ATE460398T1 - Verwendung von omega-carboxyaryl-substituierten diphenylharnstoffen als raf-kinase-inhibitoren - Google Patents

Verwendung von omega-carboxyaryl-substituierten diphenylharnstoffen als raf-kinase-inhibitoren

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Publication number
ATE460398T1
ATE460398T1 AT05028442T AT05028442T ATE460398T1 AT E460398 T1 ATE460398 T1 AT E460398T1 AT 05028442 T AT05028442 T AT 05028442T AT 05028442 T AT05028442 T AT 05028442T AT E460398 T1 ATE460398 T1 AT E460398T1
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AT
Austria
Prior art keywords
ureases
carboxyaryl
omega
kinase inhibitors
raf kinase
Prior art date
Application number
AT05028442T
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English (en)
Inventor
Bernd Riedl
Jacques Dumas
Uday Khire
Timothy Lowinger
William Scott
Roger Smith
Jill Wood
Mary-Katherine Monahan
Reina Natero
Joel Renick
Robert Sibley
Original Assignee
Bayer Healthcare Llc
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Application filed by Bayer Healthcare Llc filed Critical Bayer Healthcare Llc
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Publication of ATE460398T1 publication Critical patent/ATE460398T1/de

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    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
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    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
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AT05028442T 1999-01-13 2000-01-12 Verwendung von omega-carboxyaryl-substituierten diphenylharnstoffen als raf-kinase-inhibitoren ATE460398T1 (de)

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