AU2001238575B2 - Tyrosine kinase inhibitors - Google Patents

Tyrosine kinase inhibitors Download PDF

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Publication number
AU2001238575B2
AU2001238575B2 AU2001238575A AU2001238575A AU2001238575B2 AU 2001238575 B2 AU2001238575 B2 AU 2001238575B2 AU 2001238575 A AU2001238575 A AU 2001238575A AU 2001238575 A AU2001238575 A AU 2001238575A AU 2001238575 B2 AU2001238575 B2 AU 2001238575B2
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AU
Australia
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optionally substituted
substituents selected
alkyl
compound
mammal
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Ceased
Application number
AU2001238575A
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English (en)
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AU2001238575A1 (en
Inventor
Mark E. Fraley
George D. Hartman
Randall W. Hungate
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Merck and Co Inc
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Merck and Co Inc
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Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of AU2001238575A1 publication Critical patent/AU2001238575A1/en
Application granted granted Critical
Publication of AU2001238575B2 publication Critical patent/AU2001238575B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AU2001238575A 2000-02-25 2001-02-21 Tyrosine kinase inhibitors Ceased AU2001238575B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18502300P 2000-02-25 2000-02-25
US60/185,023 2000-02-25
PCT/US2001/005482 WO2001062251A1 (en) 2000-02-25 2001-02-21 Tyrosine kinase inhibitors

Publications (2)

Publication Number Publication Date
AU2001238575A1 AU2001238575A1 (en) 2001-11-15
AU2001238575B2 true AU2001238575B2 (en) 2005-04-07

Family

ID=22679236

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2001238575A Ceased AU2001238575B2 (en) 2000-02-25 2001-02-21 Tyrosine kinase inhibitors
AU3857501A Pending AU3857501A (en) 2000-02-25 2001-02-21 Tyrosine kinase inhibitors

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU3857501A Pending AU3857501A (en) 2000-02-25 2001-02-21 Tyrosine kinase inhibitors

Country Status (9)

Country Link
US (1) US6420382B2 (enExample)
EP (1) EP1259235B1 (enExample)
JP (1) JP2003523389A (enExample)
AT (1) ATE368457T1 (enExample)
AU (2) AU2001238575B2 (enExample)
CA (1) CA2400875A1 (enExample)
DE (1) DE60129672T2 (enExample)
ES (1) ES2288928T3 (enExample)
WO (1) WO2001062251A1 (enExample)

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DE60212627T2 (de) * 2001-06-29 2007-06-14 Ab Science Verwendung von Tyrosinkinase-Inhibitoren zur Behandlung von entzündlichen Krankheiten
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Also Published As

Publication number Publication date
EP1259235A1 (en) 2002-11-27
JP2003523389A (ja) 2003-08-05
EP1259235B1 (en) 2007-08-01
ATE368457T1 (de) 2007-08-15
ES2288928T3 (es) 2008-02-01
DE60129672D1 (de) 2007-09-13
EP1259235A4 (en) 2004-11-03
DE60129672T2 (de) 2008-04-30
CA2400875A1 (en) 2001-08-30
US6420382B2 (en) 2002-07-16
WO2001062251A1 (en) 2001-08-30
AU3857501A (en) 2001-09-03
US20010044451A1 (en) 2001-11-22

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