2015-12-09 | 上海秀新臣邦医药科技有限公司 | 一种注射用帕瑞昔布钠及其制备方法 |
| CN106580893A (zh) * | 2016-12-26 | 2017-04-26 | 上药东英（江苏）药业有限公司 | 一种帕瑞昔布钠冻干粉针制剂 |
| CN106692079A (zh) * | 2016-12-26 | 2017-05-24 | 上药东英（江苏）药业有限公司 | 一种帕瑞昔布钠长效冻干粉针制剂 |
| CN117003769B (zh) * | 2023-07-11 | 2024-11-22 | 中国科学院宁波材料技术与工程研究所 | 氯诺昔康复合物、氯诺昔康-小檗碱共晶及其制备方法和应用 |
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| EP1288206B1 (en) * | 1996-04-12 | 2008-09-17 | G.D. Searle LLC | Substituted benzenesulfonamide derivatives as prodrugs of COX-2 inhibitors |
| CN100558356C (zh) * | 1996-10-15 | 2009-11-11 | G.D.瑟尔公司 | 应用环加氧酶-2抑制剂治疗和预防肿瘤形成的方法 |
| PE20021017A1 (es) * | 2001-04-03 | 2002-11-24 | Pharmacia Corp | Composicion parenteral reconstituible |
| IL161086A0 (en) * | 2001-10-02 | 2004-08-31 | Pharmacia Corp | Method for preparing benzenesulfonyl compounds |
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- 2003-03-12 EP EP03716476A patent/EP1485362A1/en not_active Withdrawn
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2004
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Also Published As
| Publication number | Publication date |
|---|---|
| PL372880A1 (en) | 2005-08-08 |
| JP2005529084A (ja) | 2005-09-29 |
| RU2300529C2 (ru) | 2007-06-10 |
| EP1485362A1 (en) | 2004-12-15 |
| KR100763045B1 (ko) | 2007-10-04 |
| CA2478500A1 (en) | 2003-09-25 |
| KR20040095288A (ko) | 2004-11-12 |
| CO5631437A2 (es) | 2006-04-28 |
| RU2004127585A (ru) | 2005-04-10 |
| MXPA04008932A (es) | 2004-11-26 |
| US20030232871A1 (en) | 2003-12-18 |
| AR038985A1 (es) | 2005-02-02 |
| NZ535951A (en) | 2006-02-24 |
| CN1642926A (zh) | 2005-07-20 |
| IL163780A0 (en) | 2005-12-18 |
| WO2003078408A1 (en) | 2003-09-25 |
| MY148518A (en) | 2013-04-30 |
| BR0308431A (pt) | 2005-01-18 |
| TW200400949A (en) | 2004-01-16 |
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