AU2002305143A1 - Pyrazolo'1,5-a!pyridine derivatives - Google Patents

Pyrazolo'1,5-a!pyridine derivatives

Info

Publication number
AU2002305143A1
AU2002305143A1 AU2002305143A AU2002305143A AU2002305143A1 AU 2002305143 A1 AU2002305143 A1 AU 2002305143A1 AU 2002305143 A AU2002305143 A AU 2002305143A AU 2002305143 A AU2002305143 A AU 2002305143A AU 2002305143 A1 AU2002305143 A1 AU 2002305143A1
Authority
AU
Australia
Prior art keywords
pyrazolo
pyridine derivatives
same
variables
preparing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2002305143A
Other languages
English (en)
Inventor
Kristjan Gudmundsson
Brian A. Johns
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Corp
Original Assignee
SmithKline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Corp filed Critical SmithKline Beecham Corp
Publication of AU2002305143A1 publication Critical patent/AU2002305143A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biotechnology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
AU2002305143A 2001-04-27 2002-04-05 Pyrazolo'1,5-a!pyridine derivatives Abandoned AU2002305143A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US28694801P 2001-04-27 2001-04-27
US60/286,948 2001-04-27
PCT/US2002/010687 WO2002088124A2 (en) 2001-04-27 2002-04-05 Pyrazolo'1,5-a!pyridine derivatives

Publications (1)

Publication Number Publication Date
AU2002305143A1 true AU2002305143A1 (en) 2002-11-11

Family

ID=23100830

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2002305143A Abandoned AU2002305143A1 (en) 2001-04-27 2002-04-05 Pyrazolo'1,5-a!pyridine derivatives

Country Status (8)

Country Link
US (3) US6962914B2 (enExample)
EP (1) EP1385847B1 (enExample)
JP (1) JP2004527560A (enExample)
AT (1) ATE296826T1 (enExample)
AU (1) AU2002305143A1 (enExample)
DE (1) DE60204452T2 (enExample)
ES (1) ES2242028T3 (enExample)
WO (1) WO2002088124A2 (enExample)

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US9126948B2 (en) 2011-03-25 2015-09-08 Incyte Holdings Corporation Pyrimidine-4,6-diamine derivatives as PI3K inhibitors
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ES2928164T3 (es) 2015-10-19 2022-11-15 Incyte Corp Compuestos heterocíclicos como inmunomoduladores
HUE060680T2 (hu) 2015-11-19 2023-04-28 Incyte Corp Heterociklusos vegyületek mint immunmodulátorok
DK3394033T3 (da) 2015-12-22 2021-01-04 Incyte Corp Heterocykliske forbindelser som immunmodulatorer
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ES2930092T3 (es) 2016-07-14 2022-12-07 Incyte Corp Compuestos heterocíclicos como inmunomoduladores
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CA3047991A1 (en) 2016-12-22 2018-06-28 Incyte Corporation Bicyclic heteroaromatic compounds as immunomodulators
EP3558989B1 (en) 2016-12-22 2021-04-14 Incyte Corporation Triazolo[1,5-a]pyridine derivatives as immunomodulators
MA47123A (fr) 2016-12-22 2021-03-17 Incyte Corp Dérivés de benzooxazole en tant qu'mmunomodulateurs
US20180179179A1 (en) 2016-12-22 2018-06-28 Incyte Corporation Heterocyclic compounds as immunomodulators
MD3558990T2 (ro) 2016-12-22 2023-02-28 Incyte Corp Derivați tetrahidro imidazo[4,5-c]piridină ca inductori de internalizare a PD-L1
US10669271B2 (en) 2018-03-30 2020-06-02 Incyte Corporation Heterocyclic compounds as immunomodulators
LT3790877T (lt) 2018-05-11 2023-05-10 Incyte Corporation Tetrahidro-imidazo[4,5-c]piridino dariniai kaip pd-l1 imunomoduliatoriai
BR112020024427A2 (pt) 2018-06-01 2021-03-23 Incyte Corporation regime de dosagem para o tratamento de distúrbios relacionados a pi3k
TW202115059A (zh) 2019-08-09 2021-04-16 美商英塞特公司 Ｐｄ—１／ｐｄ—ｌ１抑制劑之鹽
EP4037773A1 (en) 2019-09-30 2022-08-10 Incyte Corporation Pyrido[3,2-d]pyrimidine compounds as immunomodulators
PE20230407A1 (es) 2019-11-11 2023-03-07 Incyte Corp Sales y formas cristalinas de un inhibidor de pd-1/pd-l1
US11780836B2 (en) 2020-11-06 2023-10-10 Incyte Corporation Process of preparing a PD-1/PD-L1 inhibitor
WO2022099075A1 (en) 2020-11-06 2022-05-12 Incyte Corporation Crystalline form of a pd-1/pd-l1 inhibitor
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Also Published As

Publication number Publication date
DE60204452D1 (de) 2005-07-07
US7030134B2 (en) 2006-04-18
US20040142941A1 (en) 2004-07-22
US6962914B2 (en) 2005-11-08
WO2002088124A3 (en) 2003-05-08
EP1385847A2 (en) 2004-02-04
ATE296826T1 (de) 2005-06-15
EP1385847B1 (en) 2005-06-01
ES2242028T3 (es) 2005-11-01
DE60204452T2 (de) 2005-12-15
WO2002088124A2 (en) 2002-11-07
JP2004527560A (ja) 2004-09-09
US20050192295A1 (en) 2005-09-01
US20050192303A1 (en) 2005-09-01

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase