ATE334987T1 - Artemisininderivate (endoperoxide) mit wirkung gegen parasiten - Google Patents

Artemisininderivate (endoperoxide) mit wirkung gegen parasiten

Info

Publication number
ATE334987T1
ATE334987T1 AT03743815T AT03743815T ATE334987T1 AT E334987 T1 ATE334987 T1 AT E334987T1 AT 03743815 T AT03743815 T AT 03743815T AT 03743815 T AT03743815 T AT 03743815T AT E334987 T1 ATE334987 T1 AT E334987T1
Authority
AT
Austria
Prior art keywords
endoperoxides
parasite effect
artemisinine
derivatives
artemisinine derivatives
Prior art date
Application number
AT03743815T
Other languages
English (en)
Inventor
Richard K Haynes
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Application granted granted Critical
Publication of ATE334987T1 publication Critical patent/ATE334987T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/12Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains three hetero rings
    • C07D493/20Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/12Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains three hetero rings
    • C07D493/18Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06Antimalarials

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AT03743815T 2002-03-08 2003-02-24 Artemisininderivate (endoperoxide) mit wirkung gegen parasiten ATE334987T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP02005233 2002-03-08

Publications (1)

Publication Number Publication Date
ATE334987T1 true ATE334987T1 (de) 2006-08-15

Family

ID=27798779

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03743815T ATE334987T1 (de) 2002-03-08 2003-02-24 Artemisininderivate (endoperoxide) mit wirkung gegen parasiten

Country Status (21)

Country Link
US (1) US20050119232A1 (de)
EP (1) EP1485389B1 (de)
JP (1) JP2005526073A (de)
KR (1) KR20040104493A (de)
CN (1) CN1649874A (de)
AR (1) AR038842A1 (de)
AT (1) ATE334987T1 (de)
AU (1) AU2003215584A1 (de)
BR (1) BR0308291A (de)
CA (1) CA2478600A1 (de)
DE (1) DE60307239D1 (de)
HR (1) HRP20040927A2 (de)
IL (1) IL163870A0 (de)
MX (1) MXPA04008638A (de)
NZ (1) NZ535084A (de)
PL (1) PL372341A1 (de)
RU (1) RU2004130284A (de)
TW (1) TW200400964A (de)
WO (1) WO2003076446A1 (de)
YU (1) YU79304A (de)
ZA (1) ZA200407102B (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102004027871B3 (de) * 2004-06-08 2006-03-16 Lanxess Deutschland Gmbh Verfahren zur Herstellung von 10α-[4'-(S,S-Dioxothiomorpholin-1'-yl)]-10-desoxo-10-dihydroartemisinin
EP1714967A1 (de) * 2005-04-22 2006-10-25 Bayer HealthCare AG Antiparasitär wirkende Artemisinin Derivate
CN101282722B (zh) * 2005-10-20 2011-03-30 埃皮法姆有限责任公司 用青蒿素及其衍生物治疗和预防良性色素斑(痣)的制药用途
WO2008127381A2 (en) * 2006-10-20 2008-10-23 Johns Hopkins University Artemisinin derivatives
EP2219643B1 (de) * 2007-11-15 2012-05-16 Novartis AG Anthelmintische paste mit praziquantel, einem makrolid-lacton, cyclodextrin und einem verdickungsmittel
US8815942B2 (en) 2010-10-20 2014-08-26 The Royal Institution For The Advancement Of Learning/Mcgill University Combination therapy and uses thereof for treatment and prevention of parasitic infection and disease
CN102010422B (zh) * 2010-11-23 2014-11-26 沈阳药科大学 含有胍基的青蒿素类衍生物及其应用
US8232417B1 (en) 2010-12-01 2012-07-31 Bioderm Research Artemisinin derivatives with natural amino acids, peptides, and amino sugars for skin imperfections and infection in mammals
CN103183682B (zh) * 2011-12-31 2015-10-14 沈阳药科大学 C-10位脲基取代的青蒿素衍生物及其制备方法和用途
ES2650962T3 (es) 2012-04-18 2018-01-23 The Hong Kong University Of Science And Technology Métodos y composiciones para el tratamiento de infecciones virales

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5726203A (en) * 1993-07-19 1998-03-10 Li; Zelin Qinghaosu derivatives against AIDS
EP0974594A1 (de) * 1998-07-14 2000-01-26 The Hong Kong University of Science & Technology Artemisininderivate als Mittel gegen Infektionen
TR200100073T2 (tr) * 1998-07-14 2001-05-21 Bayer Aktiengeselkschaft Antiparazitik artemisinin türevleri (endoperoksitler)

Also Published As

Publication number Publication date
CN1649874A (zh) 2005-08-03
BR0308291A (pt) 2005-01-11
MXPA04008638A (es) 2005-04-19
YU79304A (sh) 2006-08-17
CA2478600A1 (en) 2003-09-18
TW200400964A (en) 2004-01-16
IL163870A0 (en) 2005-12-18
HRP20040927A2 (en) 2005-06-30
PL372341A1 (en) 2005-07-11
JP2005526073A (ja) 2005-09-02
WO2003076446A8 (en) 2004-10-07
DE60307239D1 (de) 2006-09-14
AU2003215584A1 (en) 2003-09-22
KR20040104493A (ko) 2004-12-10
WO2003076446A1 (en) 2003-09-18
EP1485389A1 (de) 2004-12-15
ZA200407102B (en) 2005-09-06
RU2004130284A (ru) 2005-05-10
AR038842A1 (es) 2005-01-26
EP1485389B1 (de) 2006-08-02
US20050119232A1 (en) 2005-06-02
NZ535084A (en) 2006-05-26

Similar Documents

Publication Publication Date Title
ATE478870T1 (de) Spiroindolinpiperidinderivate
ATE460418T1 (de) Heterocyclocarboxamidderivate
ATE450506T1 (de) Indol-3-schwefelderivate
ATE467631T1 (de) Chinuclidinamidderivate
ATE438644T1 (de) Chinazolinderivate
IS7720A (is) Píperidín-N-oxíð-afleiður
DK2248807T3 (da) N-Phenyl-2-pyrimidinaminderivater
NO20054224D0 (no) Nye 2-pyridinkarboksamidderivater
ATE340782T1 (de) Piperidinbenzolsulfonamidderivate
DK1682493T3 (da) Amidoacetonitrilderivater
NO20043696L (no) Gamma-sekretaseinhibitorer
DE602004004553D1 (de) Chinazolinderivate
DE602004022180D1 (de) Chinazolinderivate
DK1606277T3 (da) Imidazol-4-yl-ethynyl-pyridinderivater
IS2656B (is) Nýjar besímídasólafleiður
ATE335729T1 (de) 3h-chinazoline -4-on derivaten
ATE354365T1 (de) N-thiazol-2-yl-benzamid-derivate
ATE423771T1 (de) Tetrahydrochinolinderivate
ATE334987T1 (de) Artemisininderivate (endoperoxide) mit wirkung gegen parasiten
DK1706373T3 (da) Amidoacetonitrilderivater
DE60315984D1 (de) Substituierte benzisoxazolsulfonamide mit breitbändiger hiv-protease hemmender wirkung
IS8045A (is) Púrín-6-ón-afleiður
DE50306277D1 (de) 4-alkyl-/4-alkenyl-/4-alkinylmethyl/-1-arylcyclohexylamin-derivate
DE50311770D1 (de) Oberfräse
DE50303274D1 (de) Doppeltwirkender Arbeitszylinder

Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties