ATE53585T1 - Penemverbindungen, ihre herstellung und verwendung. - Google Patents

Penemverbindungen, ihre herstellung und verwendung.

Info

Publication number
ATE53585T1
ATE53585T1 AT86301642T AT86301642T ATE53585T1 AT E53585 T1 ATE53585 T1 AT E53585T1 AT 86301642 T AT86301642 T AT 86301642T AT 86301642 T AT86301642 T AT 86301642T AT E53585 T1 ATE53585 T1 AT E53585T1
Authority
AT
Austria
Prior art keywords
denotes
production
penem compounds
gram
methylene
Prior art date
Application number
AT86301642T
Other languages
English (en)
Inventor
Masaji Ishiguro
Hiromitsu Iwata
Takashi Nakatsuka
Shimamoto-Cho
Original Assignee
Suntory Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Suntory Ltd filed Critical Suntory Ltd
Application granted granted Critical
Publication of ATE53585T1 publication Critical patent/ATE53585T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Ink Jet (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Ultra Sonic Daignosis Equipment (AREA)
  • Pens And Brushes (AREA)
  • Coupling Device And Connection With Printed Circuit (AREA)
AT86301642T 1985-03-09 1986-03-07 Penemverbindungen, ihre herstellung und verwendung. ATE53585T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP60047103A JPH075463B2 (ja) 1985-03-09 1985-03-09 抗菌剤
EP86301642A EP0199446B1 (de) 1985-03-09 1986-03-07 Penemverbindungen, ihre Herstellung und Verwendung

Publications (1)

Publication Number Publication Date
ATE53585T1 true ATE53585T1 (de) 1990-06-15

Family

ID=12765840

Family Applications (1)

Application Number Title Priority Date Filing Date
AT86301642T ATE53585T1 (de) 1985-03-09 1986-03-07 Penemverbindungen, ihre herstellung und verwendung.

Country Status (8)

Country Link
US (1) US4997829A (de)
EP (1) EP0199446B1 (de)
JP (1) JPH075463B2 (de)
AT (1) ATE53585T1 (de)
AU (1) AU585948B2 (de)
CA (1) CA1299565C (de)
DE (1) DE3671894D1 (de)
MX (1) MX9203548A (de)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2526046B2 (ja) * 1986-12-26 1996-08-21 サントリー株式会社 ペネム誘導体、その製造法およびその用途
GB8713515D0 (en) * 1987-06-10 1987-07-15 Erba Farmitalia Methoxymethyl compounds
US5191075A (en) * 1988-10-19 1993-03-02 Pfizer Inc Process for the preparation of penems
US4992543A (en) * 1988-10-19 1991-02-12 Pfizer Inc. Penem derivatives
US5416208A (en) * 1989-07-05 1995-05-16 Farmitalia Carlo Erba S R L Process for penems
GB8915392D0 (en) * 1989-07-05 1989-08-23 Erba Carlo Spa Process for penems
ATE242251T1 (de) * 1990-08-20 2003-06-15 Daiichi Suntory Pharma Co Ltd Antibakterielle penem-ester-derivate
ATE186537T1 (de) * 1990-08-20 1999-11-15 Suntory Ltd Antibakterielle penem-ester derivate
DE69130363T2 (de) * 1990-08-20 1999-04-22 Suntory Limited, Osaka Antibakterielle penemverbindungen
DE69233529T2 (de) * 1991-02-01 2005-11-24 Daiichi Suntory Pharma Co., Ltd. Orale antibakterielle Zusammensetzungen und Verfahren zur Verbesserung der Resorption von Penem-oder Carbapenem-Antibiotika im Magen-Darm-Trakt
US5602118A (en) * 1993-03-16 1997-02-11 American Cyanamid Company 2-thiosubstituted carbapenems
JPH09202789A (ja) 1995-11-20 1997-08-05 Suntory Ltd ペネム誘導体およびこれを含有する抗菌剤
JPH1059970A (ja) * 1996-08-16 1998-03-03 Suntory Ltd カルバペネム誘導体およびこれを含有する抗菌剤
KR20000076105A (ko) 1998-01-13 2000-12-26 도리이 신이찌로 항생제를 함유한 국소 투여용 항균 조성물
JP2005239696A (ja) 2004-01-30 2005-09-08 Daiichi Suntory Pharma Co Ltd 無機物質を配合した医薬硬質カプセル剤
EP1934230A1 (de) * 2005-10-05 2008-06-25 Ranbaxy Laboratories, Ltd. Verfahren zur herstellung von faropenem
WO2008012830A1 (en) * 2006-07-28 2008-01-31 Hetero Drugs Limited Soup faropenem free acid
WO2008035153A2 (en) * 2006-08-02 2008-03-27 Orchid Chemicals & Pharmaceuticals Limited Process for the preparation of beta-lactam antibiotic
CN101941981B (zh) * 2009-07-03 2015-01-21 湖南华纳大药厂有限公司 催化剂组合物以及用于制备法罗培南钠的方法
CN102964357A (zh) * 2012-11-11 2013-03-13 苏州二叶制药有限公司 法罗培南钠及其片剂

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
EP0003960B1 (de) * 1978-02-02 1983-06-29 Ciba-Geigy Ag 6-Substituierte Thia-Azaverbindungen, ihre Herstellung und diese enthaltende pharmazeutische Präparate
JPS5625110A (en) * 1978-12-18 1981-03-10 Bristol Myers Co Antibacterial
US4272437A (en) * 1978-12-18 1981-06-09 Bristol-Myers Company Antibacterial agents, and 4-thio azetidinone intermediates
US4619783A (en) * 1983-06-10 1986-10-28 Pfizer Inc. Process and intermediates for the preparation of penem derivatives
US4614737A (en) * 1983-10-14 1986-09-30 Pfizer Inc. 2-dioxacycloalkylthiopenem derivatives

Also Published As

Publication number Publication date
CA1299565C (en) 1992-04-28
DE3671894D1 (de) 1990-07-19
EP0199446A1 (de) 1986-10-29
AU585948B2 (en) 1989-06-29
MX9203548A (es) 1992-09-01
US4997829A (en) 1991-03-05
JPH075463B2 (ja) 1995-01-25
EP0199446B1 (de) 1990-06-13
JPS61207387A (ja) 1986-09-13
AU5446086A (en) 1986-09-11

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Legal Events

Date Code Title Description
EEIH Change in the person of patent owner
EELA Cancelled due to lapse of time