BR0109542A - Derivados de imidazopirina alquilados - Google Patents

Derivados de imidazopirina alquilados

Info

Publication number
BR0109542A
BR0109542A BR0109542-0A BR0109542A BR0109542A BR 0109542 A BR0109542 A BR 0109542A BR 0109542 A BR0109542 A BR 0109542A BR 0109542 A BR0109542 A BR 0109542A
Authority
BR
Brazil
Prior art keywords
alkylated
derivatives
imidazopyrine
substituents
prevention
Prior art date
Application number
BR0109542-0A
Other languages
English (en)
Inventor
Wolfgang-Alexander Simon
Stefan Postius
Wolfgang Kromer
Joerg Senn-Bilfinger
Wilm Buhr
Original Assignee
Altana Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Altana Pharma Ag filed Critical Altana Pharma Ag
Publication of BR0109542A publication Critical patent/BR0109542A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14—Ortho-condensed systems
    • C07D491/147—Ortho-condensed systems the condensed system containing one ring with oxygen as ring hetero atom and two rings with nitrogen as ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14—Ortho-condensed systems

Abstract

"DERIVADOS DE IMIDAZOPIRIDINA ALQUILADOS". Os compostos de fórmula (1), em que os substituintes têm os significados mencionados na descrição, são adequados para a prevenção e o tratamento de doenças gastrointestinais.
BR0109542-0A 2000-03-29 2001-03-28 Derivados de imidazopirina alquilados BR0109542A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00106696 2000-03-29
PCT/EP2001/003507 WO2001072754A1 (en) 2000-03-29 2001-03-28 Alkylated imidazopyridine derivatives

Publications (1)

Publication Number Publication Date
BR0109542A true BR0109542A (pt) 2003-06-10

Family

ID=8168272

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0109542-0A BR0109542A (pt) 2000-03-29 2001-03-28 Derivados de imidazopirina alquilados

Country Status (24)

Country Link
US (1) US6916825B2 (pt)
EP (1) EP1313739B1 (pt)
JP (1) JP2003528876A (pt)
KR (1) KR100823762B1 (pt)
CN (1) CN1213049C (pt)
AT (1) ATE332302T1 (pt)
AU (1) AU783764B2 (pt)
BR (1) BR0109542A (pt)
CA (1) CA2404460A1 (pt)
CZ (1) CZ20023116A3 (pt)
DE (1) DE60121345T2 (pt)
EA (1) EA005215B1 (pt)
ES (1) ES2267737T3 (pt)
HK (1) HK1056173A1 (pt)
HR (1) HRP20020853A2 (pt)
HU (1) HUP0300578A3 (pt)
IL (1) IL151201A0 (pt)
MX (1) MXPA02009552A (pt)
NO (1) NO20024597L (pt)
NZ (1) NZ520835A (pt)
PL (1) PL357811A1 (pt)
SK (1) SK13872002A3 (pt)
WO (1) WO2001072754A1 (pt)
ZA (1) ZA200207636B (pt)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2404474A1 (en) * 2000-03-29 2001-10-04 Altana Pharma Ag Prodrugs of imidazopyridine derivatives
ATE381568T1 (de) * 2000-03-29 2008-01-15 Nycomed Gmbh Pyrano(2,3-c)imidazo(1,2-a)pyridin-derivate zur behandlung von gastrointestinalen erkrankungen
EA008151B1 (ru) 2000-10-25 2007-04-27 Алтана Фарма Аг Полизамещенные имидазопиридины в качестве ингибиторов желудочной секреции
HUP0400380A3 (en) * 2001-08-03 2007-05-29 Altana Pharma Ag Alkyl-substituted imidazopyridines for the treatment of gastrointestinal disorders and pharmaceuticals containing them
DE10145457A1 (de) * 2001-09-14 2003-04-03 Basf Ag Substituierte Imidazo[1,2-a]-5,6,7,8-tetrahydropyridin-8-one, Verfahren zu ihrer Herstellung, sowie deren Verwendung zur Herstellung von Imidazo[1,2,-a]pyridinen
NZ535227A (en) 2002-02-15 2006-03-31 Altana Pharma Ag Tricyclic n-acyl compounds
BR0316201A (pt) 2002-11-19 2005-10-04 Altana Pharma Ag Imidazopiridinas 8-substituìdas
EA010107B1 (ru) * 2002-12-20 2008-06-30 Алтана Фарма Аг Силиловые простые эфиры
MXPA05008490A (es) * 2003-02-17 2005-10-18 Altana Pharma Ag Combinaciones que contienen imidazopiridinas y su uso en el tratamiento de enfermedades gastrointestinales inflamatorias.
AR044129A1 (es) 2003-05-06 2005-08-24 Altana Pharma Ag Compuestos intermedios de imidazopiridina. proceso de preparacion.
US20080280944A1 (en) 2003-11-03 2008-11-13 Paula Fernstrom Imidazo[1,2-A]Pyridine Derivatives For The Treatment Of Silent Gastro-Esophageal Reflux
EP1697358A1 (en) 2003-12-19 2006-09-06 Altana Pharma AG Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives
US7215655B2 (en) * 2004-01-09 2007-05-08 Interdigital Technology Corporation Transport format combination selection in a wireless transmit/receive unit
NZ549011A (en) * 2004-02-17 2009-04-30 Altana Pharma Ag Tricyclic imidazopyridines and intermediates for the synthesis thereof
AU2005291284A1 (en) * 2004-10-01 2006-04-13 Altana Pharma Ag Substituted tricyclic benzimidazoles
WO2007039464A1 (en) * 2005-09-22 2007-04-12 Nycomed Gmbh Isotopically substituted imidazopyridine derivatives for the treatment of gastrointestinal disorders
WO2008058990A1 (en) * 2006-11-16 2008-05-22 Nycomed Gmbh 7,7-disubstituted pyrano-[2,3-c]-imidazo-[1,2-a]-pyridine derivatives and their use as gastric acid secretion inhibitors
AU2009249069A1 (en) 2008-05-20 2009-11-26 Neurogesx, Inc. Carbonate prodrugs and methods of using the same
KR101698028B1 (ko) 2008-05-20 2017-01-26 노이로제스엑스, 인코포레이티드 수용성 아세트아미노펜 유사체
CA2969597C (en) * 2014-12-06 2023-10-24 Intra-Cellular Therapies, Inc. 1h-pyrazolo[4,3-c][1,5]naphthyridin-4(5h)-one compounds and their use as pde2 inhibitors

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4468400A (en) * 1982-12-20 1984-08-28 Schering Corporation Antiulcer tricyclic imidazo [1,2-a]pyridines
SE9401197D0 (sv) * 1994-04-11 1994-04-11 Astra Ab Active compounds
IL131407A0 (en) * 1997-03-24 2001-01-28 Byk Gulden Lomberg Chem Fab Tetrahydropyrido compounds medicaments containing the same and the use thereof
EP0984969B1 (en) * 1997-05-28 2008-07-09 Nycomed GmbH Fused dihydropyrans
HUP0001555A3 (en) * 1997-10-30 2001-01-29 Altana Pharma Ag Tetrahydro-imidazo-naphthyridine derivatives, pharmaceutical compositions thereof and process for their preparation
CA2404474A1 (en) * 2000-03-29 2001-10-04 Altana Pharma Ag Prodrugs of imidazopyridine derivatives
ATE381568T1 (de) * 2000-03-29 2008-01-15 Nycomed Gmbh Pyrano(2,3-c)imidazo(1,2-a)pyridin-derivate zur behandlung von gastrointestinalen erkrankungen
AU783724B2 (en) * 2000-03-29 2005-12-01 Altana Pharma Ag Tricyclic imidazopyridines

Also Published As

Publication number Publication date
ATE332302T1 (de) 2006-07-15
HUP0300578A3 (en) 2009-01-28
US20030158193A1 (en) 2003-08-21
CN1213049C (zh) 2005-08-03
CN1422274A (zh) 2003-06-04
HUP0300578A2 (hu) 2003-07-28
SK13872002A3 (sk) 2003-02-04
HK1056173A1 (en) 2004-02-06
WO2001072754A1 (en) 2001-10-04
EP1313739A1 (en) 2003-05-28
KR100823762B1 (ko) 2008-04-21
HRP20020853A2 (en) 2005-02-28
CZ20023116A3 (cs) 2003-01-15
WO2001072754A9 (en) 2004-05-06
DE60121345D1 (de) 2006-08-17
WO2001072754A8 (en) 2003-02-13
NZ520835A (en) 2004-05-28
ES2267737T3 (es) 2007-03-16
NO20024597D0 (no) 2002-09-25
EP1313739B1 (en) 2006-07-05
US6916825B2 (en) 2005-07-12
MXPA02009552A (es) 2004-05-14
DE60121345T2 (de) 2007-07-19
KR20030015221A (ko) 2003-02-20
EA005215B1 (ru) 2004-12-30
ZA200207636B (en) 2003-04-04
CA2404460A1 (en) 2001-10-04
IL151201A0 (en) 2003-04-10
NO20024597L (no) 2002-09-25
EA200200876A1 (ru) 2003-04-24
PL357811A1 (en) 2004-07-26
JP2003528876A (ja) 2003-09-30
AU783764B2 (en) 2005-12-01
AU4422501A (en) 2001-10-08

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.