ATE534381T1 - Pharmazeutische cetp-inhibitor-zusammensetzungen - Google Patents

Pharmazeutische cetp-inhibitor-zusammensetzungen

Info

Publication number
ATE534381T1
ATE534381T1 AT04721345T AT04721345T ATE534381T1 AT E534381 T1 ATE534381 T1 AT E534381T1 AT 04721345 T AT04721345 T AT 04721345T AT 04721345 T AT04721345 T AT 04721345T AT E534381 T1 ATE534381 T1 AT E534381T1
Authority
AT
Austria
Prior art keywords
cetp inhibitor
pharmaceutical
inhibitor compositions
pharmaceutical compositions
inhibitor
Prior art date
Application number
AT04721345T
Other languages
German (de)
English (en)
Inventor
Yoshifumi Uemoto
Original Assignee
Japan Tobacco Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33033290&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE534381(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Japan Tobacco Inc filed Critical Japan Tobacco Inc
Application granted granted Critical
Publication of ATE534381T1 publication Critical patent/ATE534381T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/70—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/82—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/095—Sulfur, selenium, or tellurium compounds, e.g. thiols
    • A61K31/10—Sulfides; Sulfoxides; Sulfones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/265—Esters, e.g. nitroglycerine, selenocyanates of carbonic, thiocarbonic, or thiocarboxylic acids, e.g. thioacetic acid, xanthogenic acid, trithiocarbonic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
AT04721345T 2003-03-17 2004-03-17 Pharmazeutische cetp-inhibitor-zusammensetzungen ATE534381T1 (de)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US45529303P 2003-03-17 2003-03-17
US46052103P 2003-04-04 2003-04-04
US47720203P 2003-06-10 2003-06-10
US49364903P 2003-08-08 2003-08-08
PCT/JP2004/003585 WO2004082593A2 (en) 2003-03-17 2004-03-17 Pharmaceutical compositions of cetp inhibitors

Publications (1)

Publication Number Publication Date
ATE534381T1 true ATE534381T1 (de) 2011-12-15

Family

ID=33033290

Family Applications (1)

Application Number Title Priority Date Filing Date
AT04721345T ATE534381T1 (de) 2003-03-17 2004-03-17 Pharmazeutische cetp-inhibitor-zusammensetzungen

Country Status (20)

Country Link
US (2) US20040225018A1 (enExample)
EP (2) EP2289507A1 (enExample)
JP (2) JP5546715B2 (enExample)
KR (2) KR20080008440A (enExample)
AT (1) ATE534381T1 (enExample)
AU (1) AU2004222434B2 (enExample)
BR (1) BRPI0408466B8 (enExample)
CA (1) CA2519432C (enExample)
CO (1) CO5640101A2 (enExample)
CY (1) CY1112324T1 (enExample)
DK (1) DK1603553T3 (enExample)
ES (1) ES2377121T3 (enExample)
IL (1) IL170749A (enExample)
MX (1) MXPA05009848A (enExample)
NO (1) NO336891B1 (enExample)
NZ (1) NZ542852A (enExample)
PL (1) PL1603553T3 (enExample)
PT (1) PT1603553E (enExample)
SI (1) SI1603553T1 (enExample)
WO (1) WO2004082593A2 (enExample)

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US7393652B2 (en) 2000-05-10 2008-07-01 The Trustees Of Columbia University In The City Of New York Methods for identifying a chemical compound that directly enhances binding of FKBP12.6 to PKA-phosphorylated type 2 ryanodine receptor (RyR2)
US7718644B2 (en) 2004-01-22 2010-05-18 The Trustees Of Columbia University In The City Of New York Anti-arrhythmic and heart failure drugs that target the leak in the ryanodine receptor (RyR2) and uses thereof
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US7544678B2 (en) 2002-11-05 2009-06-09 The Trustees Of Columbia University In The City Of New York Anti-arrythmic and heart failure drugs that target the leak in the ryanodine receptor (RyR2)
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KR20070087197A (ko) * 2003-09-26 2007-08-27 니뽄 다바코 산교 가부시키가이샤 잔여 리포프로테인 생산 저해 방법
US8710045B2 (en) 2004-01-22 2014-04-29 The Trustees Of Columbia University In The City Of New York Agents for preventing and treating disorders involving modulation of the ryanodine receptors
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US7704990B2 (en) 2005-08-25 2010-04-27 The Trustees Of Columbia University In The City Of New York Agents for preventing and treating disorders involving modulation of the RyR receptors
CN101378731B (zh) 2006-02-09 2014-03-05 默沙东公司 Cetp抑制剂的聚合物制剂
WO2010066593A1 (en) * 2008-12-08 2010-06-17 F. Hoffmann-La Roche Ag Combined drug administration
CN102293734A (zh) * 2010-06-25 2011-12-28 江苏恒瑞医药股份有限公司 托伐普坦固体分散体及其制备方法
MY164729A (en) * 2010-11-04 2018-01-30 Hoffmann La Roche A composition comprising s-[2- ( [ [1- (2-ethylbutyl) - cyclohexyl] - carbonyl]amino)phenyl] 2-methylpropanethioate and croscarmellose sodium
BR112013014291A2 (pt) * 2010-12-08 2016-09-20 Hoffmann La Roche formulação lipossômica de calcetrapib
CN103391769A (zh) * 2011-02-17 2013-11-13 霍夫曼-拉罗奇有限公司 通过热熔挤出使活性药物成分从过冷液体状态受控结晶的方法
BR112016013923A2 (pt) * 2013-12-19 2017-08-08 Hoffmann La Roche Modulador de cetp para o uso no tratamento de enfermidade ocular
JP2021534236A (ja) * 2018-08-09 2021-12-09 ダルコア ファーマ ユーケー リミテッド，レザーヘッド，ツーク ブランチ 新規発症２型糖尿病の発生遅延並びに２型糖尿病の進行緩徐化及び治療の方法
WO2023064794A1 (en) * 2021-10-12 2023-04-20 Hdl Therapeutics, Inc. Methods and systems for prophylactically preventing, slowing the progression of, or treating cerebral amyloid angiopathy, alzheimer's disease and/or acute stroke

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Also Published As

Publication number Publication date
CY1112324T1 (el) 2015-12-09
KR20080008440A (ko) 2008-01-23
WO2004082593A2 (en) 2004-09-30
CO5640101A2 (es) 2006-05-31
AU2004222434B2 (en) 2010-06-03
KR20050110019A (ko) 2005-11-22
IL170749A0 (en) 2009-02-11
EP1603553A2 (en) 2005-12-14
BRPI0408466B1 (pt) 2018-11-21
US20140243414A1 (en) 2014-08-28
EP1603553B1 (en) 2011-11-23
JP2006520808A (ja) 2006-09-14
NZ542852A (en) 2008-09-26
ES2377121T9 (es) 2012-08-21
ES2377121T3 (es) 2012-03-22
BRPI0408466A (pt) 2006-04-04
KR100857759B1 (ko) 2008-09-09
BRPI0408466B8 (pt) 2021-05-25
JP5546715B2 (ja) 2014-07-09
NO336891B1 (no) 2015-11-23
NO20054740D0 (no) 2005-10-14
PL1603553T3 (pl) 2012-04-30
SI1603553T1 (sl) 2012-03-30
NO20054740L (no) 2005-12-13
JP2011052006A (ja) 2011-03-17
EP1603553B9 (en) 2012-06-20
PT1603553E (pt) 2012-02-03
CA2519432A1 (en) 2004-09-30
MXPA05009848A (es) 2005-12-06
AU2004222434A1 (en) 2004-09-30
US20040225018A1 (en) 2004-11-11
HK1084882A1 (en) 2006-08-11
WO2004082593A3 (en) 2005-02-24
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