ATE526022T1 - Stabilisierte zusammenstellungen die benzimidazole enthalten - Google Patents

Stabilisierte zusammenstellungen die benzimidazole enthalten

Info

Publication number
ATE526022T1
ATE526022T1 AT99913726T AT99913726T ATE526022T1 AT E526022 T1 ATE526022 T1 AT E526022T1 AT 99913726 T AT99913726 T AT 99913726T AT 99913726 T AT99913726 T AT 99913726T AT E526022 T1 ATE526022 T1 AT E526022T1
Authority
AT
Austria
Prior art keywords
compositions containing
stabilized compositions
benzimidazole
type compounds
containing benzimidazoles
Prior art date
Application number
AT99913726T
Other languages
English (en)
Inventor
Koji Ukai
Masaki Ichikawa
Takashi Kato
Yukiko Sugaya
Yasuyuki Suzuki
Shigeru Aoki
Akira Kato
Masao Kawamura
Satoshi Fujioka
Original Assignee
Eisai R&D Man Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai R&D Man Co Ltd filed Critical Eisai R&D Man Co Ltd
Application granted granted Critical
Publication of ATE526022T1 publication Critical patent/ATE526022T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
AT99913726T 1998-04-20 1999-04-20 Stabilisierte zusammenstellungen die benzimidazole enthalten ATE526022T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP10928898 1998-04-20
PCT/JP1999/002098 WO1999053918A1 (fr) 1998-04-20 1999-04-20 Compositions stabilisees contenant des composes du type benzimidazole

Publications (1)

Publication Number Publication Date
ATE526022T1 true ATE526022T1 (de) 2011-10-15

Family

ID=14506385

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99913726T ATE526022T1 (de) 1998-04-20 1999-04-20 Stabilisierte zusammenstellungen die benzimidazole enthalten

Country Status (8)

Country Link
US (2) US20020039597A1 (de)
EP (1) EP1004305B1 (de)
KR (1) KR100627614B1 (de)
CN (1) CN1141097C (de)
AT (1) ATE526022T1 (de)
CA (1) CA2298823C (de)
ES (1) ES2373864T3 (de)
WO (1) WO1999053918A1 (de)

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US5840737A (en) 1996-01-04 1998-11-24 The Curators Of The University Of Missouri Omeprazole solution and method for using same
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US8906940B2 (en) 2004-05-25 2014-12-09 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
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CN102186474A (zh) * 2008-08-14 2011-09-14 杏林制药株式会社 稳定的医药组合物
KR101328383B1 (ko) * 2009-08-27 2013-11-13 한림제약(주) 유럽종 포도의 씨 추출물을 함유하는 경구용 정제
SI3158991T1 (sl) 2010-01-28 2021-10-29 Eagle Pharmaceuticals Inc Formulacije bendamustina
ES2943668T3 (es) 2012-03-20 2023-06-15 Eagle Pharmaceuticals Inc Composiciones líquidas de bendamustina para su uso en un método para tratar afecciones que responden a la bendamustina en pacientes que requieren volúmenes reducidos para administración
FI2827862T3 (fi) 2012-03-20 2024-02-13 Eagle Pharmaceuticals Inc Bendamustiinin formulaatioita
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Also Published As

Publication number Publication date
CA2298823A1 (en) 1999-10-28
KR20010013994A (ko) 2001-02-26
CN1275079A (zh) 2000-11-29
KR100627614B1 (ko) 2006-09-25
CA2298823C (en) 2011-06-07
WO1999053918A1 (fr) 1999-10-28
ES2373864T3 (es) 2012-02-09
CN1141097C (zh) 2004-03-10
US20020039597A1 (en) 2002-04-04
EP1004305A1 (de) 2000-05-31
EP1004305A4 (de) 2009-01-21
US20050042285A1 (en) 2005-02-24
EP1004305B1 (de) 2011-09-28

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