ATE311903T1 - Verfahren, zusammensetzungen und kits zur erhöhung der oralen bioverfügbarkeit von pharmazeutika - Google Patents

Verfahren, zusammensetzungen und kits zur erhöhung der oralen bioverfügbarkeit von pharmazeutika

Info

Publication number
ATE311903T1
ATE311903T1 AT96943268T AT96943268T ATE311903T1 AT E311903 T1 ATE311903 T1 AT E311903T1 AT 96943268 T AT96943268 T AT 96943268T AT 96943268 T AT96943268 T AT 96943268T AT E311903 T1 ATE311903 T1 AT E311903T1
Authority
AT
Austria
Prior art keywords
oral
agent
target
bioavailability
enhancing
Prior art date
Application number
AT96943268T
Other languages
English (en)
Inventor
Samuel Broder
Kenneth L Duchin
Sami Selim
Original Assignee
Ivax Research Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/608,776 external-priority patent/US5968972A/en
Application filed by Ivax Research Inc filed Critical Ivax Research Inc
Application granted granted Critical
Publication of ATE311903T1 publication Critical patent/ATE311903T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13—Cyclosporins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Virology (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT96943268T 1995-10-26 1996-10-24 Verfahren, zusammensetzungen und kits zur erhöhung der oralen bioverfügbarkeit von pharmazeutika ATE311903T1 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US707195P 1995-10-26 1995-10-26
US08/608,776 US5968972A (en) 1995-10-26 1996-02-29 Method for increasing the oral bioactivity of pharmaceutical agents
US08/733,142 US6245805B1 (en) 1995-10-26 1996-10-16 Method, compositions and kits for increasing the oral bioavailability of pharmaceutical agents
PCT/IB1996/001485 WO1997015269A2 (en) 1995-10-26 1996-10-24 Method, compositions and kits for increasing the oral bioavailability of pharmaceutical agents

Publications (1)

Publication Number Publication Date
ATE311903T1 true ATE311903T1 (de) 2005-12-15

Family

ID=27358262

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96943268T ATE311903T1 (de) 1995-10-26 1996-10-24 Verfahren, zusammensetzungen und kits zur erhöhung der oralen bioverfügbarkeit von pharmazeutika

Country Status (22)

Country Link
US (6) US6245805B1 (de)
EP (1) EP0794794B1 (de)
JP (1) JP3361102B2 (de)
CN (2) CN100335123C (de)
AT (1) ATE311903T1 (de)
AU (1) AU698142B2 (de)
BR (1) BR9607066A (de)
CA (1) CA2205534A1 (de)
CZ (1) CZ202897A3 (de)
DE (2) DE794794T1 (de)
DK (1) DK0794794T3 (de)
ES (1) ES2109899T3 (de)
HK (1) HK1001960A1 (de)
HU (1) HUP9900457A3 (de)
IL (1) IL121160A0 (de)
MX (1) MX9704629A (de)
NO (1) NO321091B1 (de)
NZ (1) NZ324801A (de)
PL (2) PL188281B1 (de)
RU (1) RU2217135C2 (de)
SK (1) SK85997A3 (de)
WO (1) WO1997015269A2 (de)

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GB9718903D0 (en) 1997-09-05 1997-11-12 Glaxo Group Ltd Method,compositions and kits for increasing the oral bioavailability of pharmaceutical agents
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US20030109448A1 (en) * 2001-11-07 2003-06-12 Crowley Kathleen S. Methods of promoting uptake and nuclear accumulation of polyamides in eukaryotic cells
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US20060014677A1 (en) * 2004-07-19 2006-01-19 Isotechnika International Inc. Method for maximizing efficacy and predicting and minimizing toxicity of calcineurin inhibitor compounds
US20070087977A1 (en) * 2004-11-16 2007-04-19 Wendye Robbins Methods and compositions for treating pain
AU2005307772B2 (en) * 2004-11-16 2010-06-10 Limerick Biopharma, Inc. Methods and compositions for treating pain
US7745400B2 (en) * 2005-10-14 2010-06-29 Gregg Feinerman Prevention and treatment of ocular side effects with a cyclosporin
EP2153842B1 (de) * 2005-10-14 2016-04-13 Allergan, Inc. Prävention von mit arzneimitteln in zusammenhang stehenden keratokonjunctivitis mit cyclosporin
US9839667B2 (en) 2005-10-14 2017-12-12 Allergan, Inc. Prevention and treatment of ocular side effects with a cyclosporin
KR20100023862A (ko) * 2007-06-22 2010-03-04 싸이도우스 엘엘씨. 트윈 80을 함유하지 않은 도세탁셀의 용해 제제
US20090111736A1 (en) * 2007-10-29 2009-04-30 Sri International Orally-Absorbed Solid Dose Formulation for Vancomycin
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US8541465B2 (en) * 2009-10-19 2013-09-24 Scidose, Llc Docetaxel formulations with lipoic acid and/or dihydrolipoic acid
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US20110092579A1 (en) * 2009-10-19 2011-04-21 Scidose Llc Solubilized formulation of docetaxel
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US20120295932A1 (en) * 2011-05-17 2012-11-22 Western Connecticut Health Network, Inc. Method for the treatment of cancer
JO3685B1 (ar) 2012-10-01 2020-08-27 Teikoku Pharma Usa Inc صيغ التشتيت الجسيمي للتاكسين غير المائي وطرق استخدامها
TWI752750B (zh) 2015-09-30 2022-01-11 香港商慧源香港創新有限公司 口服紫杉烷組合物及方法
CN107843966B (zh) 2016-09-18 2021-05-04 中芯国际集成电路制造(上海)有限公司 用于装配微透镜阵列组件的方法和系统
CN106822085B (zh) * 2016-12-17 2020-03-17 浙江省人民医院 表达trail的溶瘤腺病毒联合槲皮素在抑制肝癌癌细胞增殖中的用途
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Also Published As

Publication number Publication date
US6245805B1 (en) 2001-06-12
PL192544B1 (pl) 2006-11-30
CN100335123C (zh) 2007-09-05
NO972968L (no) 1997-07-23
EP0794794A1 (de) 1997-09-17
ES2109899T3 (es) 2006-05-01
ES2109899T1 (es) 1998-02-01
JP3361102B2 (ja) 2003-01-07
US20070060635A1 (en) 2007-03-15
US20040176439A1 (en) 2004-09-09
CA2205534A1 (en) 1997-05-01
EP0794794B1 (de) 2005-12-07
IL121160A0 (en) 1997-11-20
JPH10509741A (ja) 1998-09-22
RU2217135C2 (ru) 2003-11-27
NZ324801A (en) 1999-05-28
CN1490048A (zh) 2004-04-21
CZ202897A3 (cs) 1998-03-18
HUP9900457A2 (hu) 1999-06-28
US20050238634A1 (en) 2005-10-27
HK1001960A1 (en) 1998-07-24
MX9704629A (es) 1997-09-30
PL321791A1 (en) 1997-12-22
EP0794794A4 (de) 2000-03-01
US20020058616A1 (en) 2002-05-16
DE69636531T2 (de) 2006-12-07
PL188281B1 (pl) 2005-01-31
SK85997A3 (en) 1998-06-03
HUP9900457A3 (en) 2001-04-28
DE69636531D1 (de) 2006-10-19
AU1205697A (en) 1997-05-15
BR9607066A (pt) 2002-12-10
AU698142B2 (en) 1998-10-22
NO321091B1 (no) 2006-03-13
WO1997015269A3 (en) 1997-07-31
US20030069301A1 (en) 2003-04-10
CN1173817A (zh) 1998-02-18
NO972968D0 (no) 1997-06-25
US6610735B2 (en) 2003-08-26
US6818615B2 (en) 2004-11-16
US7041640B2 (en) 2006-05-09
WO1997015269A2 (en) 1997-05-01
DE794794T1 (de) 1998-03-12
DK0794794T3 (da) 2006-04-18
CN1119146C (zh) 2003-08-27

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